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Chlordiazepoxide (CID 2712) - Compound BioActivity Data
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BioActivity Outcomes:
Active(120)
 
 
Inactive(557)
 
 
Inconclusive(74)
 
 
Unspecified(313)
 
 
Top Targets:
Neur chan LBD(113)
 
 
 
 
Neur chan mem..(47)
 
 
 
 
7TM GPCR Srx(31)
 
 
 
7TM GPCR Srsx(30)
 
 
 
NR LBD ER(16)
 
 
 
BioAssay Types:
Screening(347)
 
 
 
Literature(309)
 
 
 
 
 
Confirmatory(184)
 
 
 
 
 
Summary(30)
 
 
 
 
BioActivity Types:
IC50(200)
 
 
 
 
 
Potency(193)
 
 
 
 
 
Ki(43)
 
 
EC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 825    Data Row: 1064   Total Pages: 22   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103165933]
IC50 0.2Concentration that inhibits binding of 1.5 nM [3H]diazepam to rat brain benzodiazepine receptor [AID40230, Type: Literature]
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2
[SID103165933]
IC50 0.2Inhibition of specific binding of 1.5 nM [3H]diazepam to rat brain benzodiazepine receptors [AID40519, Type: Literature]
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3
[SID103165933]
IC50 0.2Inhibitory concentration against specific binding of [3H]diazepam to Benzodiazepine receptor in rat brain [AID40521, Type: Literature]
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4
[SID103165933]
IC50 0.248In vitro for inhibition of [3H]diazepam towards Benzodiazepine receptor from rat [AID40661, Type: Literature]
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5
[SID103165933]
Ki 0.275Binding affinity by displacement of [3H]Ro-151788 from recombinant human gamma-aminobutyric-acid A receptor alpha3,beta3,gamma2 stably expressed in L cells [AID73245, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
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6
[SID103165933]
Ki 0.275Binding affinity by displacement of [3H]Ro-151788 from recombinant human gamma-aminobutyric-acid A receptor alpha3,beta3,gamma2 stably expressed in L cells [AID73245, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:462149]
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7
[SID103165933]
Ki 0.275Binding affinity by displacement of [3H]Ro-151788 from recombinant human gamma-aminobutyric-acid A receptor alpha3,beta3,gamma2 stably expressed in L cells [AID73245, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
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8
[SID103165933]
Ki 0.32Inhibition of [3H]Ro-151788 binding to human GABA A receptor (alpha-5-beta-3-gamma-2) stably expressed in L(tk-) cells. [AID73526, Type: Literature]
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9
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-6 [gi:232127]
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10
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-1 [gi:120782]
View
11
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:120788]
View
12
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-3 [gi:120790]
View
13
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-1 [gi:120769]
View
14
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-4 [gi:120763]
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15
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:120761]
View
16
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-5 [gi:120764]
View
17
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-2 [gi:120758]
View
18
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit delta [gi:544363]
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19
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit pi [gi:3023821]
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20
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]GABA theta subunit [gi:81902501]
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21
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit epsilon [gi:13959374]
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22
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-1 [gi:51317298]
View
23
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:52000955]
View
24
[SID103165933]
IC50 0.33Inhibition of [3H]flunitrazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortex [AID40231, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-2 [gi:52000957]
View
25
[SID103165933]
Ki 0.368Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-5-beta-3-gamma-2 [AID73380, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
View
26
[SID103165933]
Ki 0.368Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-5-beta-3-gamma-2 expressed in L(tk-) cells [AID239702, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
View
27
[SID103165933]
Ki 0.368Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-5-beta-3-gamma-2 [AID73380, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View
28
[SID103165933]
Ki 0.368Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-5-beta-3-gamma-2 expressed in L(tk-) cells [AID239702, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View
29
[SID103165933]
Ki 0.368Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-5-beta-3-gamma-2 [AID73380, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-5 [gi:399519]
View
30
[SID103165933]
Ki 0.368Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-5-beta-3-gamma-2 expressed in L(tk-) cells [AID239702, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-5 [gi:399519]
View
31
[SID103165933]
Ki 0.392Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-2-beta-3-gamma-2 expressed in L(tk-) cells [AID239700, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View
32
[SID103165933]
Ki 0.392Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-2-beta-3-gamma-2 [AID73080, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View
33
[SID103165933]
Ki 0.392Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-2-beta-3-gamma-2 [AID73080, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
View
34
[SID103165933]
Ki 0.392Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-2-beta-3-gamma-2 expressed in L(tk-) cells [AID239700, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
View
35
[SID103165933]
Ki 0.392Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-2-beta-3-gamma-2 expressed in L(tk-) cells [AID239700, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-2 [gi:126302547]
View
36
[SID103165933]
Ki 0.392Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-2-beta-3-gamma-2 [AID73080, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-2 [gi:126302547]
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37
[SID103165933]
Ki 0.438Binding affinity against rat benzodiazepine (BZD) receptor [AID39933, Type: Literature]
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38
[SID103165933]
IC50 0.442Inhibition of binding of tritiated 3[H]diazepam radioligand to rat brain homogenates [AID40833, Type: Literature]
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39
[SID103165933]
Ki 0.46Displacement of [3H]Ro-151788 from human Gamma-aminobutyric acid A receptor alpha-2-beta-3-gamma-2 stably expressed in L(tk-) cells [AID73090, Type: Literature]
View
40
[SID103165933]
Ki 0.46Displacement of [3H]-Ro- 15-1788 from human GABA-A alpha-2-beta-3-gamma-2 receptor subunits expressed in Xenopus oocytes [AID73081, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View
41
[SID103165933]
Ki 0.46Displacement of [3H]-Ro- 15-1788 from human GABA-A alpha-2-beta-3-gamma-2 receptor subunits expressed in Xenopus oocytes [AID73081, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-2 [gi:126302547]
View
42
[SID103165933]
Ki 0.46Displacement of [3H]-Ro- 15-1788 from human GABA-A alpha-2-beta-3-gamma-2 receptor subunits expressed in Xenopus oocytes [AID73081, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
View
43
[SID103165933]
Ki 0.471Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-3-beta-3-gamma-2 [AID73235, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
View
44
[SID103165933]
Ki 0.471Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-3-beta-3-gamma-2 expressed in L(tk-) cells [AID239701, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:116242488]
View
45
[SID103165933]
Ki 0.471Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-3-beta-3-gamma-2 [AID73235, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View
46
[SID103165933]
Ki 0.471Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-3-beta-3-gamma-2 expressed in L(tk-) cells [AID239701, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View
47
[SID103165933]
Ki 0.471Displacement of [3H]-Ro- 15-1788 from human gamma-aminobutyric-acid GABA-A receptor alpha-3-beta-3-gamma-2 expressed in L(tk-) cells [AID239701, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:462149]
View
48
[SID103165933]
Ki 0.471Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-3-beta-3-gamma-2 [AID73235, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:462149]
View
49
[SID103165933]
Ki 0.52Displacement of [3H]-Ro- 15-1788 from human GABA-A alpha-5-beta-3-gamma-2 receptor subunits expressed in Xenopus oocytes [AID73382, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-5 [gi:399519]
View
50
[SID103165933]
Ki 0.52Displacement of [3H]-Ro- 15-1788 from human GABA-A alpha-5-beta-3-gamma-2 receptor subunits expressed in Xenopus oocytes [AID73382, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:120773]
View