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STK225779 (CID 3164412) - Compound BioActivity Data
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BioActivity Outcomes:
Active(9)
 
 
Inactive(534)
 
 
Inconclusive(3)
 
 
Unspecified(1)
 
 
Top Targets:
7TM GPCR Srx(21)
 
 
7TM GPCR Srsx(20)
 
 
 
TRP 2(5)
 
 
CAP ED(5)
 
 
alkPPc(4)
 
 
BioAssay Types:
Screening(365)
 
 
 
Confirmatory(163)
 
 
 
 
 
Literature(11)
 
 
BioActivity Types:
Potency(121)
 
 
 
 
IC50(28)
 
 
EC50(12)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 498    Data Row: 547   Total Pages: 28   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID126920244]
EC50_MICROM 0.00523Counter screen for HTS for Beta-2AR agonists with FAP-tagged GPR32 with Powderset2 [AID651729, Type: confirmatory]G protein-coupled receptor 32 [Homo sapiens] [gi:119592304]
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2
[SID126920244]
EC50_MICROM 0.00746Counter screen for HTS for Beta-2AR agonists with FAP-tagged human CCR5 with Powderset2 [AID651728, Type: confirmatory]CCR5 [Homo sapiens] [gi:289466095]
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3
[SID152259017]
EC50_MICROM 0.0108Counter screen for HTS for Beta-2AR agonists with FAP-tagged human CCR5 with Powderset5 [AID651913, Type: confirmatory]CCR5 [Homo sapiens] [gi:289466095]
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4
[SID49727953]
EC50_MICROM 0.0396Dose response for HTS for Beta-2AR agonists via FAP method from CP1 [AID588763, Type: confirmatory]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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5
[SID126920244]
EC50_MICROM 0.357Dose response for HTS for Beta-2AR agonists via FAP method from Powderset2 [AID623882, Type: confirmatory]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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6
[SID49727953]
HTS for Beta-2AR agonists via FAP method [AID504454, Type: screening]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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7
[SID126920244]
Evaluation of reversibility of compound binding to AM2.2-beta2AR cells with Powder Set 3and4 [AID651936, Type: other]single chain variable fragment antibody type HL1.1-TO1 [synthetic construct] [gi:163932448]
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8
[SID126920244]
Fluorogen/soluble FAP binding competition assay [AID651938, Type: other]single chain variable fragment antibody type HL1.1-TO1 [synthetic construct] [gi:163932448]
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9
[SID49727953]
HTS for Beta-2AR agonists via FAP method, Single Point, Cherry Pick 1 [AID540358, Type: other]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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10
[SID49727953]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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11
[SID49727953]
Potency qHTS for Stage-Specific Inhibitors of Vaccinia Orthopoxvirus: mCherry Reporter Primary qHTS [AID720579, Type: confirmatory]67.9K protein [Vaccinia virus] [gi:222762]
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12
[SID49727953]
Potency qHTS for Stage-Specific Inhibitors of Vaccinia Orthopoxvirus: Venus Reporter Primary qHTS [AID720580, Type: confirmatory]67.9K protein [Vaccinia virus] [gi:222762]
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13
[SID49727953]
Potency qHTS for inhibitors of binding or entry into cells for Marburg Virus [AID540276, Type: confirmatory]gene 4 small orf - Marburg virus [gi:420597]
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14
[SID49727953]
Multiplex HTS Screen of TOR pathway GFP-fusion proteins in Saccharomyes cerevisiae_specifically_ LAP4_MLPCN. [AID2023, Type: screening]LAP4 [Saccharomyces cerevisiae] [gi:486173]
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15
[SID49727953]
Primary cell-based high-throughput screening assay for identification of compounds that protect hERG from block by proarrhythmic agents [AID1511, Type: screening]putative potassium channel subunit [Homo sapiens] [gi:487738]
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16
[SID49727953]
Potency qHTS Assay for Inhibitors and Activators of N370S glucocerebrosidase as a Potential Chaperone Treatment of Gaucher Disease [AID2101, Type: confirmatory]glucocerebrosidase [Homo sapiens] [gi:496369]
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17
[SID49727953]
Primary biochemical high throughput screening assay to identify inhibitors of BCL2-related protein, long isoform (BCLXL). [AID2129, Type: screening]bcl-xL [Homo sapiens] [gi:510901]
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18
[SID49727953]
Multiplex HTS Screen of TOR pathway GFP-fusion proteins in Saccharomyes cerevisiae_specifically_ RPL19A_MLPCN. [AID2025, Type: screening]RPL19A [Saccharomyces cerevisiae] [gi:536029]
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19
[SID49727953]
Potency Activators of T cell receptors: qHTS campaign [AID504894, Type: confirmatory]T cell receptor [Homo sapiens] [gi:553160]
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20
[SID49727953]
Potency qHTS of alpha-syn Inhibitors [AID652106, Type: confirmatory]Alpha-synuclein [gi:586067]
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