| 1 | [SID49820089] | Active | Potency | 1.6343 | qHTS for inhibitors of Phosphogylcerate Kinase: Hit Validation Screen [AID686980, Type: confirmatory] | phosphoglycerate kinase [Trypanosoma brucei] [gi:115503961] |  View X | Row No. | 1 | | Structure | 
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 1.6343 [uM] | | BioAssay | qHTS for inhibitors of Phosphogylcerate Kinase: Hit Validation Screen | | AID | 686980 | | BioAssay type | confirmatory | | Target | phosphoglycerate kinase [Trypanosoma brucei] [gi:115503961] | | PubMed | | | Data Table | |
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| 2 | [SID49820089] | Active | IC50 | 1.92 | Identification of SV40 T antigen inhibitors: A route to novel anti-viral reagents [AID1903, Type: confirmatory] | large T antigen [Simian virus 40] [gi:297591903] | View X | Row No. | 2 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | IC50 | 1.92 [uM] | | BioAssay | Identification of SV40 T antigen inhibitors: A route to novel anti-viral reagents | | AID | 1903 | | BioAssay type | confirmatory | | Target | large T antigen [Simian virus 40] [gi:297591903] | | PubMed | | | Data Table | |
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| 3 | [SID49820089] | Active | AC50 | 2.438 | C-LANA FP assay Measured in Biochemical System Using Plate Reader - 2117-01_Inhibitor_Dose_CherryPick_Activity [AID504725, Type: confirmatory] | LANA [Human herpesvirus 8] [gi:312275222] | View X | Row No. | 3 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | AC50 | 2.438 [uM] | | BioAssay | C-LANA FP assay Measured in Biochemical System Using Plate Reader - 2117-01_Inhibitor_Dose_CherryPick_Activity | | AID | 504725 | | BioAssay type | confirmatory | | Target | LANA [Human herpesvirus 8] [gi:312275222] | | PubMed | | | Data Table | |
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| 4 | [SID49820089] | Active | Potency | 2.6855 | Tb PFK orthogonal confirmatory assay using ATP depletion (Kinase-Glo Plus) as an alternative measure of Tb PFK activity: Hit Validation [AID504636, Type: confirmatory] | ATP-dependent phosphofructokinase [Trypanosoma brucei] [gi:72386991] | View X | Row No. | 4 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 2.6855 [uM] | | BioAssay | Tb PFK orthogonal confirmatory assay using ATP depletion (Kinase-Glo Plus) as an alternative measure of Tb PFK activity: Hit Validation | | AID | 504636 | | BioAssay type | confirmatory | | Target | ATP-dependent phosphofructokinase [Trypanosoma brucei] [gi:72386991] | | PubMed | | | Data Table | |
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| 5 | [SID49820089] | Active | Potency | 3.7933 | Inhibitors of T. brucei phosphofructokinase: Hit Validation [AID504637, Type: confirmatory] | ATP-dependent phosphofructokinase [Trypanosoma brucei] [gi:72386991] | View X | Row No. | 5 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 3.7933 [uM] | | BioAssay | Inhibitors of T. brucei phosphofructokinase: Hit Validation | | AID | 504637 | | BioAssay type | confirmatory | | Target | ATP-dependent phosphofructokinase [Trypanosoma brucei] [gi:72386991] | | PubMed | | | Data Table | |
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| 6 | [SID49820089] | Active | IC50 | 6.98 | Dose Response confirmation of uHTS hits from a small molecule inhibitors of mouse intestinal alkaline phosphatase via a luminescent assay [AID488785, Type: confirmatory] | intestinal alkaline phosphatase precursor [Mus musculus] [gi:124487323] | View X | Row No. | 6 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | IC50 | 6.98 [uM] | | BioAssay | Dose Response confirmation of uHTS hits from a small molecule inhibitors of mouse intestinal alkaline phosphatase via a luminescent assay | | AID | 488785 | | BioAssay type | confirmatory | | Target | intestinal alkaline phosphatase precursor [Mus musculus] [gi:124487323] | | PubMed | | | Data Table | |
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| 7 | [SID49820089] | Active | Potency | 10 | qHTS Assay for Inhibitors of BAZ2B [AID504333, Type: confirmatory] | bromodomain adjacent to zinc finger domain 2B [Homo sapiens] [gi:6683500] | View X | Row No. | 7 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 10 [uM] | | BioAssay | qHTS Assay for Inhibitors of BAZ2B | | AID | 504333 | | BioAssay type | confirmatory | | Target | bromodomain adjacent to zinc finger domain 2B [Homo sapiens] [gi:6683500] | | PubMed | | | Data Table | |
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| 8 | [SID49820089] | Active | Potency | 10 | qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory] | euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070] | View X | Row No. | 8 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 10 [uM] | | BioAssay | qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a | | AID | 504332 | | BioAssay type | confirmatory | | Target | euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070] | | PubMed | | | Data Table | |
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| 9 | [SID49820089] | Active | IC50 | 10.55 | A biochemical assay using the ADP-Hunter methodology, purified TAg, and ATP to identify compounds that inhibit the ATPase activity of Tag - Counter Screen [AID2501, Type: confirmatory] | | View X | Row No. | 9 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | IC50 | 10.55 [uM] | | BioAssay | A biochemical assay using the ADP-Hunter methodology, purified TAg, and ATP to identify compounds that inhibit the ATPase activity of Tag - Counter Screen | | AID | 2501 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 10 | [SID49820089] | Active | Potency | 14.1254 | qHTS Assay for Inhibitors of Influenza NS1 Protein Function [AID2326, Type: confirmatory] | nonstructural protein 1 [Influenza A virus (A/WSN/1933(H1N1))] [gi:194352380] | View X | Row No. | 10 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 14.1254 [uM] | | BioAssay | qHTS Assay for Inhibitors of Influenza NS1 Protein Function | | AID | 2326 | | BioAssay type | confirmatory | | Target | nonstructural protein 1 [Influenza A virus (A/WSN/1933(H1N1))] [gi:194352380] | | PubMed | | | Data Table | |
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| 11 | [SID49820089] | Active | Potency | 19.0115 | qHTS Assay to Find Inhibitors of T. brucei phosphofructokinase [AID485367, Type: confirmatory] | ATP-dependent phosphofructokinase [Trypanosoma brucei] [gi:72386991] | View X | Row No. | 11 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 19.0115 [uM] | | BioAssay | qHTS Assay to Find Inhibitors of T. brucei phosphofructokinase | | AID | 485367 | | BioAssay type | confirmatory | | Target | ATP-dependent phosphofructokinase [Trypanosoma brucei] [gi:72386991] | | PubMed | | | Data Table | |
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| 12 | [SID49820089] | Active | EC50 | 21.3 | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Human Intestinal Alkaline Phosphatase [AID488873, Type: confirmatory] | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | View X | Row No. | 12 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | EC50 | 21.3 [uM] | | BioAssay | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Human Intestinal Alkaline Phosphatase | | AID | 488873 | | BioAssay type | confirmatory | | Target | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | | PubMed | | | Data Table | |
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| 13 | [SID49820089] | Active | EC50 | 21.3 | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Human Intestinal Alkaline Phosphatase [AID488873, Type: confirmatory] | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | View X | Row No. | 13 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | EC50 | 21.3 [uM] | | BioAssay | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Human Intestinal Alkaline Phosphatase | | AID | 488873 | | BioAssay type | confirmatory | | Target | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | | PubMed | | | Data Table | |
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| 14 | [SID49820089] | Active | EC50 | 21.5 | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. [AID488880, Type: confirmatory] | alkaline phosphatase, tissue-nonspecific isozyme isoform 1 precursor [Homo sapiens] [gi:116734717] | View X | Row No. | 14 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | EC50 | 21.5 [uM] | | BioAssay | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. | | AID | 488880 | | BioAssay type | confirmatory | | Target | alkaline phosphatase, tissue-nonspecific isozyme isoform 1 precursor [Homo sapiens] [gi:116734717] | | PubMed | | | Data Table | |
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| 15 | [SID49820089] | Active | EC50 | 21.5 | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. [AID488880, Type: confirmatory] | alkaline phosphatase, tissue-nonspecific isozyme isoform 1 precursor [Homo sapiens] [gi:116734717] | View X | Row No. | 15 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | EC50 | 21.5 [uM] | | BioAssay | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. | | AID | 488880 | | BioAssay type | confirmatory | | Target | alkaline phosphatase, tissue-nonspecific isozyme isoform 1 precursor [Homo sapiens] [gi:116734717] | | PubMed | | | Data Table | |
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| 16 | [SID49820089] | Active | EC50 | 23.5 | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase [AID488878, Type: confirmatory] | alkaline phosphatase, placental-like preproprotein [Homo sapiens] [gi:157266296] | View X | Row No. | 16 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | EC50 | 23.5 [uM] | | BioAssay | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase | | AID | 488878 | | BioAssay type | confirmatory | | Target | alkaline phosphatase, placental-like preproprotein [Homo sapiens] [gi:157266296] | | PubMed | | | Data Table | |
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| 17 | [SID49820089] | Active | EC50 | 23.5 | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase [AID488878, Type: confirmatory] | alkaline phosphatase, placental-like preproprotein [Homo sapiens] [gi:157266296] | View X | Row No. | 17 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | EC50 | 23.5 [uM] | | BioAssay | Dose Response confirmation of uHTS activators of Mouse Intestinal Alkaline Phosphatase using Placental Alkaline Phosphatase | | AID | 488878 | | BioAssay type | confirmatory | | Target | alkaline phosphatase, placental-like preproprotein [Homo sapiens] [gi:157266296] | | PubMed | | | Data Table | |
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| 18 | [SID49820089] | Active | Potency | 28.1838 | qHTS Assay for Inhibitors of Bloom's syndrome helicase (BLM) [AID2528, Type: confirmatory] | Bloom syndrome protein [Homo sapiens] [gi:4557365] | View X | Row No. | 18 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | Potency | 28.1838 [uM] | | BioAssay | qHTS Assay for Inhibitors of Bloom's syndrome helicase (BLM) | | AID | 2528 | | BioAssay type | confirmatory | | Target | Bloom syndrome protein [Homo sapiens] [gi:4557365] | | PubMed | | | Data Table | |
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| 19 | [SID49820089] | Active | AC50 | 266.747 | 24 hour HeLa Cytotox assay Measured in Cell-Based System Using Plate Reader - 2117-03_Inhibitor_Dose_CherryPick_Activity [AID504726, Type: confirmatory] | LANA [Human herpesvirus 8] [gi:312275222] | View X | Row No. | 19 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | AC50 | 266.747 [uM] | | BioAssay | 24 hour HeLa Cytotox assay Measured in Cell-Based System Using Plate Reader - 2117-03_Inhibitor_Dose_CherryPick_Activity | | AID | 504726 | | BioAssay type | confirmatory | | Target | LANA [Human herpesvirus 8] [gi:312275222] | | PubMed | | | Data Table | |
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| 20 | [SID49820089] | Active | | | uHTS identification of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, via a fluorescence intensity assay [AID651560, Type: screening] | Low molecular weight phosphotyrosine protein phosphatase [gi:1709543] | View X | Row No. | 20 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS identification of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, via a fluorescence intensity assay | | AID | 651560 | | BioAssay type | screening | | Target | Low molecular weight phosphotyrosine protein phosphatase [gi:1709543] | | PubMed | | | Data Table | |
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| 21 | [SID49820089] | Active | | | uHTS identification of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, via a fluorescence intensity assay [AID651560, Type: screening] | Low molecular weight phosphotyrosine protein phosphatase [gi:1709543] | View X | Row No. | 21 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS identification of small molecule inhibitors of Low Molecular Weight Protein Tyrosine Phosphatase, LMPTP, via a fluorescence intensity assay | | AID | 651560 | | BioAssay type | screening | | Target | Low molecular weight phosphotyrosine protein phosphatase [gi:1709543] | | PubMed | | | Data Table | |
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| 22 | [SID49820089] | Active | | | Counterscreen for inhibitors of 5-meCpG-binding domain protein 2 (MBD2): TRFRET-based biochemical primary high throughput screening assay to identify inhibitors of binding of ubiquitin-like with PHD and ring finger domains 1 (UHRF1) to methylated oligonucleotide [AID687016, Type: screening] | UHRF1 gene product [Homo sapiens] [gi:115430235] | View X | Row No. | 22 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Counterscreen for inhibitors of 5-meCpG-binding domain protein 2 (MBD2): TRFRET-based biochemical primary high throughput screening assay to identify inhibitors of binding of ubiquitin-like with PHD and ring finger domains 1 (UHRF1) to methylated oligonucleotide | | AID | 687016 | | BioAssay type | screening | | Target | UHRF1 gene product [Homo sapiens] [gi:115430235] | | PubMed | | | Data Table | |
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| 23 | [SID49820089] | Active | | | RNA aptamer-based HTS for inhibitors of GRK2 [AID488847, Type: screening] | beta-adrenergic receptor kinase 1 [Homo sapiens] [gi:148539876] | View X | Row No. | 23 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | RNA aptamer-based HTS for inhibitors of GRK2 | | AID | 488847 | | BioAssay type | screening | | Target | beta-adrenergic receptor kinase 1 [Homo sapiens] [gi:148539876] | | PubMed | | | Data Table | |
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| 24 | [SID49820089] | Active | | | VEID(2) R110 Enzymatic Primary HTS to identify Inhibitors of Caspase 6 Measured in Biochemical System Using Plate Reader - 7052-01_Inhibitor_SinglePoint_HTS_Activity_Set2 [AID686996, Type: screening] | | View X | Row No. | 24 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | VEID(2) R110 Enzymatic Primary HTS to identify Inhibitors of Caspase 6 Measured in Biochemical System Using Plate Reader - 7052-01_Inhibitor_SinglePoint_HTS_Activity_Set2 | | AID | 686996 | | BioAssay type | screening | | Target | | | PubMed | | | Data Table | |
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| 25 | [SID49820089] | Active | | | uHTS identification of DNMT1 inhibitors in a Fluorescent Molecular Beacon assay [AID588458, Type: screening] | DNA (cytosine-5)-methyltransferase 1 isoform b [Homo sapiens] [gi:4503351] | View X | Row No. | 25 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS identification of DNMT1 inhibitors in a Fluorescent Molecular Beacon assay | | AID | 588458 | | BioAssay type | screening | | Target | DNA (cytosine-5)-methyltransferase 1 isoform b [Homo sapiens] [gi:4503351] | | PubMed | | | Data Table | |
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| 26 | [SID49820089] | Active | | | uHTS identification of DNMT1 inhibitors in a Fluorescent Molecular Beacon assay [AID588458, Type: screening] | DNA (cytosine-5)-methyltransferase 1 isoform b [Homo sapiens] [gi:4503351] | View X | Row No. | 26 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS identification of DNMT1 inhibitors in a Fluorescent Molecular Beacon assay | | AID | 588458 | | BioAssay type | screening | | Target | DNA (cytosine-5)-methyltransferase 1 isoform b [Homo sapiens] [gi:4503351] | | PubMed | | | Data Table | |
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| 27 | [SID49820089] | Active | | | uHTS Colorimetric assay for identification of inhibitors of Scp-1 [AID493091, Type: screening] | carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1 [Homo sapiens] [gi:10864009] | View X | Row No. | 27 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS Colorimetric assay for identification of inhibitors of Scp-1 | | AID | 493091 | | BioAssay type | screening | | Target | carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1 [Homo sapiens] [gi:10864009] | | PubMed | | | Data Table | |
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| 28 | [SID49820089] | Active | | | Primary cell-based high-throughput screening for identification of compounds that activate/potentiate calcium-activated chloride channels (TMEM16A) [AID623877, Type: screening] | Ano1 gene product [Mus musculus] [gi:334278898] | View X | Row No. | 28 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Primary cell-based high-throughput screening for identification of compounds that activate/potentiate calcium-activated chloride channels (TMEM16A) | | AID | 623877 | | BioAssay type | screening | | Target | Ano1 gene product [Mus musculus] [gi:334278898] | | PubMed | | | Data Table | |
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| 29 | [SID49820089] | Active | | | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet-activating factor acetylhydrolase 1b, catalytic subunit 2 (PAFAH1B2) [AID492953, Type: screening] | platelet-activating factor acetylhydrolase IB subunit beta isoform b [Homo sapiens] [gi:296080766] | View X | Row No. | 29 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet-activating factor acetylhydrolase 1b, catalytic subunit 2 (PAFAH1B2) | | AID | 492953 | | BioAssay type | screening | | Target | platelet-activating factor acetylhydrolase IB subunit beta isoform b [Homo sapiens] [gi:296080766] | | PubMed | | | Data Table | |
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| 30 | [SID49820089] | Active | IC50 | | uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (eIF4H) [AID2012, Type: confirmatory] | Eukaryotic translation initiation factor 4H [Homo sapiens] [gi:45219878] | View X | Row No. | 30 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | IC50 | [uM] | | BioAssay | uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (eIF4H) | | AID | 2012 | | BioAssay type | confirmatory | | Target | Eukaryotic translation initiation factor 4H [Homo sapiens] [gi:45219878] | | PubMed | | | Data Table | |
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| 31 | [SID49820089] | Active | | | MLPCN SirT-5 Measured in Biochemical System Using Imaging - 7044-01_Inhibitor_SinglePoint_HTS_Activity_Set5 [AID652115, Type: screening] | NAD-dependent protein deacylase sirtuin-5, mitochondrial [gi:38258652] | View X | Row No. | 31 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | MLPCN SirT-5 Measured in Biochemical System Using Imaging - 7044-01_Inhibitor_SinglePoint_HTS_Activity_Set5 | | AID | 652115 | | BioAssay type | screening | | Target | NAD-dependent protein deacylase sirtuin-5, mitochondrial [gi:38258652] | | PubMed | | | Data Table | |
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| 32 | [SID49820089] | Active | | | MLPCN SirT-5 Measured in Biochemical System Using Imaging - 7044-01_Inhibitor_SinglePoint_HTS_Activity_Set5 [AID652115, Type: screening] | NAD-dependent protein deacylase sirtuin-5, mitochondrial [gi:38258652] | View X | Row No. | 32 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | MLPCN SirT-5 Measured in Biochemical System Using Imaging - 7044-01_Inhibitor_SinglePoint_HTS_Activity_Set5 | | AID | 652115 | | BioAssay type | screening | | Target | NAD-dependent protein deacylase sirtuin-5, mitochondrial [gi:38258652] | | PubMed | | | Data Table | |
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| 33 | [SID49820089] | Active | IC50 | | uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (PABP) [AID2014, Type: confirmatory] | polyadenylate-binding protein 1 [Homo sapiens] [gi:46367787] | View X | Row No. | 33 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | IC50 | [uM] | | BioAssay | uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (PABP) | | AID | 2014 | | BioAssay type | confirmatory | | Target | polyadenylate-binding protein 1 [Homo sapiens] [gi:46367787] | | PubMed | | | Data Table | |
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| 34 | [SID49820089] | Active | | | HTS-Luminescent assay for inhibitors of ALR by detection of hydrogen peroxide production Measured in Biochemical System Using Plate Reader - 2036-02_Inhibitor_SinglePoint_HTS [AID485317, Type: screening] | FAD-linked sulfhydryl oxidase ALR [Homo sapiens] [gi:54112432] | View X | Row No. | 34 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | HTS-Luminescent assay for inhibitors of ALR by detection of hydrogen peroxide production Measured in Biochemical System Using Plate Reader - 2036-02_Inhibitor_SinglePoint_HTS | | AID | 485317 | | BioAssay type | screening | | Target | FAD-linked sulfhydryl oxidase ALR [Homo sapiens] [gi:54112432] | | PubMed | | | Data Table | |
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| 35 | [SID49820089] | Active | | | uHTS Luminescent assay for identification of inhibitors of human intestinal alkaline phosphatase [AID2544, Type: screening] | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | View X | Row No. | 35 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS Luminescent assay for identification of inhibitors of human intestinal alkaline phosphatase | | AID | 2544 | | BioAssay type | screening | | Target | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | | PubMed | | | Data Table | |
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| 36 | [SID49820089] | Active | | | uHTS Luminescent assay for identification of inhibitors of human intestinal alkaline phosphatase [AID2544, Type: screening] | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | View X | Row No. | 36 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS Luminescent assay for identification of inhibitors of human intestinal alkaline phosphatase | | AID | 2544 | | BioAssay type | screening | | Target | Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142] | | PubMed | | | Data Table | |
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| 37 | [SID49820089] | Active | | | Fluorescence-based biochemical primary high throughput assay to identify inhibitors of T-cell receptor (TCR)-CD3 interaction using a TAMRA-labeled TCR probe [AID651800, Type: screening] | TCRAV4S1 [Homo sapiens] [gi:2358024] | View X | Row No. | 37 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence-based biochemical primary high throughput assay to identify inhibitors of T-cell receptor (TCR)-CD3 interaction using a TAMRA-labeled TCR probe | | AID | 651800 | | BioAssay type | screening | | Target | TCRAV4S1 [Homo sapiens] [gi:2358024] | | PubMed | | | Data Table | |
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| 38 | [SID49820089] | Active | | | Fluorescence-based biochemical primary high throughput confirmation assay to identify inhibitors of T-cell receptor (TCR)-CD3 interaction using a TAMRA-labeled TCR probe [AID652036, Type: screening] | TCRAV4S1 [Homo sapiens] [gi:2358024] | View X | Row No. | 38 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence-based biochemical primary high throughput confirmation assay to identify inhibitors of T-cell receptor (TCR)-CD3 interaction using a TAMRA-labeled TCR probe | | AID | 652036 | | BioAssay type | screening | | Target | TCRAV4S1 [Homo sapiens] [gi:2358024] | | PubMed | | | Data Table | |
|
| 39 | [SID49820089] | Active | | | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet activating factor acetylhydrolase 2 (PAFAH2) [AID492956, Type: screening] | platelet-activating factor acetylhydrolase 2, cytoplasmic [Homo sapiens] [gi:4758878] | View X | Row No. | 39 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet activating factor acetylhydrolase 2 (PAFAH2) | | AID | 492956 | | BioAssay type | screening | | Target | platelet-activating factor acetylhydrolase 2, cytoplasmic [Homo sapiens] [gi:4758878] | | PubMed | | | Data Table | |
|
| 40 | [SID49820089] | Active | | | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet activating factor acetylhydrolase 2 (PAFAH2) [AID492956, Type: screening] | platelet-activating factor acetylhydrolase 2, cytoplasmic [Homo sapiens] [gi:4758878] | View X | Row No. | 40 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet activating factor acetylhydrolase 2 (PAFAH2) | | AID | 492956 | | BioAssay type | screening | | Target | platelet-activating factor acetylhydrolase 2, cytoplasmic [Homo sapiens] [gi:4758878] | | PubMed | | | Data Table | |
|
| 41 | [SID49820089] | Active | | | uHTS identification of SUMO1-mediated protein-protein interactions [AID602429, Type: screening] | SUMO-1 [Homo sapiens] [gi:1762973] | View X | Row No. | 41 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | uHTS identification of SUMO1-mediated protein-protein interactions | | AID | 602429 | | BioAssay type | screening | | Target | SUMO-1 [Homo sapiens] [gi:1762973] | | PubMed | | | Data Table | |
|
| 42 | [SID49820089] | Active | | | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) [AID463082, Type: screening] | PLA2G7 gene product [Homo sapiens] [gi:270133071] | View X | Row No. | 42 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) | | AID | 463082 | | BioAssay type | screening | | Target | PLA2G7 gene product [Homo sapiens] [gi:270133071] | | PubMed | | | Data Table | |
|
| 43 | [SID49820089] | Active | | | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) [AID463082, Type: screening] | PLA2G7 gene product [Homo sapiens] [gi:270133071] | View X | Row No. | 43 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) | | AID | 463082 | | BioAssay type | screening | | Target | PLA2G7 gene product [Homo sapiens] [gi:270133071] | | PubMed | | | Data Table | |
|
| 44 | [SID49820089] | Active | | | Fluorescence polarization-based counterscreen for RBBP9 inhibitors: primary biochemical high throughput screening assay to identify inhibitors of the oxidoreductase glutathione S-transferase omega 1(GSTO1). [AID1974, Type: screening] | glutathione S-transferase omega-1 isoform 1 [Homo sapiens] [gi:4758484] | View X | Row No. | 44 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence polarization-based counterscreen for RBBP9 inhibitors: primary biochemical high throughput screening assay to identify inhibitors of the oxidoreductase glutathione S-transferase omega 1(GSTO1). | | AID | 1974 | | BioAssay type | screening | | Target | glutathione S-transferase omega-1 isoform 1 [Homo sapiens] [gi:4758484] | | PubMed | | | Data Table | |
|
| 45 | [SID49820089] | Active | | | Fluorescence polarization-based counterscreen for RBBP9 inhibitors: primary biochemical high throughput screening assay to identify inhibitors of the oxidoreductase glutathione S-transferase omega 1(GSTO1). [AID1974, Type: screening] | glutathione S-transferase omega-1 isoform 1 [Homo sapiens] [gi:4758484] | View X | Row No. | 45 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Fluorescence polarization-based counterscreen for RBBP9 inhibitors: primary biochemical high throughput screening assay to identify inhibitors of the oxidoreductase glutathione S-transferase omega 1(GSTO1). | | AID | 1974 | | BioAssay type | screening | | Target | glutathione S-transferase omega-1 isoform 1 [Homo sapiens] [gi:4758484] | | PubMed | | | Data Table | |
|
| 46 | [SID49820089] | Active | | | Primary biochemical high throughput screening assay to identify inhibitors of VIM-2 metallo-beta-lactamase [AID1527, Type: screening] | metallo beta-lactamase [Pseudomonas aeruginosa] [gi:7381449] | View X | Row No. | 46 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Primary biochemical high throughput screening assay to identify inhibitors of VIM-2 metallo-beta-lactamase | | AID | 1527 | | BioAssay type | screening | | Target | metallo beta-lactamase [Pseudomonas aeruginosa] [gi:7381449] | | PubMed | | | Data Table | |
|
| 47 | [SID49820089] | Active | | | Primary biochemical high throughput screening assay to identify inhibitors of VIM-2 metallo-beta-lactamase [AID1527, Type: screening] | metallo beta-lactamase [Pseudomonas aeruginosa] [gi:7381449] | View X | Row No. | 47 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | Primary biochemical high throughput screening assay to identify inhibitors of VIM-2 metallo-beta-lactamase | | AID | 1527 | | BioAssay type | screening | | Target | metallo beta-lactamase [Pseudomonas aeruginosa] [gi:7381449] | | PubMed | | | Data Table | |
|
| 48 | [SID49820089] | Active | | | qHTS of Yeast-based Assay for SARS-CoV PLP [AID485353, Type: confirmatory] | orf1ab polyprotein (pp1ab) [SARS coronavirus] [gi:30124074] | View X | Row No. | 48 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | qHTS of Yeast-based Assay for SARS-CoV PLP | | AID | 485353 | | BioAssay type | confirmatory | | Target | orf1ab polyprotein (pp1ab) [SARS coronavirus] [gi:30124074] | | PubMed | | | Data Table | |
|
| 49 | [SID49820089] | Active | | | qHTS of Yeast-based Assay for SARS-CoV PLP [AID485353, Type: confirmatory] | orf1ab polyprotein (pp1ab) [SARS coronavirus] [gi:30124074] | View X | Row No. | 49 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | qHTS of Yeast-based Assay for SARS-CoV PLP | | AID | 485353 | | BioAssay type | confirmatory | | Target | orf1ab polyprotein (pp1ab) [SARS coronavirus] [gi:30124074] | | PubMed | | | Data Table | |
|
| 50 | [SID49820089] | Active | | | qHTS of Yeast-based Assay for SARS-CoV PLP [AID485353, Type: confirmatory] | orf1ab polyprotein (pp1ab) [SARS coronavirus] [gi:30124074] | View X | Row No. | 50 | | Structure |
| | Substance | | | SID | 49820089 | | CID | 24818067 | | Outcome | Active | | BioAssay | qHTS of Yeast-based Assay for SARS-CoV PLP | | AID | 485353 | | BioAssay type | confirmatory | | Target | orf1ab polyprotein (pp1ab) [SARS coronavirus] [gi:30124074] | | PubMed | | | Data Table | |
|
Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
