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CHEMBL261515 (CID 16203668) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
Unspecified(4)
 
 
Top Targets:
7tm 4(7)
 
 
 
BioAssay Types:
Literature(7)
 
 
 
BioActivity Types:
Ki(2)
 
 
EC50(2)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 7    Data Row: 7   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103566191]
Ki 0.03Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells [AID281463, Type: Literature]Adenosine receptor A3 [gi:1351831]
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2
[SID103566191]
Ki 0.64Displacement of [3H]CPPA from human adenosine A1 receptor expressed in CHO cells [AID281459, Type: Literature]Adenosine receptor A1 [gi:231473]
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3
[SID103566191]
EC50 3.27Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of cAMP production [AID281466, Type: Literature]Adenosine receptor A2b [gi:112938]
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4
[SID103566191]
EC50 Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of adenylate cyclase [AID330858, Type: Literature]Adenosine receptor A2b [gi:112938]
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5
[SID103566191]
Agonist activity human adenosine A2B receptor expressed in CHO cells assessed as stimulation of adenylate cyclase relative to NECA [AID330859, Type: Literature]Adenosine receptor A2b [gi:112938]
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6
[SID103566191]
Maximum efficacy at human recombinant adenosine A3 receptor expressed in CHO cells assessed as inhibition of cAMP production at 10 uM relative to NECA [AID281469, Type: Literature]Adenosine receptor A3 [gi:1351831]
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7
[SID103566191]
Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cells at 10 uM [AID281462, Type: Literature]Adenosine receptor A2a [gi:543740]
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