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CHEMBL384153 (CID 24825431) - Compound BioActivity Data
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BioActivity Outcomes:
Active(4)
 
 
Unspecified(4)
 
 
Top Targets:
NR LBD Lrh-1(4)
 
 
 
NR LBD SF-1(3)
 
 
 
BioAssay Types:
Literature(8)
 
 
 
BioActivity Types:
EC50(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 8   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103501444]
EC50 0.03162Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to control [AID593528, Type: Literature]Nuclear receptor subfamily 5 group A member 2 [gi:7676156]
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2
[SID103501444]
EC50 0.034Binding affinity to human LRH1 by FRET-based peptide recruitment assay [AID271721, Type: Literature]Nuclear receptor subfamily 5 group A member 2 [gi:7676156]
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3
[SID103501444]
EC50 0.03981Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to control [AID593529, Type: Literature]Steroidogenic factor 1 [gi:3121738]
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4
[SID103501444]
EC50 0.043Binding affinity to human SF1 by FRET-based peptide recruitment assay [AID271722, Type: Literature]Steroidogenic factor 1 [gi:3121738]
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5
[SID103501444]
Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay [AID593527, Type: Literature]Steroidogenic factor 1 [gi:3121738]
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6
[SID103501444]
Binding affinity to human LRH1 relative to 3-(E-Oct-4-en-4-yl)-1-phenylamino-2-phenyl-cis-bicyclo[3.3.0]oct-2-ene by FRET-based peptide recruitment assay [AID271715, Type: Literature]Nuclear receptor subfamily 5 group A member 2 [gi:7676156]
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7
[SID103501444]
Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay [AID593526, Type: Literature]Nuclear receptor subfamily 5 group A member 2 [gi:7676156]
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8
[SID103501444]
Stability in 1 M acetic acid [AID271720, Type: Literature]
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