CHEMBL400388 (CID 25138030) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Inactive(1)
 
 
Inconclusive(1)
 
 
Top Targets:
Firefly Luc l..(1)
 
 
PTKc Lck Blk(1)
 
 
BioAssay Types:
Confirmatory(3)
 
 
 
 
Literature(1)
 
 
BioActivity Types:
Potency(3)
 
 
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID124349826]
Potency 0.73qHTS Assay for Inhibitors of Firefly Luciferase from the GSK Published Protein Kinase Inhibitor Set [AID652016, Type: confirmatory]Luciferase [Photinus pyralis] [gi:160794]
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2
[SID103551391]
IC50 3.3Inhibition of murine Lck by TR-FRET assay [AID308759, Type: Literature]Proto-oncogene tyrosine-protein kinase LCK [gi:78099784]
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3
[SID124349826]
Potency qHTS Assay for Inhibitors of Sea Pansy Luciferase from the GSK Published Protein Kinase Inhibitor Set [AID652015, Type: confirmatory]Renilla-luciferin 2-monooxygenase (EC 1.13.12.5) - sea pansy (Renilla reniformis) (fragment) [gi:84399]
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4
[SID124349826]
Potency 2.5018qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID540256, Type: confirmatory]
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