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CHEMBL9306 (CID 23714647) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
Inactive(62)
 
 
Inconclusive(6)
 
 
Unspecified(2)
 
 
Top Targets:
NR LBD AR(7)
 
 
 
NR LBD ER(7)
 
 
NR LBD GR(4)
 
 
 
NR LBD TR(3)
 
 
PAS(2)
 
 
BioAssay Types:
Confirmatory(53)
 
 
 
 
Summary(15)
 
 
 
 
Screening(2)
 
 
Literature(1)
 
 
BioActivity Types:
Potency(65)
 
 
 
Kd(1)
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 73    Data Row: 73   Total Pages: 4   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103168543]
IC50 0.068Inhibition of Citrobacter freundii PER2 beta lactamase [AID405083, Type: Literature]PER-2 beta-lactamase [Citrobacter freundii] [gi:124248221]
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2
[SID103168543]
Kd 0.4Kd for TEM-1 beta-lactamase [AID218698, Type: confirmatory]
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3
[SID144205100]
qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway: Summary [AID720725, Type: summary]glucocorticoid receptor [Homo sapiens] [gi:311348376]
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4
[SID103168543]
Effect on rate of recovery of TEM-2 beta lactamase from transient inhibition [AID44088, Type: other]
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5
[SID103168543]
Partition ratio between Kcat (for beta lactamase) and Kinact (for beta lactamase) was determined [AID231063, Type: other]
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6
[SID144205100]
Potency-Replicate_1 qHTS assay for small molecule agonists of the p53 signaling pathway - cell viability [AID651633, Type: confirmatory]
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7
[SID144205100]
Potency-Replicate_1 qHTS assay for small molecules that induce genotoxicity in human embryonic kidney cells expressing luciferase-tagged ATAD5 - cell viability [AID651634, Type: confirmatory]
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8
[SID144205100]
Potency qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID720533, Type: confirmatory]
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9
[SID144205100]
Potency-Replicate_1 qHTS assay for small molecule disruptors of the mitochondrial membrane potential - cell viability [AID720634, Type: confirmatory]
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10
[SID144205100]
Potency-Replicate_1 qHTS assay for small molecule disruptors of the mitochondrial membrane potential [AID720635, Type: confirmatory]
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11
[SID144205100]
Ratio Potency (uM) qHTS assay for small molecule disruptors of the mitochondrial membrane potential: Summary [AID720637, Type: summary]
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12
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 590 nm (red) in HepG2 cells [AID720674, Type: confirmatory]
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13
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 535 nm (green) in HepG2 cells [AID720675, Type: confirmatory]
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14
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 460 nm (blue) in HEK293 cells [AID720678, Type: confirmatory]
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15
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 590 nm (red) in HEK293 cells [AID720679, Type: confirmatory]
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16
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 535 nm (green) in HEK293 cells [AID720680, Type: confirmatory]
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17
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 460 nm (blue) in HEK293 cell free culture [AID720681, Type: confirmatory]
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18
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 535 nm (green) in HEK293 cell free culture [AID720682, Type: confirmatory]
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19
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 590 nm (red) in HEK293 cell free culture [AID720683, Type: confirmatory]
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20
[SID144205100]
Potency-Replicate_1 qHTS assay to test for compound auto fluorescence at 590 nm (red) in HepG2 cell free culture [AID720684, Type: confirmatory]
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