Bookmark and Share

BioActivity Data for Compound CHEMBL9306 (CID 23714647)

BioActivity Outcomes:
Active(3)
 
 
Inactive(62)
 
 
Inconclusive(6)
 
 
Unspecified(2)
 
 
Top Targets:
NR LBD AR(7)
 
 
 
NR LBD ER(7)
 
 
NR LBD GR(4)
 
 
 
NR LBD TR(3)
 
 
7tm 4(2)
 
 
BioAssay Types:
Confirmatory(53)
 
 
 
 
Summary(15)
 
 
 
 
Screening(2)
 
 
Literature(1)
 
 
BioAssay Categories:
Biochemical(4)
 
 
 
Toxicity(6)
 
 
BioActivity Types:
Potency(65)
 
 
 
IC50(1)
 
 
Kd(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 73    Data Row: 73   Total Pages: 4   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103168543]
IC50 0.068Inhibition of Citrobacter freundii PER2 beta lactamase [AID405083, Type: Literature]PER-2 beta-lactamase [Citrobacter freundii] [gi:695212376]
View
2
[SID103168543]
Kd 0.4Kd for TEM-1 beta-lactamase [AID218698, Type: confirmatory]
View
3
[SID144205100]
qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway: Summary [AID720725, Type: summary]glucocorticoid receptor [Homo sapiens] [gi:311348376]
View
4
[SID103168543]
Partition ratio between Kcat (for beta lactamase) and Kinact (for beta lactamase) was determined [AID231063, Type: other]
View
5
[SID103168543]
Effect on rate of recovery of TEM-2 beta lactamase from transient inhibition [AID44088, Type: other]
View
6
[SID144205100]
Potency-Replicate_1 qHTS assay for small molecule agonists of the p53 signaling pathway - cell viability [AID651633, Type: confirmatory]
View
7
[SID144205100]
Potency qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID720533, Type: confirmatory]
View
8
[SID144205100]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway - cell viability counter screen [AID743033, Type: confirmatory]
View
9
[SID144205100]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line - cell viability counter screen [AID743041, Type: confirmatory]
View
10
[SID144205100]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the thyroid receptor (TR) signaling pathway - cell viability counter screen [AID743064, Type: confirmatory]
View
11
[SID144205100]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway - cell viability counter screen [AID720693, Type: confirmatory]
View
12
[SID144205100]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line - cell viability counter screen [AID743081, Type: confirmatory]
View
13
[SID144205100]
Potency-Replicate_1 qHTS assay to identify aromatase inhibitors - cell viability counter screen [AID743084, Type: confirmatory]
View
14
[SID144205100]
Potency-Replicate_1 qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway - cell viability counter screen [AID743086, Type: confirmatory]
View
15
[SID144205100]
Potency qHTS Assay for Identifying Gametocytocidal Compounds [AID743244, Type: confirmatory]
View
16
[SID144205100]
Potency-Replicate_1 qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rad54/Ku70 mutant cell line [AID743015, Type: confirmatory]
View
17
[SID144205100]
Potency-Replicate_1 qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rev3 mutant cell line [AID743014, Type: confirmatory]
View
18
[SID144205100]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the estrogen receptor alpha (ER-alpha) signaling pathway - cell viability counter screen [AID743074, Type: confirmatory]
View
19
[SID144205100]
Potency-Replicate_1 qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - wild type cell line [AID743012, Type: confirmatory]
View
20
[SID144205100]
Potency-Replicate_1 qHTS assay for small molecules that induce genotoxicity in human embryonic kidney cells expressing luciferase-tagged ATAD5 - cell viability [AID651634, Type: confirmatory]
View