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Tannins (CID 16129778) - Compound BioActivity Data
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BioActivity Outcomes:
Active(104)
 
 
Inactive(143)
 
 
Inconclusive(72)
 
 
Unspecified(1275)
 
 
Top Targets:
7tm 4(44)
 
 
 
NR LBD ER(16)
 
 
 
 
NR LBD AR(15)
 
 
 
 
 
p450(12)
 
 
 
 
NR LBD PPAR(10)
 
 
 
BioAssay Types:
Confirmatory(286)
 
 
 
 
 
Screening(72)
 
 
 
Literature(57)
 
 
 
 
Summary(39)
 
 
 
 
BioActivity Types:
Potency(192)
 
 
 
 
 
IC50(128)
 
 
 
 
Ki(6)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1526    Data Row: 1594   Total Pages: 80   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID57260395]
Potency 0.0053qHTS Assay for Inhibitors of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1) [AID2517, Type: confirmatory]Chain A, Human Ape1 Endonuclease With Bound Abasic Dna And Mn2+ Ion [gi:6980812]
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2
[SID103600468]
IC50 0.022DRUGMATRIX: Protein Tyrosine Kinase, Fyn enzyme inhibition (substrate: Poly(Glu:Tyr)) [AID625185, Type: confirmatory]Tyrosine-protein kinase Fyn [gi:125370]
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3
[SID103600468]
IC50 0.029Inhibition of H(+)/K(+) ATPase from pig gastric mucosa [AID334756, Type: Literature]
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4
[SID103600468]
IC50 0.079DRUGMATRIX: Protein Tyrosine Kinase, LCK enzyme inhibition (substrate: Poly(Glu:Tyr)) [AID625187, Type: confirmatory]Tyrosine-protein kinase Lck [gi:125474]
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5
[SID57260395]
Potency 0.0953qHTS Assay to Find Inhibitors of T. brucei phosphofructokinase [AID485367, Type: confirmatory]ATP-dependent phosphofructokinase [Trypanosoma brucei brucei strain 927/4 GUTat10.1] [gi:72386991]
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6
[SID57260395]
Potency 0.1qHTS Assay for the Inhibitors of L3MBTL1 [AID485360, Type: confirmatory]lethal(3)malignant brain tumor-like protein 1 isoform I [Homo sapiens] [gi:117938328]
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7
[SID57260395]
IC50 0.16Identification of SV40 T antigen inhibitors: A route to novel anti-viral reagents [AID1903, Type: confirmatory]large T antigen [Simian virus 40] [gi:297591903]
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8
[SID103600468]
IC50 0.185DRUGMATRIX: Protein Serine/Threonine Kinase, ERK2 enzyme inhibition (substrate: Myelin Basic Protein) [AID625181, Type: confirmatory]Mitogen-activated protein kinase 1 [gi:119554]
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9
[SID103600468]
IC50 0.268DRUGMATRIX: Lipoxygenase 15-LO enzyme inhibition (substrate: Linoleic acid) [AID625146, Type: confirmatory]Arachidonate 15-lipoxygenase [gi:126397]
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10
[SID103600468]
IC50 0.325DRUGMATRIX: Thromboxane Synthetase enzyme inhibition (substrate: PGH2) [AID625229, Type: confirmatory]Thromboxane-A synthase [gi:254763392]
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11
[SID103600468]
IC50 0.346DRUGMATRIX: Aldose Reductase enzyme inhibition (substrate: DL-Glyceraldehyde) [AID625208, Type: confirmatory]Aldose reductase [gi:1168407]
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12
[SID144204975]
Potency 0.3534qHTS for Inhibitors of binding or entry into cells for Marburg Virus [AID720532, Type: confirmatory]gene 4 small orf - Marburg virus [Marburg marburgvirus] [gi:420597]
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13
[SID103600468]
IC50 0.375DRUGMATRIX: Protein Serine/Threonine Kinase, p38alpha enzyme inhibition (substrate: Myelin Basic Protein) [AID625182, Type: confirmatory]Mitogen-activated protein kinase 14 [gi:2499600]
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14
[SID103600468]
IC50 0.41Inhibition of K+ dependent pNPPase from pig gastric mucosa [AID334757, Type: Literature]
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15
[SID103600468]
IC50 0.714DRUGMATRIX: Phosphodiesterase PDE3 enzyme inhibition (substrate: [3H]cAMP + cAMP) [AID625165, Type: confirmatory]
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16
[SID57260395]
Potency 0.7943qHTS Assay for Inhibitors of BAZ2B [AID504333, Type: confirmatory]bromodomain adjacent to zinc finger domain 2B [Homo sapiens] [gi:6683500]
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17
[SID103600468]
IC50 0.919DRUGMATRIX: CYP450, 1A2 enzyme inhibition (substrate: 3-Cyano-7-ethoxycoumarin) [AID625245, Type: confirmatory]Cytochrome P450 1A2 [gi:117144]
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18
[SID103600468]
IC50 1.043DRUGMATRIX: Phosphodiesterase PDE4 enzyme inhibition (substrate: [3H]cAMP + cAMP) [AID625166, Type: confirmatory]
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19
[SID103600468]
IC50 1.335DRUGMATRIX: ATPase, Na+/K+ enzyme inhibition (substrate: ATP) [AID625210, Type: confirmatory]
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20
[SID57260395]
Potency 1.4125qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory]euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070]
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