Bookmark and Share
Agmatine (CID 199) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(11)
 
 
Inactive(281)
 
 
Inconclusive(17)
 
 
Unspecified(24)
 
 
Top Targets:
p450(18)
 
 
 
 
PLDc mTdp1 2(9)
 
 
 
MFS(9)
 
 
HSD10-like SD..(8)
 
 
Tubulin-bindi..(8)
 
 
 
BioAssay Types:
Confirmatory(278)
 
 
 
 
 
Literature(29)
 
 
 
 
Screening(2)
 
 
BioActivity Types:
Potency(231)
 
 
 
 
Ki(7)
 
 
 
IC50(3)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 207    Data Row: 333   Total Pages: 17   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103249647]
Ki 3Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot method [AID419311, Type: Literature]Polyamine oxidase [gi:6225822]
View
2
[SID124879247]
Potency 6.6838qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
View
3
[SID124879247]
Potency 8.4144qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
View
4
[SID103249647]
Ki 31.7Inhibition of Wistar rat alpha-2 adrenergic receptor [AID552777, Type: Literature]
View
5
[SID103249647]
Ki 31.7Displacement of [3H]RX821002 from alpha2 adrenoceptor in Wistar rat kidney by liquid scintillation counting [AID371650, Type: Literature]
View
6
[SID103249647]
IC50 36.532Displacement of [3H]clonidine from imidazoline I1 receptor in Wistar rat kidney by liquid scintillation counting [AID371648, Type: Literature]Nischarin [gi:205829312]
View
7
[SID103249647]
IC50 36.532Inhibition of Wistar rat imidazoline I1 receptor [AID552775, Type: Literature]Nischarin [gi:205829312]
View
8
[SID11113734]
qHTS Assay for Tau Filament Binding [AID596, Type: confirmatory]Microtubule-associated protein tau [Homo sapiens] [gi:92096784]
View
9
[SID11113734]
p450-cyp1a2 [AID410, Type: confirmatory]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
View
10
[SID11110769]
qHTS Assay for Spectroscopic Profiling in 4-MU Spectral Region [AID589, Type: other]
View
11
[SID11110769]
qHTS Assay for Spectroscopic Profiling in A350 Spectral Region [AID590, Type: other]
View
12
[SID103249647]
IC50 156In vitro IC50 value by measuring the inhibition of deoxyhypusine synthase. [AID56588, Type: Literature]
View
13
[SID103249647]
Ki 416.7Displacement of [3H]2BFI from imidazoline I2 receptor in Wistar rat brain by liquid scintillation counting [AID371649, Type: Literature]
View
14
[SID103249647]
Ki 416.7Inhibition of Wistar rat imidazoline I2 receptor [AID552776, Type: Literature]
View
15
[SID103249647]
Km 900TP_TRANSPORTER: uptake in OCT3-expressing 293 cells [AID680327, Type: Literature]Solute carrier family 22 member 3 [gi:24212062]
View
16
[SID103249647]
Km 950TP_TRANSPORTER: uptake in OCT2-expressing 293 cells [AID679634, Type: Literature]Solute carrier family 22 member 2 [gi:81872789]
View
17
[SID103249647]
Km 1400TP_TRANSPORTER: uptake in OCT2-expressing 293 cells [AID680367, Type: Literature]Solute carrier family 22 member 2 [gi:313104182]
View
18
[SID103249647]
Km 2500TP_TRANSPORTER: uptake in OCT3-expressing 293 cells [AID681688, Type: Literature]Solute carrier family 22 member 3 [gi:24212063]
View
19
[SID103249647]
Ki 8600TP_TRANSPORTER: inhibition of uptake of 0.1 uM MPP+ in OCT1-expressing 293 cells [AID679198, Type: Literature]Solute carrier family 22 member 1 [gi:81872095]
View
20
[SID103249647]
Ki 24000TP_TRANSPORTER: inhibition of uptake of 0.1 uM MPP+ in OCT1-expressing 293 cells [AID681936, Type: Literature]Solute carrier family 22 member 1 [gi:313104181]
View