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BioActivity Data for Compound cimaterol (CID 2755)

BioActivity Outcomes:
Active(4)
 
 
Inactive(273)
 
 
Inconclusive(8)
 
 
Unspecified(5)
 
 
Top Targets:
7tm 4(8)
 
 
 
 
NR LBD PPAR(8)
 
 
NR LBD AR(7)
 
 
 
NR LBD ER(7)
 
 
NR LBD TR(7)
 
 
BioAssay Types:
Confirmatory(162)
 
 
 
 
 
Literature(71)
 
 
 
 
 
Summary(26)
 
 
 
Screening(23)
 
 
BioAssay Categories:
Biochemical(10)
 
 
 
 
Toxicity(6)
 
 
Cell-based(22)
 
 
 
 
BioActivity Types:
Potency(170)
 
 
 
 
AC50(6)
 
 
 
EC50(3)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 193    Data Row: 290   Total Pages: 15   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID160687845]
EC50 0.00741Partial agonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrs [AID739708, Type: Literature]Beta-1 adrenergic receptor [gi:48429211]
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2
[SID160687845]
EC50 10Agonist activity at human beta2 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrs [AID739706, Type: Literature]Beta-2 adrenergic receptor [gi:296439450]
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3
[SID160687845]
EC50 10Agonist activity at human beta3 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrs [AID739704, Type: Literature]Beta-3 adrenergic receptor [gi:461604]
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4
[SID26751720]
Potency 11.9955Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation [AID504834, Type: confirmatory]
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5
[SID26751720]
qHTS profiling for inhibitors of Plasmodium falciparum proliferation [AID504749, Type: Literature]
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6
[SID170466620]
AC50 (uM) qHTS Assay for Identifying Compounds that block Entry of Ebola Virus, Screen 2 ratio channel [AID1117305, Type: confirmatory]
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7
[SID160687845]
Agonist activity at human beta3 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrs relative to isoprenaline [AID739703, Type: Literature]Beta-3 adrenergic receptor [gi:461604]
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8
[SID160687845]
Partial agonist activity at human beta1 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation measured after 5 hrs relative to isoprenaline [AID739707, Type: Literature]Beta-1 adrenergic receptor [gi:48429211]
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9
[SID160687845]
Agonist activity at human beta2 adrenoceptor expressed in CHOK1 cells assessed as induction of 3H]cAMP accumulation after 5 hrs relative to isoprenaline [AID739700, Type: Literature]Beta-2 adrenergic receptor [gi:296439450]
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10
[SID170466620]
Potency-Replicate_1 7.4978qHTS assay to identify small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID1159521, Type: confirmatory]RAR-related orphan receptor gamma [Mus musculus] [gi:15928672]
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11
[SID170466620]
AC50 (uM) 10qHTS Assay for Identifying Compounds that block Entry of Ebola Virus, Screen 2 green channel [AID1117298, Type: confirmatory]
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12
[SID170466620]
Ac50 10qHTS Assay for Identifying Compounds that block Entry of Ebola Virus: Screen 2, green channel [AID1117310, Type: confirmatory]
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13
[SID170466620]
AC50 (uM) 12.5893qHTS Assay for Identifying Compounds that block Entry of Ebola Virus, Screen 2 blue channel [AID1117304, Type: confirmatory]
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14
[SID170466620]
Ac50 12.5893qHTS Assay for Identifying Compounds that block Entry of Ebola Virus: Screen 2, blue channel [AID1117314, Type: confirmatory]
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15
[SID26751721]
Potency 100qHTS Assay for Inhibitors of Bacillus subtilis Sfp phosphopantetheinyl transferase (PPTase) [AID1490, Type: confirmatory]phosphopantetheinyl transferase [Bacillus subtilis] [gi:10954339]
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16
[SID85788751]
Luminescence Cell-Based Primary HTS to Identify Inhibitors of STK33 [AID2330, Type: screening]serine/threonine kinase 33 [Homo sapiens] [gi:12830367]
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17
[SID99302430]
A screen for compounds that inhibit the MenB enzyme of Mycobacterium tuberculosis [AID540299, Type: Literature]1,4-dihydroxy-2-naphthoyl-CoA synthase [Mycobacterium tuberculosis H37Rv] [gi:15607688]
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18
[SID92308879]
A screen for compounds that inhibit the activity of LtaS in Staphylococcus aureus [AID720641, Type: other]anion-binding protein [Staphylococcus aureus subsp. aureus Mu50] [gi:15923709]
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19
[SID170466620]
Potency-Replicate_1 qHTS assay to identify small molecule agonists of the vitamin D receptor (VDR) signaling pathway - cell viability counter screen [AID743224, Type: confirmatory]
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20
[SID170466620]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the vitamin D receptor (VDR) signaling pathway - cell viability counter screen [AID743225, Type: confirmatory]
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