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Clomipramine (CID 2801) - Compound BioActivity Data
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BioActivity Outcomes:
Active(121)
 
 
Inactive(403)
 
 
Inconclusive(165)
 
 
Unspecified(1420)
 
 
Top Targets:
p450(39)
 
 
 
 
 
7TM GPCR Srx(28)
 
 
 
 
7TM GPCR Srsx(24)
 
 
 
 
HSD10-like SD..(12)
 
 
NR LBD GR(11)
 
 
 
 
BioAssay Types:
Confirmatory(554)
 
 
 
 
 
Literature(271)
 
 
 
 
 
Screening(24)
 
 
 
Summary(24)
 
 
 
 
BioActivity Types:
Potency(385)
 
 
 
 
 
IC50(168)
 
 
 
 
 
Ki(12)
 
 
 
EC50(2)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1807    Data Row: 2109   Total Pages: 106   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103164619]
IC50 4e-05Compound was tested for its inhibitory activity against Alpha-1 adrenergic receptor [AID36031, Type: Literature]
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2
[SID103164619]
IC50 8.8e-05DRUGMATRIX: Transporter, Serotonin (5-Hydroxytryptamine) (SERT) radioligand binding (ligand: [3H] Paroxetine) [AID625222, Type: confirmatory]Sodium-dependent serotonin transporter [gi:400630]
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3
[SID103164619]
IC50 0.0002Compound tested for its inhibitory activity against Histamine H1 receptor [AID87513, Type: Literature]
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4
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 1F [gi:398968]
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5
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 2B [gi:398970]
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6
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 2A [gi:112808]
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7
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 1A [gi:112812]
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8
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 1B [gi:112815]
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9
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 2C [gi:112817]
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10
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 1D [gi:112820]
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11
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 7 [gi:461440]
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12
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 5A [gi:543729]
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13
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 5B [gi:543730]
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14
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 6 [gi:1168221]
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15
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 3A [gi:1168223]
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16
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 4 [gi:2494928]
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17
[SID103164619]
IC50 0.005Compound was tested for its inhibitory activity against 5-hydroxytryptamine receptor [AID6418, Type: Literature]5-hydroxytryptamine receptor 3B [gi:81868595]
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18
[SID103164619]
Ki 0.0083Binding affinity towards 5-hydroxytryptamine 2 receptor [AID5241, Type: Literature]
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19
[SID103164619]
IC50 0.02Inhibition of uptake of 5-HT in rat brain cortex [AID181682, Type: Literature]
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20
[SID103164619]
IC50 0.034DRUGMATRIX: Serotonin (5-Hydroxytryptamine) 5-HT2C radioligand binding (ligand: [3H] Mesulergine) [AID625218, Type: confirmatory]5-hydroxytryptamine receptor 2C [gi:112816]
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