2,2',4'-trichloroacetophenone (CID 20250) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(231)
 
 
Inactive(76)
 
 
Inconclusive(23)
 
 
Unspecified(3)
 
 
Top Targets:
NR LBD PPAR(5)
 
 
 
NR LBD TR(4)
 
 
 
P53(3)
 
 
 
NR LBD ROR li..(3)
 
 
 
BRCT(2)
 
 
BioAssay Types:
Confirmatory(155)
 
 
 
 
Screening(4)
 
 
Literature(1)
 
 
BioActivity Types:
Potency(119)
 
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 154    Data Row: 333   Total Pages: 7   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID17389431]
Potency 0.1585qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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2
[SID17389431]
Potency 0.1585qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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3
[SID17389431]
Potency 1.9953Cell Viability - LYMP2-022 [AID987, Type: confirmatory]
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4
[SID17389431]
Potency 2.5119Cell Viability - LYMP2-024 [AID988, Type: confirmatory]
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5
[SID17389431]
Potency 2.5119Cell Viability - LYMP2-010 [AID981, Type: confirmatory]
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6
[SID17389431]
Potency 3.1623Cell Viability - LYMP2-012 [AID982, Type: confirmatory]
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7
[SID17389431]
Potency 3.1623Cell Viability - LYMP2-017 [AID972, Type: confirmatory]
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8
[SID17389431]
Potency 3.1623Cell Viability - LYMP2-018 [AID985, Type: confirmatory]
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9
[SID17389431]
Potency 3.7578qHTS assay to identify small molecules that stimulate interleukin-8 (IL-8) secretion [AID651758, Type: confirmatory]interleukin 8 [Homo sapiens] [gi:186368]
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10
[SID17389431]
Potency 3.7578qHTS assay to identify small molecules that stimulate interleukin-8 (IL-8) secretion [AID651758, Type: confirmatory]interleukin 8 [Homo sapiens] [gi:186368]
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11
[SID17389431]
Potency 3.7578qHTS assay to identify small molecules that stimulate interleukin-8 (IL-8) secretion [AID651758, Type: confirmatory]interleukin 8 [Homo sapiens] [gi:186368]
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12
[SID17389431]
Potency 3.9811Cell Viability - LYMP2-001 [AID921, Type: confirmatory]
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13
[SID17389431]
Potency 3.9811Cell Viability - LYMP2-021 [AID974, Type: confirmatory]
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14
[SID17389431]
Potency 5.0119Cell Viability - LYMP2-014 [AID983, Type: confirmatory]
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15
[SID17389431]
Potency 5.0119Cell Viability - LYMP2-016 [AID984, Type: confirmatory]
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16
[SID17389431]
Potency 5.0119Cell Viability - LYMP2-020 [AID986, Type: confirmatory]
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17
[SID17389431]
Potency 5.0119Cell Viability - LYMP2-007 [AID979, Type: confirmatory]
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18
[SID17389431]
Potency 5.0119Cell Viability - LYMP2-015 [AID971, Type: confirmatory]
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19
[SID17389431]
Potency 5.0119qHTS Assay for Anthrax Lethal Toxin Internalization [AID912, Type: confirmatory]lethal factor [Bacillus anthracis str. A2012] [gi:21392848]
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20
[SID144206797]
Potency 5.9569qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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21
[SID144206797]
Potency 5.9569qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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22
[SID144206797]
Potency 5.9569qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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23
[SID17389431]
Potency 6.3096Cell Viability - LYMP2-023 [AID975, Type: confirmatory]
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24
[SID17389431]
Potency 6.3096Cell Viability - LYMP2-026 [AID989, Type: confirmatory]
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25
[SID17389431]
Potency 6.3096Cell Viability - LYMP2-009 [AID968, Type: confirmatory]
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26
[SID17389431]
Potency 6.3096Cell Viability - LYMP2-011 [AID969, Type: confirmatory]
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27
[SID17389431]
Potency 6.3096Cell Viability - LYMP2-004 [AID966, Type: confirmatory]
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28
[SID144206797]
Potency 6.6838qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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29
[SID144206797]
Potency 6.6838qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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30
[SID144206797]
Potency 6.6838qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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31
[SID17389431]
Potency 7.4978qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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32
[SID17389431]
Potency 7.4978qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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33
[SID17389431]
Potency 7.4978qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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34
[SID17389431]
Potency 7.4978qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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35
[SID17389431]
Potency 7.4978qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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36
[SID17389431]
Potency 7.9433Cell Viability - LYMP2-013 [AID970, Type: confirmatory]
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37
[SID17389431]
Potency 7.9433Cell Viability - LYMP2-019 [AID973, Type: confirmatory]
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38
[SID17389431]
Potency 7.9433MultiTox-Fluor Cytotoxicity Assay - LYMP1-002 - Live Cells [AID955, Type: confirmatory]
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39
[SID17389431]
Potency 7.9433MultiTox-Fluor Cytotoxicity Assay - LYMP1-002 - Dead Cells [AID960, Type: confirmatory]
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40
[SID17389431]
Potency 7.9433Cell Viability - LYMP2-025 [AID976, Type: confirmatory]
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41
[SID17389431]
Potency 7.9433Cell Viability - LYMP2-002 [AID977, Type: confirmatory]
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42
[SID17389431]
Potency 7.9433Cell Viability - LYMP2-006 [AID978, Type: confirmatory]
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43
[SID17389431]
Potency 7.9433Cell Viability - LYMP2-008 [AID980, Type: confirmatory]
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44
[SID17389431]
Potency 8.9125qHTS for inhibitors of ROR gamma transcriptional activity [AID2551, Type: confirmatory]nuclear receptor ROR-gamma [Mus musculus] [gi:188536040]
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45
[SID17389431]
Potency 10MultiTox-Fluor Cytotoxicity Assay - LYMP1-003 - Dead Cells [AID961, Type: confirmatory]
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46
[SID17389431]
Potency 10MultiTox-Fluor Cytotoxicity Assay - LYMP1-001 - Dead Cells [AID946, Type: confirmatory]
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47
[SID17389431]
Potency 10Cell Viability - LYMP2-005 [AID967, Type: confirmatory]
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48
[SID17389431]
Potency 10Cell Viability - LYMP2-003 [AID965, Type: confirmatory]
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49
[SID17389431]
Potency 12.5893MultiTox-Fluor Cytotoxicity Assay - LYMP1-001 - Live Cells [AID947, Type: confirmatory]
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50
[SID144207010]
Potency 13.6854qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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