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benzophenone (CID 3102) - Compound BioActivity Data
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BioActivity Outcomes:
Active(10)
 
 
Inactive(932)
 
 
Inconclusive(26)
 
 
Unspecified(23)
 
 
Top Targets:
NR LBD PPAR(34)
 
 
 
NR LBD AR(25)
 
 
 
 
NR LBD ER(25)
 
 
 
 
7TM GPCR Srx(19)
 
 
NR LBD TR(19)
 
 
 
BioAssay Types:
Confirmatory(530)
 
 
 
 
 
Screening(316)
 
 
 
Summary(72)
 
 
 
Literature(42)
 
 
 
 
 
BioActivity Types:
Potency(534)
 
 
 
 
 
IC50(17)
 
 
 
 
 
Ki(5)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 683    Data Row: 991   Total Pages: 50   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID46391755]
IC50 3.6Experimentally measured binding affinity data (IC50) for protein-ligand complexes derived from PDB [AID977608, Type: Literature]Chain B, Porcine Odorant Binding Protein Complexed With Diphenylmethanone [gi:12084616]
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2
[SID46391755]
IC50 3.6Experimentally measured binding affinity data (IC50) for protein-ligand complexes derived from PDB [AID977608, Type: Literature]Chain B, Porcine Odorant Binding Protein Complexed With Diphenylmethanone [gi:12084616]
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3
[SID17389587]
Potency 25.1189qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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4
[SID144207014]
Potency-Replicate_1 26.6032qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743040, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
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5
[SID144210378]
Potency-Replicate_1 30.6379qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line [AID743079, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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6
[SID46391755]
Experimentally measured binding affinity data derived from PDB [AID1811, Type: Literature]Chain A, Porcine Odorant Binding Protein Complexed With Diphenylmethanone [gi:12084615]
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7
[SID49816673]
uHTS Fluorescent Assay Using Nedd8 Protein Substrate for Identification of Inhibitors of Sentrin-Specific Protease 8 (SENP8) [AID602440, Type: screening]sentrin-specific protease 8 [Homo sapiens] [gi:262118306]
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8
[SID49816673]
Fluorescence-based biochemical high throughput primary assay to identify inhibitors of phospholipase C isozymes (PLC-beta3). [AID720704, Type: screening]Phospholipase C, beta 3 (phosphatidylinositol-specific) [Homo sapiens] [gi:148745659]
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9
[SID103300986]
Inhibition of apolipoprotein E production in human CCF-STTG1 cells at 10 uM after 24 hrs by ELISA relative to vehicle-treated control [AID684467, Type: Literature]
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10
[SID48415153]
DSSTox (EPAFHM) EPA Fathead Minnow Acute Toxicity [AID1188, Type: other]
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11
[SID103300986]
Ki 100Inhibition constant against rabbit liver carboxylesterase (rCE) using nitrophenyl acetate (o-NPA) as substrate [AID239167, Type: Literature]
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12
[SID103300986]
Ki 100Inhibition constant against human Acetylcholinesterase (hAcChE) using acetylthiocholine (AcTCh) as substrate [AID239122, Type: Literature]Acetylcholinesterase [gi:113037]
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13
[SID103300986]
Ki 100Inhibition constant against human Butyrylcholinesterase (hBuChE) using butyrylthiocholine (BuTCh) as substrate [AID239166, Type: Literature]Cholinesterase [gi:116353]
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14
[SID103300986]
Ki 100Inhibition constant against human liver carboxylesterase 1 (hCE1) using nitrophenyl acetate (o-NPA) as substrate [AID239197, Type: Literature]Liver carboxylesterase 1 [gi:119576]
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15
[SID103300986]
Ki 100Inhibition constant against human intestinal carboxylesterase 2 (hiCE) using nitrophenyl acetate (o-NPA) as substrate [AID239272, Type: Literature]Cocaine esterase [gi:46576349]
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16
[SID103300986]
IC50 128.825Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881) [AID255211, Type: Literature]
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17
[SID103300986]
IC50 288.8Inhibition of cathepsin B by spectrofluorimetry [AID351454, Type: Literature]
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18
[SID103300986]
IC50 1000Inhibition of human recombinant IDO expressed in Escherichia coli BL21 AI [AID443993, Type: Literature]Indoleamine 2,3-dioxygenase 1 [gi:123948]
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19
[SID103300986]
IC50 3465Inhibition of Carica papaya papain by spectrofluorimetry [AID351452, Type: Literature]Papain [gi:129614]
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20
[SID103300986]
IC50 3466Inhibition of trypsin by spectrofluorimetry [AID351453, Type: Literature]
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