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Canertinib (CID 156414) - Compound BioActivity Data
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BioActivity Outcomes:
Active(350)
 
 
Inactive(210)
 
 
Inconclusive(40)
 
 
Unspecified(543)
 
 
Top Targets:
PKc(98)
 
 
 
 
PKc like(79)
 
 
 
 
STKc AGC(45)
 
 
 
 
PTKc EGFR(40)
 
 
PTKc Abl(39)
 
 
 
BioAssay Types:
Literature(929)
 
 
 
 
Confirmatory(181)
 
 
 
 
Summary(24)
 
 
 
 
Screening(2)
 
 
BioActivity Types:
Kd(877)
 
 
 
 
Potency(108)
 
 
 
 
IC50(32)
 
 
 
EC50(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1050    Data Row: 1143   Total Pages: 58   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103202250]
Kd 0.0001Binding constant for EGFR(T790M) kinase domain [AID625007, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
2
[SID103202250]
Kd 0.00013Binding constant for EGFR(G719C) kinase domain [AID624998, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
3
[SID103202250]
Kd 0.00013Binding constant for EGFR(G719C) kinase domain [AID435157, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
4
[SID103202250]
Kd 0.00017Binding constant for EGFR(L747-E749del, A750P) kinase domain [AID435652, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
5
[SID103202250]
Kd 0.00017Binding constant for EGFR(L747-E749del, A750P) kinase domain [AID625000, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
6
[SID103202250]
Kd 0.00019Binding constant for EGFR(G719S) kinase domain [AID624999, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
7
[SID103202250]
Kd 0.00019Binding constant for EGFR(S752-I759del) kinase domain [AID625006, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
8
[SID103202250]
Kd 0.00019Binding constant for EGFR(S752-I759del) kinase domain [AID435792, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
9
[SID103202250]
Kd 0.00019Binding constant for EGFR kinase domain [AID435156, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
10
[SID103202250]
Kd 0.00019Binding constant for EGFR kinase domain [AID624996, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
11
[SID103202250]
Kd 0.00019Binding constant for EGFR(G719S) kinase domain [AID435402, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
12
[SID103202250]
Kd 0.00022Binding constant for EGFR(L861Q) kinase domain [AID435907, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
13
[SID103202250]
Kd 0.00022Binding constant for EGFR(L861Q) kinase domain [AID625005, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
14
[SID103202250]
Kd 0.00024Binding constant for EGFR(L858R) kinase domain [AID625003, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
15
[SID103202250]
Kd 0.00024Binding constant for EGFR(L858R) kinase domain [AID435525, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
16
[SID103202250]
Kd 0.00026Binding constant for EGFR(E746-A750del) kinase domain [AID624997, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
17
[SID103202250]
Kd 0.00026Binding constant for EGFR(L747-T751del,Sins) kinase domain [AID435906, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
18
[SID103202250]
Kd 0.00026Binding constant for EGFR(L747-S752del, P753S) kinase domain [AID435653, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
19
[SID103202250]
Kd 0.00026Binding constant for EGFR(E746-A750del) kinase domain [AID435791, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View
20
[SID103202250]
Kd 0.00026Binding constant for EGFR(L747-S752del, P753S) kinase domain [AID625001, Type: Literature]Epidermal growth factor receptor [gi:2811086]
View