| 1 | [SID14741546] | Active | Potency | 8.9125 | qHTS Assay for Identifying the Cell-Membrane Permeable IMPase Inhibitors: Potentiation with Lithium [AID1457, Type: confirmatory] | Inositol monophosphatase [gi:44888968] |  View X | Row No. | 1 | | Structure | 
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | Potency | 8.9125 [uM] | | BioAssay | qHTS Assay for Identifying the Cell-Membrane Permeable IMPase Inhibitors: Potentiation with Lithium | | AID | 1457 | | BioAssay type | confirmatory | | Target | Inositol monophosphatase [gi:44888968] | | PubMed | | | Data Table | |
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| 2 | [SID14741546] | Active | Potency | 8.9125 | qHTS Assay for Identifying the Cell-Membrane Permeable IMPase Inhibitors: Potentiation with Lithium [AID1457, Type: confirmatory] | Inositol monophosphatase [gi:44888968] | View X | Row No. | 2 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | Potency | 8.9125 [uM] | | BioAssay | qHTS Assay for Identifying the Cell-Membrane Permeable IMPase Inhibitors: Potentiation with Lithium | | AID | 1457 | | BioAssay type | confirmatory | | Target | Inositol monophosphatase [gi:44888968] | | PubMed | | | Data Table | |
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| 3 | [SID14741546] | Active | Potency | 15.8489 | qHTS Assay for Agonists of the Relaxin Receptor RXFP1 [AID2676, Type: confirmatory] | relaxin receptor 1 isoform 1 [Homo sapiens] [gi:85986601] | View X | Row No. | 3 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | Potency | 15.8489 [uM] | | BioAssay | qHTS Assay for Agonists of the Relaxin Receptor RXFP1 | | AID | 2676 | | BioAssay type | confirmatory | | Target | relaxin receptor 1 isoform 1 [Homo sapiens] [gi:85986601] | | PubMed | | | Data Table | |
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| 4 | [SID14741546] | Active | Potency | 15.8489 | qHTS Assay for Agonists of the Relaxin Receptor RXFP1 [AID2676, Type: confirmatory] | relaxin receptor 1 isoform 1 [Homo sapiens] [gi:85986601] | View X | Row No. | 4 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | Potency | 15.8489 [uM] | | BioAssay | qHTS Assay for Agonists of the Relaxin Receptor RXFP1 | | AID | 2676 | | BioAssay type | confirmatory | | Target | relaxin receptor 1 isoform 1 [Homo sapiens] [gi:85986601] | | PubMed | | | Data Table | |
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| 5 | [SID14741546] | Active | | | Counterscreen for discovery of small molecules that bind to the HIV-1-gp120 binding antibody, PG9: TR-FRET-based biochemical high throughput assay to identify small molecules that bind to the control antibody, PGV04, which binds to a site on the HIV envelope different from the PG9 binding site [AID651604, Type: screening] | Envelope surface glycoprotein gp160, precursor [Human immunodeficiency virus 1] [gi:9629363] | View X | Row No. | 5 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Counterscreen for discovery of small molecules that bind to the HIV-1-gp120 binding antibody, PG9: TR-FRET-based biochemical high throughput assay to identify small molecules that bind to the control antibody, PGV04, which binds to a site on the HIV envelope different from the PG9 binding site | | AID | 651604 | | BioAssay type | screening | | Target | Envelope surface glycoprotein gp160, precursor [Human immunodeficiency virus 1] [gi:9629363] | | PubMed | | | Data Table | |
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| 6 | [SID14741546] | Active | | | TRFRET-based biochemical primary high throughput screening assay to identify small molecules that bind to the HIV-1-gp120 binding antibody, PG9 [AID624416, Type: screening] | Envelope surface glycoprotein gp160, precursor [Human immunodeficiency virus 1] [gi:9629363] | View X | Row No. | 6 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | TRFRET-based biochemical primary high throughput screening assay to identify small molecules that bind to the HIV-1-gp120 binding antibody, PG9 | | AID | 624416 | | BioAssay type | screening | | Target | Envelope surface glycoprotein gp160, precursor [Human immunodeficiency virus 1] [gi:9629363] | | PubMed | | | Data Table | |
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| 7 | [SID14741546] | Active | | | TRFRET-based biochemical high throughput confirmation assay for small molecules that bind to the HIV-1-gp120 binding antibody, PG9 [AID651571, Type: screening] | Envelope surface glycoprotein gp160, precursor [Human immunodeficiency virus 1] [gi:9629363] | View X | Row No. | 7 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | TRFRET-based biochemical high throughput confirmation assay for small molecules that bind to the HIV-1-gp120 binding antibody, PG9 | | AID | 651571 | | BioAssay type | screening | | Target | Envelope surface glycoprotein gp160, precursor [Human immunodeficiency virus 1] [gi:9629363] | | PubMed | | | Data Table | |
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| 8 | [SID14741546] | Active | | | Modulators of the EP2 prostaglandin E2 receptor - Primary Screening [AID940, Type: screening] | prostaglandin E receptor 2 (subtype EP2), 53kDa [Homo sapiens] [gi:31881630] | View X | Row No. | 8 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Modulators of the EP2 prostaglandin E2 receptor - Primary Screening | | AID | 940 | | BioAssay type | screening | | Target | prostaglandin E receptor 2 (subtype EP2), 53kDa [Homo sapiens] [gi:31881630] | | PubMed | | | Data Table | |
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| 9 | [SID14741546] | Active | | | Modulators of the EP2 prostaglandin E2 receptor - Primary Screening [AID940, Type: screening] | prostaglandin E receptor 2 (subtype EP2), 53kDa [Homo sapiens] [gi:31881630] | View X | Row No. | 9 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Modulators of the EP2 prostaglandin E2 receptor - Primary Screening | | AID | 940 | | BioAssay type | screening | | Target | prostaglandin E receptor 2 (subtype EP2), 53kDa [Homo sapiens] [gi:31881630] | | PubMed | | | Data Table | |
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| 10 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 10 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 11 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 11 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 12 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 12 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 13 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 13 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 14 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1032, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 14 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1032 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 15 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1032, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 15 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1032 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
|
| 16 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1032, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 16 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1032 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 17 | [SID14741546] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1032, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 17 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1032 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 18 | [SID14741546] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 18 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 19 | [SID14741546] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 19 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 20 | [SID14741546] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 20 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
|
| 21 | [SID14741546] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 21 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 22 | [SID14741546] | Unspecified | | | Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening] | metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471] | View X | Row No. | 22 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Unspecified | | BioAssay | Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening | | AID | 488969 | | BioAssay type | screening | | Target | metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471] | | PubMed | | | Data Table | |
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| 23 | [SID14741546] | Unspecified | | | Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening] | metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471] | View X | Row No. | 23 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Unspecified | | BioAssay | Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening | | AID | 488969 | | BioAssay type | screening | | Target | metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471] | | PubMed | | | Data Table | |
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| 24 | [SID14741546] | Unspecified | | | Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening] | metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471] | View X | Row No. | 24 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Unspecified | | BioAssay | Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening | | AID | 488969 | | BioAssay type | screening | | Target | metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471] | | PubMed | | | Data Table | |
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| 25 | [SID14741546] | Inactive | Potency | 14.7157 | Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation [AID504834, Type: confirmatory] | | View X | Row No. | 25 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | 14.7157 [uM] | | BioAssay | Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation | | AID | 504834 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 26 | [SID14741546] | Inactive | Potency | 19.9526 | qHTS Assay for Inhibitors of Influenza NS1 Protein Function [AID2326, Type: confirmatory] | nonstructural protein 1 [Influenza A virus (A/WSN/1933(H1N1))] [gi:194352380] | View X | Row No. | 26 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | 19.9526 [uM] | | BioAssay | qHTS Assay for Inhibitors of Influenza NS1 Protein Function | | AID | 2326 | | BioAssay type | confirmatory | | Target | nonstructural protein 1 [Influenza A virus (A/WSN/1933(H1N1))] [gi:194352380] | | PubMed | | | Data Table | |
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| 27 | [SID14741546] | Inactive | Potency | | qHTS Assay for Inhibitors of Leishmania Mexicana Pyruvate Kinase (LmPK) [AID1721, Type: confirmatory] | pyruvate kinase [Leishmania mexicana mexicana] [gi:290753097] | View X | Row No. | 27 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Leishmania Mexicana Pyruvate Kinase (LmPK) | | AID | 1721 | | BioAssay type | confirmatory | | Target | pyruvate kinase [Leishmania mexicana mexicana] [gi:290753097] | | PubMed | | | Data Table | |
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| 28 | [SID14741546] | Inactive | Potency | | qHTS Assay for Activators of Leishmania Mexicana Pyruvate Kinase (LmPK) [AID1722, Type: confirmatory] | pyruvate kinase [Leishmania mexicana mexicana] [gi:290753097] | View X | Row No. | 28 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Activators of Leishmania Mexicana Pyruvate Kinase (LmPK) | | AID | 1722 | | BioAssay type | confirmatory | | Target | pyruvate kinase [Leishmania mexicana mexicana] [gi:290753097] | | PubMed | | | Data Table | |
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| 29 | [SID14741546] | Inactive | Potency | | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor [AID492947, Type: confirmatory] | ADRB2 gene product [Homo sapiens] [gi:4501969] | View X | Row No. | 29 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor | | AID | 492947 | | BioAssay type | confirmatory | | Target | ADRB2 gene product [Homo sapiens] [gi:4501969] | | PubMed | | | Data Table | |
|
| 30 | [SID14741546] | Inactive | Potency | | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor [AID492947, Type: confirmatory] | ADRB2 gene product [Homo sapiens] [gi:4501969] | View X | Row No. | 30 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor | | AID | 492947 | | BioAssay type | confirmatory | | Target | ADRB2 gene product [Homo sapiens] [gi:4501969] | | PubMed | | | Data Table | |
|
| 31 | [SID14741546] | Inactive | Potency | | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor [AID492947, Type: confirmatory] | ADRB2 gene product [Homo sapiens] [gi:4501969] | View X | Row No. | 31 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor | | AID | 492947 | | BioAssay type | confirmatory | | Target | ADRB2 gene product [Homo sapiens] [gi:4501969] | | PubMed | | | Data Table | |
|
| 32 | [SID14741546] | Inactive | Potency | | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor [AID492947, Type: confirmatory] | ADRB2 gene product [Homo sapiens] [gi:4501969] | View X | Row No. | 32 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor | | AID | 492947 | | BioAssay type | confirmatory | | Target | ADRB2 gene product [Homo sapiens] [gi:4501969] | | PubMed | | | Data Table | |
|
| 33 | [SID14741546] | Inactive | | | uHTS identification of small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay [AID2520, Type: screening] | APLNR gene product [Homo sapiens] [gi:4885057] | View X | Row No. | 33 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | uHTS identification of small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay | | AID | 2520 | | BioAssay type | screening | | Target | APLNR gene product [Homo sapiens] [gi:4885057] | | PubMed | | | Data Table | |
|
| 34 | [SID14741546] | Inactive | | | uHTS identification of small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay [AID2520, Type: screening] | APLNR gene product [Homo sapiens] [gi:4885057] | View X | Row No. | 34 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | uHTS identification of small molecule agonists of the APJ receptor via a luminescent beta-arrestin assay | | AID | 2520 | | BioAssay type | screening | | Target | APLNR gene product [Homo sapiens] [gi:4885057] | | PubMed | | | Data Table | |
|
| 35 | [SID14741546] | Inactive | | | uHTS identification of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2521, Type: screening] | APLNR gene product [Homo sapiens] [gi:4885057] | View X | Row No. | 35 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | uHTS identification of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay | | AID | 2521 | | BioAssay type | screening | | Target | APLNR gene product [Homo sapiens] [gi:4885057] | | PubMed | | | Data Table | |
|
| 36 | [SID14741546] | Inactive | | | uHTS identification of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay [AID2521, Type: screening] | APLNR gene product [Homo sapiens] [gi:4885057] | View X | Row No. | 36 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | uHTS identification of small molecule antagonists of the APJ receptor via a luminescent beta-arrestin assay | | AID | 2521 | | BioAssay type | screening | | Target | APLNR gene product [Homo sapiens] [gi:4885057] | | PubMed | | | Data Table | |
|
| 37 | [SID14741546] | Inactive | | | Luminescence-based cell-based primary high throughput screening assay for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): repression of SF-1 (NR5A1) activated StAR promoter by full-length DAX-1 [AID652010, Type: screening] | NR0B1 gene product [Homo sapiens] [gi:5016090] | View X | Row No. | 37 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Luminescence-based cell-based primary high throughput screening assay for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): repression of SF-1 (NR5A1) activated StAR promoter by full-length DAX-1 | | AID | 652010 | | BioAssay type | screening | | Target | NR0B1 gene product [Homo sapiens] [gi:5016090] | | PubMed | | | Data Table | |
|
| 38 | [SID14741546] | Inactive | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 38 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
|
| 39 | [SID14741546] | Inactive | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 39 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
|
| 40 | [SID14741546] | Inactive | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 40 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
|
| 41 | [SID14741546] | Inactive | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 41 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
|
| 42 | [SID14741546] | Inactive | | | Fluorescence polarization assay for PKD inhibitors [AID797, Type: screening] | serine/threonine-protein kinase D1 [Homo sapiens] [gi:115529463] | View X | Row No. | 42 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Fluorescence polarization assay for PKD inhibitors | | AID | 797 | | BioAssay type | screening | | Target | serine/threonine-protein kinase D1 [Homo sapiens] [gi:115529463] | | PubMed | | | Data Table | |
|
| 43 | [SID14741546] | Inactive | | | Fluorescence polarization assay for PKD inhibitors [AID797, Type: screening] | serine/threonine-protein kinase D1 [Homo sapiens] [gi:115529463] | View X | Row No. | 43 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Fluorescence polarization assay for PKD inhibitors | | AID | 797 | | BioAssay type | screening | | Target | serine/threonine-protein kinase D1 [Homo sapiens] [gi:115529463] | | PubMed | | | Data Table | |
|
| 44 | [SID14741546] | Inactive | | | Fluorescence Intensity-based biochemical primary high throughput screening assay to identify activators of kallikrein-7 (K7) zymogen [AID652039, Type: screening] | KLK7 gene product [Homo sapiens] [gi:21327705] | View X | Row No. | 44 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Fluorescence Intensity-based biochemical primary high throughput screening assay to identify activators of kallikrein-7 (K7) zymogen | | AID | 652039 | | BioAssay type | screening | | Target | KLK7 gene product [Homo sapiens] [gi:21327705] | | PubMed | | | Data Table | |
|
| 45 | [SID14741546] | Inactive | | | Fluorescence Intensity-based biochemical primary high throughput screening assay to identify activators of kallikrein-7 (K7) zymogen [AID652039, Type: screening] | KLK7 gene product [Homo sapiens] [gi:21327705] | View X | Row No. | 45 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Fluorescence Intensity-based biochemical primary high throughput screening assay to identify activators of kallikrein-7 (K7) zymogen | | AID | 652039 | | BioAssay type | screening | | Target | KLK7 gene product [Homo sapiens] [gi:21327705] | | PubMed | | | Data Table | |
|
| 46 | [SID14741546] | Inactive | | | High Content Assay for Compounds that inhibit the Assembly of the Perinucleolar Compartment [AID2417, Type: screening] | polypyrimidine tract-binding protein 1 isoform a [Homo sapiens] [gi:4506243] | View X | Row No. | 46 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | High Content Assay for Compounds that inhibit the Assembly of the Perinucleolar Compartment | | AID | 2417 | | BioAssay type | screening | | Target | polypyrimidine tract-binding protein 1 isoform a [Homo sapiens] [gi:4506243] | | PubMed | | | Data Table | |
|
| 47 | [SID14741546] | Inactive | | | qHTS for Small Molecule Agonists and Allosteric Enhancers of Human TRH Receptor: Primary Screen for Enhancers [AID493056, Type: screening] | thyrotropin-releasing hormone receptor [Homo sapiens] [gi:4507681] | View X | Row No. | 47 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | qHTS for Small Molecule Agonists and Allosteric Enhancers of Human TRH Receptor: Primary Screen for Enhancers | | AID | 493056 | | BioAssay type | screening | | Target | thyrotropin-releasing hormone receptor [Homo sapiens] [gi:4507681] | | PubMed | | | Data Table | |
|
| 48 | [SID14741546] | Inactive | | | qHTS for Small Molecule Agonists and Allosteric Enhancers of Human TRH Receptor: Primary Screen for Agonists. [AID493084, Type: screening] | thyrotropin-releasing hormone receptor [Homo sapiens] [gi:4507681] | View X | Row No. | 48 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | qHTS for Small Molecule Agonists and Allosteric Enhancers of Human TRH Receptor: Primary Screen for Agonists. | | AID | 493084 | | BioAssay type | screening | | Target | thyrotropin-releasing hormone receptor [Homo sapiens] [gi:4507681] | | PubMed | | | Data Table | |
|
| 49 | [SID14741546] | Inactive | | | Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign [AID504810, Type: Literature] | TSHR protein [Homo sapiens] [gi:118341367] |  View X | Row No. | 49 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | | AID | 504810 | | BioAssay type | Literature | | Target | TSHR protein [Homo sapiens] [gi:118341367] | | PubMed | 20427476 | | Data Table | |
|
| 50 | [SID14741546] | Inactive | | | Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign [AID504810, Type: Literature] | TSHR protein [Homo sapiens] [gi:118341367] | View X | Row No. | 50 | | Structure |
| | Substance | | | SID | 14741546 | | CID | 23663723 | | Outcome | Inactive | | BioAssay | Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | | AID | 504810 | | BioAssay type | Literature | | Target | TSHR protein [Homo sapiens] [gi:118341367] | | PubMed | 20427476 | | Data Table | |
|
Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
