CHEMBL462373 (CID 25169254) - BioAssay Data Summary for Compound
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BioActivity Outcomes:
Active(3)
 
 
BioAssay Types:
Literature(3)
 
 
BioActivity Types:
IC50(2)
 
 
Ki(1)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103588729]
Ki 0.07Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cells [AID409975, Type: Literature]P2Y purinoceptor 1 [gi:1352692]
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2
[SID103588729]
IC50 0.504Inhibition of ADP-induced human platelet aggregation [AID409976, Type: Literature]
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3
[SID103588729]
IC50 0.6Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPR [AID409974, Type: Literature]P2Y purinoceptor 1 [gi:1352692]
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