Bookmark and Share
CHEMBL599052 (CID 24952580) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(3)
 
 
Unspecified(7)
 
 
Top Targets:
7tm 4(3)
 
 
 
BioAssay Types:
Literature(10)
 
 
 
BioActivity Types:
Ki(9)
 
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 10    Data Row: 10   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103722865]
Ki 0.0013Displacement of [3H]PGE2 from human EP4 receptor expressed in HEK293-EBNA cells by scintillation counting [AID459005, Type: Literature]Prostaglandin E2 receptor EP4 subtype [gi:548476]
View
2
[SID103722865]
IC50 0.0036Antagonist activity at human EP4 receptor expressed in HEK293 cells assessed as inhibition of PGE2-induced cAMP accumulation by scintillation proximity assay [AID459014, Type: Literature]Prostaglandin E2 receptor EP4 subtype [gi:548476]
View
3
[SID103722865]
Ki 0.746Displacement of [3H]PGE2 from human EP2 receptor expressed in HEK293-EBNA cells by scintillation counting [AID459006, Type: Literature]Prostaglandin E2 receptor EP2 subtype [gi:38258920]
View
4
[SID103722865]
Ki 0.456Displacement of [3H]PGE2 from human EP1 receptor expressed in HEK293-EBNA cells by scintillation counting [AID459007, Type: Literature]Prostaglandin E2 receptor EP1 subtype [gi:83287886]
View
5
[SID103722865]
Ki 0.456Displacement of [3H]SQ29548 from human TP receptor expressed in HEK293-EBNA cells by scintillation counting [AID459012, Type: Literature]Thromboxane A2 receptor [gi:229463010]
View
6
[SID103722865]
Ki 0.456Displacement of [3H]PGD2 from human DP2 receptor expressed in HEK293-EBNA cells by scintillation counting [AID459010, Type: Literature]Prostaglandin D2 receptor 2 [gi:296439334]
View
7
[SID103722865]
Ki 0.456Displacement of [3H]PGE2 from human EP3 receptor expressed in HEK293-EBNA cells by scintillation counting [AID459008, Type: Literature]Prostaglandin E2 receptor EP3 subtype [gi:1172071]
View
8
[SID103722865]
Ki 0.456Displacement of [3H]PGF2alpha from human FP receptor expressed in HEK293-EBNA cells by scintillation counting [AID459013, Type: Literature]Prostaglandin F2-alpha receptor [gi:1172442]
View
9
[SID103722865]
Ki 0.456Displacement of [3H]iloprost from human IP receptor expressed in HEK293-EBNA cells by scintillation counting [AID459011, Type: Literature]Prostacyclin receptor [gi:1172500]
View
10
[SID103722865]
Ki 0.456Displacement of [3H]PGD2 from human DP1 receptor expressed in HEK293-EBNA cells by scintillation counting [AID459009, Type: Literature]Prostaglandin D2 receptor [gi:2495009]
View