CHEMBL473126
(CID
15665937
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(
2
)
Inactive(
3
)
Top Targets:
Firefly Luc l..(
5
)
BioAssay Types:
Literature(
5
)
BioActivity Types:
IC50(
5
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 5 Data Row: 5 Total Pages: 1
Sort:
[Click the result table header to sort]
#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
103591778
]
Active
IC50
0.32
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive inhibition assay [AID
366888
, Type: Literature]
Luciferin 4-monooxygenase [gi:
41688574
]
View
X
Row No.
1
Structure
Substance
SID
103591778
CID
15665937
Outcome
Active
IC50
0.32 [uM]
BioAssay
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive inhibition assay
AID
366888
BioAssay type
Literature
Target
Luciferin 4-monooxygenase [gi:
41688574
]
PubMed
19215089
Data Table
2
[SID
103591778
]
Active
IC50
0.5
Inhibition of luciferin binding site of Photinus pyralis luciferase by noncompetitive inhibition assay [AID
366887
, Type: Literature]
Luciferin 4-monooxygenase [gi:
126501
]
View
X
Row No.
2
Structure
Substance
SID
103591778
CID
15665937
Outcome
Active
IC50
0.5 [uM]
BioAssay
Inhibition of luciferin binding site of Photinus pyralis luciferase by noncompetitive inhibition assay
AID
366887
BioAssay type
Literature
Target
Luciferin 4-monooxygenase [gi:
126501
]
PubMed
19215089
Data Table
3
[SID
103591778
]
Inactive
IC50
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive KinaseGlo luminescent assay [AID
366886
, Type: Literature]
Luciferin 4-monooxygenase [gi:
41688574
]
View
X
Row No.
3
Structure
Substance
SID
103591778
CID
15665937
Outcome
Inactive
IC50
[uM]
BioAssay
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive KinaseGlo luminescent assay
AID
366886
BioAssay type
Literature
Target
Luciferin 4-monooxygenase [gi:
41688574
]
PubMed
19215089
Data Table
4
[SID
103591778
]
Inactive
IC50
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive KinaseGlo Plus luminescent assay [AID
366897
, Type: Literature]
Luciferin 4-monooxygenase [gi:
41688574
]
View
X
Row No.
4
Structure
Substance
SID
103591778
CID
15665937
Outcome
Inactive
IC50
[uM]
BioAssay
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive KinaseGlo Plus luminescent assay
AID
366897
BioAssay type
Literature
Target
Luciferin 4-monooxygenase [gi:
41688574
]
PubMed
19215089
Data Table
5
[SID
103591778
]
Inactive
IC50
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive KinaseGlo Plus Max luminescent assay [AID
366898
, Type: Literature]
Luciferin 4-monooxygenase [gi:
41688574
]
View
X
Row No.
5
Structure
Substance
SID
103591778
CID
15665937
Outcome
Inactive
IC50
[uM]
BioAssay
Inhibition of luciferin binding site of Photuris pennsylvanica luciferase by noncompetitive KinaseGlo Plus Max luminescent assay
AID
366898
BioAssay type
Literature
Target
Luciferin 4-monooxygenase [gi:
41688574
]
PubMed
19215089
Data Table