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BioActivity Data for Compound MLS000438623 (CID 16745748)

BioActivity Outcomes:
Active(5)
 
 
Inactive(255)
 
 
Inconclusive(18)
 
 
Top Targets:
7tm 4(12)
 
 
Pyruvate Kina..(8)
 
 
G-alpha(7)
 
 
 
TRP 2(5)
 
 
GH27(4)
 
 
BioAssay Types:
Confirmatory(150)
 
 
 
 
Screening(123)
 
 
 
 
Literature(2)
 
 
BioAssay Categories:
Organism-base..(4)
 
 
Biochemical(2)
 
 
Toxicity(1)
 
 
Cell-based(19)
 
 
BioActivity Types:
Potency(110)
 
 
 
 
IC50(26)
 
 
 
EC50(6)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 225    Data Row: 278   Total Pages: 14   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID26756132]
Potency 3.9811qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E) [AID2147, Type: confirmatory]Chain A, Crystal Structure Of The Human 2-Oxoglutarate Oxygenase Loc390245 [gi:221046486]
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2
[SID26725526]
IC50 uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (PABP) [AID2014, Type: confirmatory]polyadenylate-binding protein 1 [Homo sapiens] [gi:46367787]
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3
[SID26725526]
qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen [AID2472, Type: screening]glyceraldehyde-3-phosphate dehydrogenase isoform 1 [Homo sapiens] [gi:7669492]
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4
[SID26756132]
qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen [AID2472, Type: screening]glyceraldehyde-3-phosphate dehydrogenase isoform 1 [Homo sapiens] [gi:7669492]
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5
[SID26725526]
Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 binding to MEK Kinase 2 Wildtype [AID1531, Type: screening]mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens] [gi:22035600]
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6
[SID104233240]
Potency 0.0027qHTS for Inhibitors of binding or entry into cells for Marburg Virus [AID720532, Type: confirmatory]gene 4 small orf - Marburg virus [Marburg marburgvirus] [gi:420597]
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7
[SID26725526]
Heat Shock Factor-1 (HSF-1) Measured in Cell-Based System Using Plate Reader - 2038-01_Activator_SinglePoint_HTS_Activity [AID504408, Type: screening]
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8
[SID26756132]
Potency qHTS for Inhibitors of Plasmodium falciparum (DD2) proliferation [AID504314, Type: confirmatory]
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9
[SID26756132]
Potency qHTS for Inhibitors of Plasmodium falciparum (GB4) proliferation [AID504315, Type: confirmatory]
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10
[SID104233240]
Potency qHTS for Inhibitors of Plasmodium falciparum (GB4) proliferation [AID504315, Type: confirmatory]
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11
[SID104233240]
Potency qHTS for Inhibitors of Plasmodium falciparum (7G8) proliferation [AID504316, Type: confirmatory]
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12
[SID104233240]
Potency qHTS for Inhibitors of Plasmodium falciparum (HB3) proliferation [AID504318, Type: confirmatory]
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13
[SID104233240]
Potency qHTS for Inhibitors of Plasmodium falciparum (CP250) proliferation [AID504320, Type: confirmatory]
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14
[SID104233240]
Potency qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID540256, Type: confirmatory]
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15
[SID26756132]
Potency qHTS for Inhibitors of Plasmodium falciparum (7G8) proliferation [AID504316, Type: confirmatory]
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16
[SID26756132]
Potency qHTS for Inhibitors of Plasmodium falciparum (HB3) proliferation [AID504318, Type: confirmatory]
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17
[SID26756132]
Potency qHTS for Inhibitors of Plasmodium falciparum (CP250) proliferation [AID504320, Type: confirmatory]
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18
[SID104233240]
Potency qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID720533, Type: confirmatory]
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19
[SID26725526]
Potency qHTS profiling assay for firefly luciferase inhibitor/activator using purifed enzyme and Km concentrations of substrates (counterscreen for miR-21 project) [AID588342, Type: confirmatory]Luciferase [Photinus pyralis] [gi:160794]
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20
[SID26725526]
Factor XIa 1536 HTS [AID798, Type: screening]coagulation factor XI [Homo sapiens] [gi:180352]
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