| 1 | [SID24823750] | Active | EC50 | 0.458 | Luminescence Cell-Based/Microorganism Dose Confirmation HTS to Identify Inhibitors of T.Cruzi Replication. [AID2044, Type: confirmatory] | |  View X | Row No. | 1 | | Structure | 
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | EC50 | 0.458 [uM] | | BioAssay | Luminescence Cell-Based/Microorganism Dose Confirmation HTS to Identify Inhibitors of T.Cruzi Replication. | | AID | 2044 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 2 | [SID24823750] | Active | Potency | 2.6169 | Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation [AID504832, Type: confirmatory] | | View X | Row No. | 2 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 2.6169 [uM] | | BioAssay | Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation | | AID | 504832 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 3 | [SID24823750] | Active | Potency | 2.8184 | qHTS for inhibitors of ROR gamma transcriptional activity [AID2551, Type: confirmatory] | nuclear receptor ROR-gamma [Mus musculus] [gi:188536040] | View X | Row No. | 3 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 2.8184 [uM] | | BioAssay | qHTS for inhibitors of ROR gamma transcriptional activity | | AID | 2551 | | BioAssay type | confirmatory | | Target | nuclear receptor ROR-gamma [Mus musculus] [gi:188536040] | | PubMed | | | Data Table | |
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| 4 | [SID24823750] | Active | Potency | 4.1475 | Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation [AID504834, Type: confirmatory] | | View X | Row No. | 4 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 4.1475 [uM] | | BioAssay | Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation | | AID | 504834 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 5 | [SID24823750] | Active | Potency | 5.8048 | A quantitative high throughput screen for small molecules that induce DNA re-replication in MCF 10a normal breast cells. [AID624296, Type: confirmatory] | GMNN gene product [Homo sapiens] [gi:7705682] | View X | Row No. | 5 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 5.8048 [uM] | | BioAssay | A quantitative high throughput screen for small molecules that induce DNA re-replication in MCF 10a normal breast cells. | | AID | 624296 | | BioAssay type | confirmatory | | Target | GMNN gene product [Homo sapiens] [gi:7705682] | | PubMed | | | Data Table | |
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| 6 | [SID24823750] | Active | Potency | 14.581 | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory] | TDP1 protein [Homo sapiens] [gi:79154014] | View X | Row No. | 6 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 14.581 [uM] | | BioAssay | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT | | AID | 686978 | | BioAssay type | confirmatory | | Target | TDP1 protein [Homo sapiens] [gi:79154014] | | PubMed | | | Data Table | |
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| 7 | [SID24823750] | Active | Potency | 14.581 | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory] | TDP1 protein [Homo sapiens] [gi:79154014] | View X | Row No. | 7 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 14.581 [uM] | | BioAssay | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT | | AID | 686978 | | BioAssay type | confirmatory | | Target | TDP1 protein [Homo sapiens] [gi:79154014] | | PubMed | | | Data Table | |
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| 8 | [SID24823750] | Active | Potency | 14.581 | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory] | TDP1 protein [Homo sapiens] [gi:79154014] | View X | Row No. | 8 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 14.581 [uM] | | BioAssay | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT | | AID | 686978 | | BioAssay type | confirmatory | | Target | TDP1 protein [Homo sapiens] [gi:79154014] | | PubMed | | | Data Table | |
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| 9 | [SID24823750] | Active | Potency | 39.8107 | qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory] | euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070] | View X | Row No. | 9 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | Potency | 39.8107 [uM] | | BioAssay | qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a | | AID | 504332 | | BioAssay type | confirmatory | | Target | euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070] | | PubMed | | | Data Table | |
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| 10 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1048, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 10 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1048 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 11 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1048, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 11 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1048 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 12 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1048, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 12 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1048 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 13 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1048, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 13 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1048 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 14 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 14 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 15 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 15 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 16 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 16 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 17 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1049, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 17 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 2 (SRC-2) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1049 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 18 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1051, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 18 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1051 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 19 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1051, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 19 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1051 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 20 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1051, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 20 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1051 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 21 | [SID24823750] | Active | | | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID1051, Type: other] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 21 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Measurement of TR-FRET detection format artefact in the screen for agonists of steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 1051 | | BioAssay type | other | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 22 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 22 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 23 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 23 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 24 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 24 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 25 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID731, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 25 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 3 (SRC-3) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 731 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 26 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 26 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 27 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 27 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 28 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 28 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 29 | [SID24823750] | Active | | | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) [AID631, Type: screening] | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | View X | Row No. | 29 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Primary biochemical High Throughput Screening assay for agonists of the steroid receptor coactivator 1 (SRC-1) recruitment by the peroxisome proliferator-activated receptor gamma (PPARgamma) | | AID | 631 | | BioAssay type | screening | | Target | peroxisome proliferator-activated receptor gamma isoform 2 [Homo sapiens] [gi:20336229] | | PubMed | | | Data Table | |
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| 30 | [SID24823750] | Active | | | Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput primary assay to identify inhibitors of Protein Phosphatase 1 (PP1). [AID2235, Type: screening] | PPP1CA gene product [Homo sapiens] [gi:56790945] | View X | Row No. | 30 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput primary assay to identify inhibitors of Protein Phosphatase 1 (PP1). | | AID | 2235 | | BioAssay type | screening | | Target | PPP1CA gene product [Homo sapiens] [gi:56790945] | | PubMed | | | Data Table | |
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| 31 | [SID24823750] | Active | | | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) [AID463082, Type: screening] | PLA2G7 gene product [Homo sapiens] [gi:270133071] | View X | Row No. | 31 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) | | AID | 463082 | | BioAssay type | screening | | Target | PLA2G7 gene product [Homo sapiens] [gi:270133071] | | PubMed | | | Data Table | |
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| 32 | [SID24823750] | Active | | | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) [AID463082, Type: screening] | PLA2G7 gene product [Homo sapiens] [gi:270133071] | View X | Row No. | 32 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of the plasma platelet activating factor acetylhydrolase (pPAFAH) | | AID | 463082 | | BioAssay type | screening | | Target | PLA2G7 gene product [Homo sapiens] [gi:270133071] | | PubMed | | | Data Table | |
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| 33 | [SID24823750] | Active | | | Leishmania major promastigote HTS [AID1063, Type: screening] | | View X | Row No. | 33 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Leishmania major promastigote HTS | | AID | 1063 | | BioAssay type | screening | | Target | | | PubMed | | | Data Table | |
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| 34 | [SID24823750] | Active | | | Luminescence Cell-Based/Microorganism Primary HTS to Identify Inhibitors of T.Cruzi Replication [AID1885, Type: screening] | | View X | Row No. | 34 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Luminescence Cell-Based/Microorganism Primary HTS to Identify Inhibitors of T.Cruzi Replication | | AID | 1885 | | BioAssay type | screening | | Target | | | PubMed | | | Data Table | |
|
| 35 | [SID24823750] | Active | | | Screen for Chemicals that Inhibit the RAM Network [AID868, Type: screening] | | View X | Row No. | 35 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | Screen for Chemicals that Inhibit the RAM Network | | AID | 868 | | BioAssay type | screening | | Target | | | PubMed | | | Data Table | |
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| 36 | [SID24823750] | Active | | | TR-FRET-based primary biochemical high-throughput screening assay to identify inhibitors of Hepatitis C Virus (HCV) core protein dimerization [AID1899, Type: screening] | core protein [Hepatitis C virus] [gi:83779224] | View X | Row No. | 36 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | TR-FRET-based primary biochemical high-throughput screening assay to identify inhibitors of Hepatitis C Virus (HCV) core protein dimerization | | AID | 1899 | | BioAssay type | screening | | Target | core protein [Hepatitis C virus] [gi:83779224] | | PubMed | | | Data Table | |
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| 37 | [SID24823750] | Active | | | uHTS identification of inhibitors of NadD in a Colorimetric assay [AID602399, Type: screening] | hypothetical protein SA1422 [Staphylococcus aureus subsp. aureus N315] [gi:15927174] | View X | Row No. | 37 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Active | | BioAssay | uHTS identification of inhibitors of NadD in a Colorimetric assay | | AID | 602399 | | BioAssay type | screening | | Target | hypothetical protein SA1422 [Staphylococcus aureus subsp. aureus N315] [gi:15927174] | | PubMed | | | Data Table | |
|
| 38 | [SID24823750] | Unspecified | Potency | | qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory] | acid sphingomyelinase [Homo sapiens] [gi:179095] | View X | Row No. | 38 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Unspecified | | Potency | [uM] | | BioAssay | qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate | | AID | 624178 | | BioAssay type | confirmatory | | Target | acid sphingomyelinase [Homo sapiens] [gi:179095] | | PubMed | | | Data Table | |
|
| 39 | [SID24823750] | Unspecified | Potency | | qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory] | acid sphingomyelinase [Homo sapiens] [gi:179095] | View X | Row No. | 39 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Unspecified | | Potency | [uM] | | BioAssay | qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate | | AID | 624178 | | BioAssay type | confirmatory | | Target | acid sphingomyelinase [Homo sapiens] [gi:179095] | | PubMed | | | Data Table | |
|
| 40 | [SID24823750] | Unspecified | Potency | | qHTS Assay for Enhancers of SMN2 Splice Variant Expression [AID1458, Type: confirmatory] | survival motor neuron protein isoform d [Homo sapiens] [gi:10937869] | View X | Row No. | 40 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Unspecified | | Potency | [uM] | | BioAssay | qHTS Assay for Enhancers of SMN2 Splice Variant Expression | | AID | 1458 | | BioAssay type | confirmatory | | Target | survival motor neuron protein isoform d [Homo sapiens] [gi:10937869] | | PubMed | | | Data Table | |
|
| 41 | [SID24823750] | Unspecified | Potency | | qHTS Assay for Enhancers of SMN2 Splice Variant Expression [AID1458, Type: confirmatory] | survival motor neuron protein isoform d [Homo sapiens] [gi:10937869] | View X | Row No. | 41 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Unspecified | | Potency | [uM] | | BioAssay | qHTS Assay for Enhancers of SMN2 Splice Variant Expression | | AID | 1458 | | BioAssay type | confirmatory | | Target | survival motor neuron protein isoform d [Homo sapiens] [gi:10937869] | | PubMed | | | Data Table | |
|
| 42 | [SID24823750] | Inactive | Potency | 5.2119 | qHTS Assay for Modulators of miRNAs and/orActivators of miR-21 [AID2288, Type: confirmatory] | | View X | Row No. | 42 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | Potency | 5.2119 [uM] | | BioAssay | qHTS Assay for Modulators of miRNAs and/orActivators of miR-21 | | AID | 2288 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
|
| 43 | [SID24823750] | Inactive | Potency | 25.1189 | Inhibitors of Secretory Acid Sphingomyelinase (S-ASM): qHTS [AID504937, Type: confirmatory] | acid sphingomyelinase [Homo sapiens] [gi:179095] | View X | Row No. | 43 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | Potency | 25.1189 [uM] | | BioAssay | Inhibitors of Secretory Acid Sphingomyelinase (S-ASM): qHTS | | AID | 504937 | | BioAssay type | confirmatory | | Target | acid sphingomyelinase [Homo sapiens] [gi:179095] | | PubMed | | | Data Table | |
|
| 44 | [SID24823750] | Inactive | Potency | 25.1189 | Inhibitors of Secretory Acid Sphingomyelinase (S-ASM): qHTS [AID504937, Type: confirmatory] | acid sphingomyelinase [Homo sapiens] [gi:179095] | View X | Row No. | 44 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | Potency | 25.1189 [uM] | | BioAssay | Inhibitors of Secretory Acid Sphingomyelinase (S-ASM): qHTS | | AID | 504937 | | BioAssay type | confirmatory | | Target | acid sphingomyelinase [Homo sapiens] [gi:179095] | | PubMed | | | Data Table | |
|
| 45 | [SID24823750] | Inactive | Potency | 31.6228 | qHTS for Inhibitors of ATXN expression [AID651635, Type: confirmatory] | ATXN2 gene product [Homo sapiens] [gi:171543895] | View X | Row No. | 45 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | Potency | 31.6228 [uM] | | BioAssay | qHTS for Inhibitors of ATXN expression | | AID | 651635 | | BioAssay type | confirmatory | | Target | ATXN2 gene product [Homo sapiens] [gi:171543895] | | PubMed | | | Data Table | |
|
| 46 | [SID24823750] | Inactive | EC50 | 60 | Luminescence Cell-Based Dose Response HTS Screen to Identify Cytotoxic Compounds of NIH3T3 cells. [AID2010, Type: confirmatory] | | View X | Row No. | 46 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | EC50 | 60 [uM] | | BioAssay | Luminescence Cell-Based Dose Response HTS Screen to Identify Cytotoxic Compounds of NIH3T3 cells. | | AID | 2010 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
|
| 47 | [SID24823750] | Inactive | Potency | 89.1251 | qHTS for Inhibitors of Polymerase Iota [AID588590, Type: confirmatory] | DNA polymerase iota [Homo sapiens] [gi:154350220] | View X | Row No. | 47 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | Potency | 89.1251 [uM] | | BioAssay | qHTS for Inhibitors of Polymerase Iota | | AID | 588590 | | BioAssay type | confirmatory | | Target | DNA polymerase iota [Homo sapiens] [gi:154350220] | | PubMed | | | Data Table | |
|
| 48 | [SID24823750] | Inactive | Potency | 89.1251 | qHTS for Inhibitors of Polymerase Iota [AID588590, Type: confirmatory] | DNA polymerase iota [Homo sapiens] [gi:154350220] | View X | Row No. | 48 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | Potency | 89.1251 [uM] | | BioAssay | qHTS for Inhibitors of Polymerase Iota | | AID | 588590 | | BioAssay type | confirmatory | | Target | DNA polymerase iota [Homo sapiens] [gi:154350220] | | PubMed | | | Data Table | |
|
| 49 | [SID24823750] | Inactive | Concentration @ Maximum % Inhibition | 100 | Screen for Chemicals that Inhibit the RAM Network - Dose Response with Drug Efflux Deficient Sensitized Control Strain [AID1305, Type: confirmatory] | | View X | Row No. | 49 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | Concentration @ Maximum % Inhibition | 100 [uM] | | BioAssay | Screen for Chemicals that Inhibit the RAM Network - Dose Response with Drug Efflux Deficient Sensitized Control Strain | | AID | 1305 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
|
| 50 | [SID24823750] | Inactive | IC50 | | Screen for Chemicals that Inhibit the RAM Network - Confirmatory Dose Response [AID1307, Type: confirmatory] | | View X | Row No. | 50 | | Structure |
| | Substance | | | SID | 24823750 | | CID | 16195562 | | Outcome | Inactive | | IC50 | [uM] | | BioAssay | Screen for Chemicals that Inhibit the RAM Network - Confirmatory Dose Response | | AID | 1307 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
|
Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
