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TG101348 (CID 16722836) - Compound BioActivity Data
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BioActivity Outcomes:
Active(329)
 
 
Inactive(17)
 
 
Inconclusive(1)
 
 
Unspecified(119)
 
 
Top Targets:
PKc(48)
 
 
 
PKc like(40)
 
 
 
STKc AGC(17)
 
 
 
PTKc Abl(16)
 
 
PTKc EGFR(12)
 
 
 
BioAssay Types:
Literature(447)
 
 
 
 
Confirmatory(18)
 
 
 
 
BioActivity Types:
Kd(442)
 
 
 
Potency(20)
 
 
 
 
IC50(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 466    Data Row: 466   Total Pages: 24   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID123089189]
Kd 0.0011Binding constant for JAK2(JH1domain-catalytic) kinase domain [AID624973, Type: Literature]Tyrosine-protein kinase JAK2 [gi:12643404]
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2
[SID123089189]
Kd 0.0011Binding constant for GAK kinase domain [AID625012, Type: Literature]Cyclin-G-associated kinase [gi:17375734]
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3
[SID123089189]
Kd 0.0012Binding constant for DAPK3 kinase domain [AID624834, Type: Literature]Death-associated protein kinase 3 [gi:38604691]
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4
[SID123089189]
IC50 0.003Inhibition of human recombinant JAK2 by TR-FRET assay [AID538224, Type: Literature]Tyrosine-protein kinase JAK2 [gi:12643404]
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5
[SID123089189]
Kd 0.0049Binding constant for FLT3(D835H) kinase domain [AID624935, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
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6
[SID123089189]
Kd 0.0064Binding constant for FLT3(D835Y) kinase domain [AID624936, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
7
[SID123089189]
Kd 0.0066Binding constant for STK16 kinase domain [AID624775, Type: Literature]Serine/threonine-protein kinase 16 [gi:46577677]
View
8
[SID123089189]
Kd 0.013Binding constant for FLT3 kinase domain [AID624934, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
9
[SID123089189]
Kd 0.013Binding constant for FLT3(K663Q) kinase domain [AID624938, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
10
[SID123089189]
Kd 0.013Binding constant for DCAMKL3 kinase domain [AID624707, Type: Literature]Serine/threonine-protein kinase DCLK3 [gi:115502142]
View
11
[SID123089189]
Kd 0.016Binding constant for FLT3(ITD) kinase domain [AID624937, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
12
[SID123089189]
Kd 0.016Binding constant for DAPK1 kinase domain [AID624971, Type: Literature]Death-associated protein kinase 1 [gi:317373595]
View
13
[SID123089189]
Kd 0.018Binding constant for JAK1(JH1domain-catalytic) kinase domain [AID624859, Type: Literature]Tyrosine-protein kinase JAK1 [gi:215274013]
View
14
[SID123089189]
Kd 0.019Binding constant for YSK4 kinase domain [AID625136, Type: Literature]Mitogen-activated protein kinase kinase kinase 19 [gi:74755104]
View
15
[SID123089189]
Kd 0.02Binding constant for FLT3(N841I) kinase domain [AID624939, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
16
[SID123089189]
Kd 0.021Binding constant for TYK2(JH1domain-catalytic) kinase domain [AID624912, Type: Literature]Non-receptor tyrosine-protein kinase TYK2 [gi:56405328]
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17
[SID123089189]
Kd 0.029Binding constant for DAPK2 kinase domain [AID625077, Type: Literature]Death-associated protein kinase 2 [gi:38605084]
View
18
[SID123089189]
Kd 0.029Binding constant for FLT3(R834Q) kinase domain [AID624940, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
19
[SID123089189]
Kd 0.032Binding constant for BIKE kinase domain [AID625109, Type: Literature]BMP-2-inducible protein kinase [gi:34222653]
View
20
[SID123089189]
Kd 0.034Binding constant for ARK5 kinase domain [AID625088, Type: Literature]NUAK family SNF1-like kinase 1 [gi:14424095]
View