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Coumaphos (CID 2871) - Compound BioActivity Data
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BioActivity Outcomes:
Active(44)
 
 
Inactive(563)
 
 
Inconclusive(116)
 
 
Unspecified(8)
 
 
Top Targets:
NR LBD PPAR(29)
 
 
 
NR LBD AR(23)
 
 
 
 
NR LBD ER(23)
 
 
 
7tm 4(20)
 
 
NR LBD VDR(16)
 
 
 
BioAssay Types:
Confirmatory(373)
 
 
 
 
 
Screening(179)
 
 
 
Literature(88)
 
 
 
 
 
Summary(72)
 
 
 
 
BioActivity Types:
Potency(423)
 
 
 
 
 
Ki(12)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 449    Data Row: 731   Total Pages: 37   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144211086]
AhR Potency (uM) 0.0432771qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway: Summary [AID743122, Type: summary]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
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2
[SID144209039]
AhR Potency (uM) 0.0654778qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway: Summary [AID743122, Type: summary]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
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3
[SID144209039]
Potency-Replicate_1 0.098qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway [AID743085, Type: confirmatory]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
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4
[SID144204842]
AhR Potency (uM) 0.438128qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway: Summary [AID743122, Type: summary]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
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5
[SID144204842]
Potency-Replicate_1 0.5956qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway [AID743085, Type: confirmatory]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
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6
[SID50107237]
Potency 1.7783qHTS assay for small molecule activators of the rat pregnane X receptor (rPXR) signaling pathway [AID651751, Type: confirmatory]pregnane X receptor [Rattus norvegicus] [gi:5702233]
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7
[SID50107237]
Potency-Replicate_1 1.7783qHTS assay for small molecule activators of the human pregnane X receptor (PXR) signaling pathway [AID720659, Type: confirmatory]pregnane X nuclear receptor [Homo sapiens] [gi:325495557]
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8
[SID26747703]
Potency 1.9953qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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9
[SID103558152]
Ki 2.23Inhibition of human recombinant carbonic anhydrase 6 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649885, Type: Literature]Carbonic anhydrase 6 [gi:116241278]
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10
[SID103558152]
Ki 3.41Inhibition of human recombinant carbonic anhydrase 5B preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649886, Type: Literature]Carbonic anhydrase 5B, mitochondrial [gi:8928041]
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11
[SID103558152]
Ki 4.14Inhibition of human recombinant carbonic anhydrase 14 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649880, Type: Literature]Carbonic anhydrase 14 [gi:8928036]
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12
[SID103558152]
Ki 4.23Inhibition of human recombinant carbonic anhydrase 13 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649881, Type: Literature]Carbonic anhydrase 13 [gi:30580350]
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13
[SID103558152]
Ki 4.62Inhibition of human recombinant carbonic anhydrase 3 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649889, Type: Literature]Carbonic anhydrase 3 [gi:134047703]
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14
[SID103558152]
Ki 4.68Inhibition of human recombinant carbonic anhydrase 7 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649884, Type: Literature]Carbonic anhydrase 7 [gi:1168744]
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15
[SID103558152]
Ki 5.09Inhibition of human recombinant carbonic anhydrase 5A preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649887, Type: Literature]Carbonic anhydrase 5A, mitochondrial [gi:461680]
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16
[SID103558152]
Ki 5.48Inhibition of human recombinant carbonic anhydrase 4 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649888, Type: Literature]Carbonic anhydrase 4 [gi:115465]
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17
[SID103558152]
Ki 6.41Inhibition of human recombinant carbonic anhydrase 9 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649883, Type: Literature]Carbonic anhydrase 9 [gi:83300925]
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18
[SID89854493]
Potency 6.5131qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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19
[SID26747703]
Potency 8.0875S16 Schwann cell PMP22 intronic element firefly luciferase assay [AID624032, Type: confirmatory]peripheral myelin protein 22 [Rattus norvegicus] [gi:8393992]
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20
[SID103558152]
Ki 9.52Inhibition of human recombinant carbonic anhydrase 12 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649882, Type: Literature]Carbonic anhydrase 12 [gi:5915866]
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