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NCGC00262691-01 (CID 3201893) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Inactive(1)
 
 
Inconclusive(1)
 
 
Top Targets:
PTZ00435(3)
 
 
 
 
BioAssay Types:
Confirmatory(4)
 
 
 
 
BioActivity Types:
Potency(3)
 
 
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134958860]
Potency 0.903qHTS for Inhibitors of mutant isocitrate dehydrogenase 1 (IDH1): confirmation assay for probe SAR [AID624023, Type: confirmatory]isocitrate dehydrogenase 1, partial [Homo sapiens] [gi:89573979]
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2
[SID163338939]
IC50 1.8Inhibition of IDH1 R132H mutant using alpha-ketoglutarate as substrate after 60 mins by resazurin-based fluorimetric analysis [AID704657, Type: confirmatory]
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3
[SID134958860]
Potency qHTS for Inhibitors of mutant isocitrate dehydrogenase 1 (IDH1): WT assay for probe SAR [AID624021, Type: confirmatory]isocitrate dehydrogenase 1, partial [Homo sapiens] [gi:89573979]
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4
[SID134958860]
Potency 1.189qHTS for Inhibitors of mutant isocitrate dehydrogenase 1 (IDH1): 2HG production assay for probe SAR [AID624019, Type: confirmatory]isocitrate dehydrogenase 1, partial [Homo sapiens] [gi:89573979]
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