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CHEMBL2113271 (CID 16203667) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
Unspecified(2)
 
 
Top Targets:
7TM GPCR Srsx(5)
 
 
 
BioAssay Types:
Literature(5)
 
 
 
BioActivity Types:
Ki(3)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID163319488]
Ki 0.0736Displacement of [3H]CPPA from human adenosine A1 receptor expressed in CHO cells [AID281459, Type: Literature]Adenosine receptor A1 [gi:231473]
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2
[SID163319488]
Ki 0.09Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells [AID281463, Type: Literature]Adenosine receptor A3 [gi:1351831]
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3
[SID163319488]
Ki 0.277Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cells [AID281461, Type: Literature]Adenosine receptor A2a [gi:543740]
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4
[SID163319488]
Maximum efficacy at human recombinant adenosine A3 receptor expressed in CHO cells assessed as inhibition of cAMP production at 10 uM relative to NECA [AID281469, Type: Literature]Adenosine receptor A3 [gi:1351831]
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5
[SID163319488]
Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of cAMP production at 10 uM [AID281467, Type: Literature]Adenosine receptor A2b [gi:112938]
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