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MLS001199812 (CID 15997213) - Compound BioActivity Data
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BioActivity Outcomes:
Active(20)
 
 
Inactive(530)
 
 
Inconclusive(5)
 
 
Unspecified(1)
 
 
Top Targets:
7TM GPCR Srx(21)
 
 
7TM GPCR Srsx(15)
 
 
CAP ED(5)
 
 
TRP 2(5)
 
 
ABCC CFTR1(4)
 
 
BioAssay Types:
Screening(364)
 
 
Confirmatory(178)
 
 
 
 
 
Literature(5)
 
 
BioActivity Types:
Potency(118)
 
 
 
 
 
IC50(44)
 
 
 
EC50(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 511    Data Row: 556   Total Pages: 12   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144108867]
IC50 Rep 1 0.325A Cell-Based Counter Screen testing Compounds that Inhibit VEEV TC-83, in strain KU V3526 (2) [AID651884, Type: confirmatory]
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2
[SID131341903]
Average IC50 0.37A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, Trinidad Donkey (TrD) (1) [AID602484, Type: confirmatory]
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3
[SID144108867]
IC50 Rep 1 0.557A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, Trinidad Donkey (TrD) (2) [AID651874, Type: confirmatory]
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4
[SID131341903]
IC50 0.67A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV TC-83 (4) [AID624063, Type: confirmatory]
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5
[SID143472910]
Average IC50 0.695A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83 (8) [AID651917, Type: confirmatory]
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6
[SID144108867]
Average IC50 0.81A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83 (7) [AID651734, Type: confirmatory]
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7
[SID144108867]
Average IC50 0.81A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83 (8) [AID651917, Type: confirmatory]
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8
[SID131341903]
Average IC50 0.96A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83 (3) [AID602455, Type: confirmatory]
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9
[SID131341903]
IC50 0.97A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83 (2) [AID602241, Type: confirmatory]
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10
[SID131341903]
IC50 0.97A Cell-Based Counter Screen testing Compounds that Inhibit VEEV TC-83, in strain KU V3526 [AID602242, Type: confirmatory]
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11
[SID131341903]
Average IC50 1.01A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83 (6) [AID624449, Type: confirmatory]
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12
[SID49668524]
IC50 1.91A Cell-Based Confirmatory Screen for Compounds that Inhibit VEEV, TC-83 [AID588727, Type: confirmatory]
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13
[SID49668524]
Potency 10qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Texas Red Labeled MLL-derived Mutant Peptide [AID1768, Type: confirmatory]histone-lysine N-methyltransferase 2A isoform 2 precursor [Homo sapiens] [gi:56550039]
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14
[SID49668524]
Potency 10qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Texas Red Labeled MLL-derived Mutant Peptide [AID1768, Type: confirmatory]menin isoform 1 [Homo sapiens] [gi:18860839]
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15
[SID131341903]
CC50 100Vero 76 Cytoxicity Assay for VEEV Compounds (4) [AID623936, Type: confirmatory]
View
16
[SID131341903]
Virus Titer Reduction Secondary Screen for Compounds that Inhibit VEEV (TC-83 strain) [AID602307, Type: other]
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17
[SID131341903]
Virus Titer Reduction Secondary Screen for Compounds that Inhibit VEEV (2) Trinidad donkey strain [AID602411, Type: other]
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18
[SID131341903]
Virus Titer Reduction Secondary Screen for Compounds that Inhibit VEEV (TC-83 strain) (4) [AID651578, Type: other]
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19
[SID144108867]
Virus Titer Reduction Secondary Screen for Compounds that Inhibit VEEV (strain Trinidad donkey) (03) [AID651883, Type: other]
View
20
[SID144108867]
Virus Titer Reduction Secondary Screen for Compounds that Inhibit VEEV (TC-83 strain) (5) [AID651886, Type: other]
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21
[SID49668524]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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22
[SID49668524]
Potency 8.9125qHTS for Agonist of gsp, the Etiologic Mutation Responsible for Fibrous Dysplasia/McCune-Albright Syndrome: qHTS [AID624287, Type: confirmatory]Guanine nucleotide-binding protein G(s) subunit alpha isoforms short [gi:52000961]
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23
[SID131341903]
IC50 100A Cell-Based Secondary Assay for Compounds that Inhibit VEEV, TC-83 and other Alphaviruses (Chikungunya virus) [AID623935, Type: confirmatory]
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24
[SID131341903]
IC50 A Counter Screen of Venezuelan Equine Encephalitis Virus (VEEV) Inhibitors in a Cell-Based Anti-Respiratory Syncytial Virus (RSV) Assay [AID602470, Type: confirmatory]
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25
[SID131341903]
CC50 HEp2 Cytoxicity Assay for VEEV Compounds (1) [AID602483, Type: confirmatory]
View
26
[SID131341903]
CC50 Vero 76 Cytoxicity Assay for VEEV Compounds (3) [AID602439, Type: confirmatory]
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27
[SID131341903]
CC50 Vero 76 Cytoxicity Assay for VEEV Compounds (2) [AID602240, Type: confirmatory]
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28
[SID131341903]
CC50 Vero 76 Cytoxicity Assay for VEEV Compounds (5) [AID624069, Type: confirmatory]
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29
[SID144108867]
CC50 Vero 76 Cytoxicity Assay for VEEV Compounds (8) [AID651735, Type: confirmatory]
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30
[SID144108867]
IC50 A Cell-Based Secondary Assay for Compounds that Inhibit VEEV, TC-83 and other Alphaviruses (Chikungunya virus) (2) [AID651738, Type: confirmatory]
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31
[SID143472910]
CC50 Vero 76 Cytoxicity Assay for VEEV Compounds (9) [AID651930, Type: confirmatory]
View
32
[SID131341903]
CC50 Vero 76 Cytoxicity Assay for VEEV Compounds (7) [AID624450, Type: confirmatory]
View
33
[SID49668524]
Potency qHTS of GLP-1 Receptor Inverse Agonists: Cytotox Screen [AID624418, Type: confirmatory]
View
34
[SID49668524]
Counterscreen of compound fluorescence effects on High-throughput multiplex microsphere screening for inhibitors of toxin protease [AID624483, Type: screening]
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35
[SID49668524]
HIV entry: Env-mediated Cell Fusion Measured in Cell-Based System Using Plate Reader - 7013-01_Inhibitor_SinglePoint_HTS_Activity [AID651610, Type: screening]
View
36
[SID49668524]
DENV2 CPE-Based HTS Measured in Cell-Based and Microorganism Combination System Using Plate Reader - 2149-01_Other_SinglePoint_HTS_Activity [AID651640, Type: screening]
View
37
[SID49668524]
HTS for the detection of C. neoformans cell lysis via adenylate kinase (AK) release Measured in Microorganism System Using Plate Reader - 2162-01_Inhibitor_SinglePoint_HTS_Activity [AID651654, Type: screening]
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38
[SID49668524]
Luminescence Cell-Based Primary HTS to identify inhibitors of the oncoprotein EWS/Fli transcriptional activity Measured in Cell-Based System Using Plate Reader - 7014-01_Inhibitor_SinglePoint_HTS_Activity [AID651661, Type: screening]
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39
[SID49668524]
Flow Cytometric HTS Screening for Inhibitors of Lytic Granule Exocytosis with MLPCN Compound Library [AID651702, Type: screening]
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40
[SID49668524]
Potency qHTS Assay for Inhibitors of Hepatitis C Virus (HCV) [AID651820, Type: confirmatory]
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41
[SID49668524]
Fluorescence-based biochemical primary high throughput screening assay to identify molecules that bind r(CAG) RNA repeats [AID651821, Type: screening]
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42
[SID49668524]
Potency qHTS for induction of synthetic lethality in tumor cells producing 2HG: qHTS for the HT-1080-IDH1KD cell line [AID686971, Type: confirmatory]
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43
[SID49668524]
7011-01_Antagonist_SinglePoint_HTS_Activity [AID720647, Type: screening]
View
44
[SID49668524]
HTS for Bacterial rRNA inhibitors Measured in Microorganism-Based System Using Plate Reader - 7056-01_Inhibitor_SinglePoint_HTS_Activity [AID720706, Type: screening]
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45
[SID49668524]
High Content Cell-Based Imaging Primary HTS to Identify Small Molecules Involved in X-Chromosome Reactivation and Reprogramming Measured in Cell-Based System Using Imaging - 7015-01_Activator_SinglePoint_HTS_Activity_Set2 [AID743238, Type: screening]
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46
[SID49668524]
Inhibition of Alexa 488-Fibronectin deposition #on AH1F cell monolayers Measured in Cell-Based System Using Plate Reader - 7059-01_Inhibitor_SinglePoint_HTS_Activity [AID743247, Type: screening]
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47
[SID49668524]
Luminescent GLuc Reporter Gene Assay Primary HTS to Identify Small Molecule Activator of Glucose Dependent Insulin Secretion Measured in Cell-Based System Using Plate Reader - 7055-01_Activator_SinglePoint_HTS_Activity [AID743287, Type: screening]
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48
[SID49668524]
HTS for Inhibition of CaV1.3 ICDI/IQ interaction using a live-cell FRET assay Measured in Cell-Based System Using Plate Reader - 7081-01_Inhibitor_SinglePoint_HTS_Activity [AID743397, Type: screening]
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49
[SID49668524]
Wnt/Beta-catenin HTS Measured in Cell-Based System Using Plate Reader - 2161-01_Activator_SinglePoint_HTS_Activity [AID743398, Type: screening]
View
50
[SID144108867]
CC50 Vero 76 Cytoxicity Assay for VEEV Compounds (9) [AID651930, Type: confirmatory]
View