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Chlordiazepoxide (CID 2712) - Compound BioActivity Data
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BioActivity Outcomes:
Active(121)
 
 
Inactive(568)
 
 
Inconclusive(72)
 
 
Unspecified(499)
 
 
Top Targets:
Neur chan LBD(113)
 
 
 
 
7tm 4(61)
 
 
 
Neur chan mem..(47)
 
 
 
 
NR LBD ER(16)
 
 
 
NR LBD AR(15)
 
 
 
 
 
BioAssay Types:
Literature(352)
 
 
 
 
 
Screening(348)
 
 
 
Confirmatory(302)
 
 
 
 
 
Summary(30)
 
 
 
 
BioActivity Types:
IC50(200)
 
 
 
 
 
Potency(195)
 
 
 
 
 
Ki(43)
 
 
EC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1014    Data Row: 1260   Total Pages: 63   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103165933]
IC50 0.2Concentration that inhibits binding of 1.5 nM [3H]diazepam to rat brain benzodiazepine receptor [AID40230, Type: Literature]
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2
[SID103165933]
IC50 0.2Inhibition of specific binding of 1.5 nM [3H]diazepam to rat brain benzodiazepine receptors [AID40519, Type: Literature]
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3
[SID103165933]
IC50 0.2Inhibitory concentration against specific binding of [3H]diazepam to Benzodiazepine receptor in rat brain [AID40521, Type: Literature]
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4
[SID103165933]
IC50 0.248In vitro for inhibition of [3H]diazepam towards Benzodiazepine receptor from rat [AID40661, Type: Literature]
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5
[SID103165933]
Ki 0.275Binding affinity by displacement of [3H]Ro-151788 from recombinant human gamma-aminobutyric-acid A receptor alpha3,beta3,gamma2 stably expressed in L cells [AID73245, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
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6
[SID103165933]
Ki 0.275Binding affinity by displacement of [3H]Ro-151788 from recombinant human gamma-aminobutyric-acid A receptor alpha3,beta3,gamma2 stably expressed in L cells [AID73245, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:462149]
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7
[SID103165933]
Ki 0.275Binding affinity by displacement of [3H]Ro-151788 from recombinant human gamma-aminobutyric-acid A receptor alpha3,beta3,gamma2 stably expressed in L cells [AID73245, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
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8
[SID103165933]
Ki 0.32Inhibition of [3H]Ro-151788 binding to human GABA A receptor (alpha-5-beta-3-gamma-2) stably expressed in L(tk-) cells. [AID73526, Type: Literature]
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9
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-1 [gi:120769]
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10
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-1 [gi:120782]
View
11
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-2 [gi:120758]
View
12
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:120761]
View
13
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-4 [gi:120763]
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14
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-5 [gi:120764]
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15
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:52000955]
View
16
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-2 [gi:52000957]
View
17
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]GABA theta subunit [gi:81902501]
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18
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit delta [gi:544363]
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19
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:120788]
View
20
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-3 [gi:120790]
View