AN-329/42612985 (CID 1792197) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(11)
 
 
Inactive(621)
 
 
Inconclusive(7)
 
 
Unspecified(2)
 
 
Top Targets:
7TM GPCR Srx(19)
 
 
alkPPc(12)
 
 
7TM GPCR Srsx(10)
 
 
Bcl-2 like(10)
 
 
G-alpha(6)
 
 
BioAssay Types:
Screening(431)
 
 
 
 
Confirmatory(190)
 
 
 
 
 
Literature(5)
 
 
BioActivity Types:
Potency(131)
 
 
 
 
 
IC50(44)
 
 
EC50(9)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 641    Data Row: 641   Total Pages: 13   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID87225722]
EC50 0.114SAR analysis of selective Agonists of GPR55 using an Image-Based Assay [AID2347, Type: confirmatory]G-protein coupled receptor 55 [Homo sapiens] [gi:33695107]
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2
[SID17407323]
EC50 0.5Image-based HTS for Selective Agonists of GPR55 [AID1961, Type: confirmatory]G-protein coupled receptor 55 [Homo sapiens] [gi:33695107]
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3
[SID17407323]
Potency 3.9811qHTS Assay for Promiscuous and Specific Inhibitors of Cruzain (without detergent) [AID1476, Type: confirmatory]Chain A, Crystal Structure Of Cruzain Covalently Bound To A Purine Nitrile [gi:281307097]
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4
[SID17407323]
Potency 12.5893qHTS for inhibitors of ROR gamma transcriptional activity [AID2551, Type: confirmatory]nuclear receptor ROR-gamma [Mus musculus] [gi:188536040]
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5
[SID17407323]
Potency 23.1093qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]
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6
[SID17407323]
Potency 28.1838qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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7
[SID17407323]
Potency 28.1838qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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8
[SID17407323]
 Leishmania major promastigote HTS [AID1063, Type: screening]
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9
[SID17407323]
 Activator for delta FosB/delta FosB homodimer Measured in Biochemical System Using Plate Reader - 2072-01_Activator_SinglePoint_HTS_Activity [AID493131, Type: screening]protein fosB [Mus musculus] [gi:6679827]
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10
[SID87225722]
 SAR Analysis for the identification of Selective Agonists of GPR55 using an Image-Based Screen [AID463192, Type: other]G-protein coupled receptor 55 [Homo sapiens] [gi:33695107]
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11
[SID87225722]
 SAR analysis of Agonists of GPR55 using MAPK Activation Assay [AID485279, Type: other]G-protein coupled receptor 55 [Homo sapiens] [gi:33695107]
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12
[SID17407323]
 uHTS identification of inhibitors of NadD in a Colorimetric assay [AID602399, Type: screening]hypothetical protein SA1422 [Staphylococcus aureus subsp. aureus N315] [gi:15927174]
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13
[SID17407323]
 Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
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14
[SID17407323]
 Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
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15
[SID17407323]
 Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
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16
[SID17407323]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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17
[SID17407323]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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18
[SID87225722]
IC50 32SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay [AID2338, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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19
[SID87225722]
IC50 32SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay [AID2338, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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20
[SID87225722]
IC50 32SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay [AID2338, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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21
[SID87225722]
IC50 32SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay [AID2340, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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22
[SID87225722]
IC50 32SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay [AID2340, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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23
[SID87225722]
IC50 32SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay [AID2340, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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24
[SID87225722]
IC50 32SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay [AID2339, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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25
[SID87225722]
IC50 32SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay [AID2339, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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26
[SID87225722]
IC50 32SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay [AID2339, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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27
[SID87225722]
IC50 32SAR analysis of agonists of the Cannabinoid Receptor 1 using an Image-Based Assay [AID2341, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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28
[SID87225722]
IC50 32SAR analysis of agonists of the Cannabinoid Receptor 1 using an Image-Based Assay [AID2341, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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29
[SID87225722]
IC50 32SAR analysis of agonists of the Cannabinoid Receptor 1 using an Image-Based Assay [AID2341, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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30
[SID87225722]
IC50 32SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 [AID434922, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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31
[SID87225722]
IC50 32SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 [AID434922, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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32
[SID87225722]
IC50 32SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 [AID434922, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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33
[SID87225722]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 [AID434928, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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34
[SID87225722]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 [AID434928, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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35
[SID87225722]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 2 [AID434928, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
View
36
[SID87225722]
IC50 100SAR VHR1 Fluorescent Assay for In Vitro dose response studies Set 2 [AID2684, Type: confirmatory]dual specificity protein phosphatase 3 [Homo sapiens] [gi:4758208]
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37
[SID87225722]
IC50 100SAR VHR1 Fluorescent Assay for In Vitro dose response studies Set 2 [AID2684, Type: confirmatory]dual specificity protein phosphatase 3 [Homo sapiens] [gi:4758208]
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38
[SID87225722]
IC50 100SAR analysis of chemical inhibitors of HePTP using a Fluorescent assay - Set 2 [AID2678, Type: confirmatory]tyrosine-protein phosphatase non-receptor type 7 isoform 2 [Homo sapiens] [gi:18375660]
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39
[SID87225722]
IC50 100SAR analysis of chemical inhibitors of HePTP using a Fluorescent assay - Set 2 [AID2678, Type: confirmatory]tyrosine-protein phosphatase non-receptor type 7 isoform 2 [Homo sapiens] [gi:18375660]
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40
[SID87225722]
IC50 100SAR analysis of chemical inhibitors of HePTP using a Fluorescent assay - Set 2 [AID2678, Type: confirmatory]tyrosine-protein phosphatase non-receptor type 7 isoform 2 [Homo sapiens] [gi:18375660]
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41
[SID17407323]
 Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 MEK Kinase 2 mutant [AID1530, Type: screening]mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens] [gi:22035600]
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42
[SID17407323]
 Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 MEK Kinase 2 mutant [AID1530, Type: screening]mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens] [gi:22035600]
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43
[SID17407323]
 Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 binding to MEK Kinase 2 Wildtype [AID1531, Type: screening]mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens] [gi:22035600]
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44
[SID17407323]
 Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 binding to MEK Kinase 2 Wildtype [AID1531, Type: screening]mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens] [gi:22035600]
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45
[SID17407323]
 HTS to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac wildtype [AID757, Type: screening]Rac1 protein [Homo sapiens] [gi:8574038]
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46
[SID17407323]
 HTS to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac wildtype [AID757, Type: screening]Rac1 protein [Homo sapiens] [gi:8574038]
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47
[SID17407323]
 HTS to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac activated mutant [AID764, Type: screening]Rac1 protein [Homo sapiens] [gi:8574038]
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48
[SID17407323]
 HTS to identify specific small molecule inhibitors of Ras and Ras-related GTPases specifically Rac activated mutant [AID764, Type: screening]Rac1 protein [Homo sapiens] [gi:8574038]
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49
[SID17407323]
 Homologous recombination - Rad 51 [AID1385, Type: screening]RAD51 [Homo sapiens] [gi:49168602]
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50
[SID17407323]
 Homologous recombination - Rad 51 [AID1385, Type: screening]RAD51 [Homo sapiens] [gi:49168602]
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