AC1MDZT5 (CID 2798335) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(1)
 
 
Inactive(11)
 
 
Unspecified(1)
 
 
Top Targets:
7TM GPCR Srx(1)
 
 
Ggt(1)
 
 
Lipase(1)
 
 
MarR(1)
 
 
NOD(1)
 
 
BioAssay Types:
Screening(8)
 
 
Literature(3)
 
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 13    Data Row: 13   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103272489]
 Antihypertensive activity in spontaneously hypertensive rats at 100 mg/kg po/day for 2 days [AID167922, Type: Literature]
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2
[SID103272489]
 Inhibitory activity for thromboxane synthetase determined by TXB2 levels in platelets from spontaneously hypertensive rats. [AID213137, Type: Literature]
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3
[SID26529986]
 Primary Cell Based High Throughput Screening Assay for Inhibitors of TLR4-MyD88 binding [AID811, Type: screening]toll-like receptor 4 [Homo sapiens] [gi:55662034]
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4
[SID26529986]
 Primary cell-based high-throughput screening assay to identify agonists of Sphingosine 1-Phosphate receptor 1 (S1P1) [AID1044, Type: screening]S1PR1 gene product [Homo sapiens] [gi:13027636]
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5
[SID26529986]
 Primary cell-based high-throughput screening assay to identify agonists of Sphingosine 1-Phosphate receptor 1 (S1P1) [AID1044, Type: screening]S1PR1 gene product [Homo sapiens] [gi:13027636]
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6
[SID26529986]
 Cell-based luminescence-based Maybridge primary high throughput screening assay to identify agonists of NOTCH [AID434982, Type: screening]NOTCH 1 [Homo sapiens] [gi:11275980]
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7
[SID26529986]
 Maybridge screen to identify antagonists of kappa opioid receptor 1 (OPRK1): fluorescence-based cell-based assay [AID652031, Type: screening]opioid receptor, kappa 1 [Homo sapiens] [gi:119607129]
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8
[SID26529986]
 Maybridge screen to identify antagonists of kappa opioid receptor 1 (OPRK1): fluorescence-based cell-based assay [AID652031, Type: screening]opioid receptor, kappa 1 [Homo sapiens] [gi:119607129]
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9
[SID26529986]
 Maybridge screen to identify antagonists of kappa opioid receptor 1 (OPRK1): fluorescence-based cell-based assay [AID652031, Type: screening]opioid receptor, kappa 1 [Homo sapiens] [gi:119607129]
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10
[SID26529986]
 Maybridge screen to identify antagonists of kappa opioid receptor 1 (OPRK1): fluorescence-based cell-based assay [AID652031, Type: screening]opioid receptor, kappa 1 [Homo sapiens] [gi:119607129]
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11
[SID26529986]
 Luminescence-based primary cell-based high throughput screening assay to identify inhibitors of NADPH oxidase 1 (Nox1): Maybridge Library [AID1792, Type: screening]NADPH oxidase 1 [Homo sapiens] [gi:83699673]
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12
[SID26529986]
 Luminescence-based primary cell-based high throughput screening assay to identify inhibitors of NADPH oxidase 1 (Nox1): Maybridge Library [AID1792, Type: screening]NADPH oxidase 1 [Homo sapiens] [gi:83699673]
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13
[SID26529986]
 Primary Cell Based High Throughput Screening Assay for Agonists of GALR2 [AID833, Type: screening]galanin receptor type 2 [Rattus norvegicus] [gi:2578455]
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14
[SID26529986]
 Primary Cell Based High Throughput Screening Assay for Agonists of GALR2 [AID833, Type: screening]galanin receptor type 2 [Rattus norvegicus] [gi:2578455]
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15
[SID26529986]
 Fluorescence polarization-based Maybridge primary biochemical high throughput screening assay to identify inhibitors of Protein Phosphatase Methylesterase 1 (PME-1). [AID2291, Type: screening]protein phosphatase methylesterase 1 [Homo sapiens] [gi:7706645]
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16
[SID92253549]
 A screen for compounds that inhibit the CapD enzyme of Bacillus anthracis [AID492967, Type: other]gamma-glutamyltranspeptidase [Bacillus anthracis str. 'Ames Ancestor'] [gi:47566732]
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17
[SID92253549]
 A screen for compounds that modulate the activity of the Staphylococcus aureus MgrA protein [AID602314, Type: other]MarR family regulatory protein [Staphylococcus aureus subsp. aureus str. Newman] [gi:151220867]
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18
[SID103272489]
 Tested for antihypertensive activity in spontaneously hypertensive rats at 100 mg/kg peroral dosage for 2 days; I is inactive [AID190211, Type: Literature]
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19
[SID26529986]
 Luminescence-based counterscreen for inhibitors of NADPH oxidase 1 (Nox1): biochemical high throughput screening assay to identify inhibitors of luminol (Maybridge Library) [AID1823, Type: screening]
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