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Idazoxan (CID 154494) - Compound BioActivity Data
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Filters: All Data » Active      
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BioActivity Outcomes:
Active(27)
 
 
Top Targets:
7TM GPCR Srx(3)
 
 
7TM GPCR Srsx(2)
 
 
Geminin(2)
 
 
PLDc mTdp1 2(2)
 
 
Aldo ket red(1)
 
 
BioAssay Types:
Literature(13)
 
 
Confirmatory(9)
 
 
Screening(4)
 
 
BioActivity Types:
Potency(9)
 
 
Kd(8)
 
 
IC50(5)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 22    Data Row: 27   Total Pages: 2   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103674322]
Kd 0.01047Alpha-2 adrenergic receptor agonist activity in mouse vas deferens assay compared to clonidine [AID36495, Type: Literature]Alpha-2A adrenergic receptor [gi:231460]
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2
[SID103674322]
Kd 0.01047Alpha-2 adrenergic receptor agonist activity in mouse vas deferens assay compared to clonidine [AID36495, Type: Literature]Alpha-2B adrenergic receptor [gi:68067981]
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3
[SID103674322]
Kd 0.01047Alpha-2 adrenergic receptor agonist activity in mouse vas deferens assay compared to clonidine [AID36495, Type: Literature]Alpha-2C adrenergic receptor [gi:231463]
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4
[SID103674322]
Kd 0.01585Antagonistic activity against Alpha-2 adrenergic receptor in the prostatic portion of the rat vas deferens [AID35359, Type: Literature]
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5
[SID103674322]
Kd 0.50119Alpha-1 adrenergic receptor agonist activity in rat anococcygeus assay [AID36173, Type: Literature]Alpha-1A adrenergic receptor [gi:1168247]
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6
[SID103674322]
Kd 0.50119Alpha-1 adrenergic receptor agonist activity in rat anococcygeus assay [AID36173, Type: Literature]Alpha-1D adrenergic receptor [gi:1168244]
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7
[SID103674322]
Kd 0.50119Alpha-1 adrenergic receptor agonist activity in rat anococcygeus assay [AID36173, Type: Literature]Alpha-1B adrenergic receptor [gi:543734]
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8
[SID103674322]
Kd 1.58489Agonistic activity against aAlpha-1 adrenergic receptor in the epidermal portion of the rat vas deferens; Compound contracture of vas at conc. grater than 10E-6 [AID35718, Type: Literature]
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9
[SID50106461]
Potency 7.9433Validation screen for small molecules that induce DNA re-replication in MCF 10A normal breast cells [AID463097, Type: confirmatory]geminin [Homo sapiens] [gi:7705682]
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10
[SID50106461]
Potency 8.9125qHTS for differential inhibitors of proliferation of Plasmodium falciparum line 7G8 [AID1815, Type: confirmatory]
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11
[SID103674322]
IC50 10Antiplasmodial activity against Plasmodium falciparum HB3 after 72 hrs by SYBR green assay [AID524795, Type: Literature]
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12
[SID103674322]
IC50 10Antiplasmodial activity against Plasmodium falciparum 7G8 after 72 hrs by SYBR green assay [AID524791, Type: Literature]
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13
[SID103674322]
IC50 12.5892Antiplasmodial activity against Plasmodium falciparum GB4 after 72 hrs by SYBR green assay [AID524794, Type: Literature]
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14
[SID103674322]
IC50 12.5892Antiplasmodial activity against Plasmodium falciparum 3D7 after 72 hrs by SYBR green assay [AID524790, Type: Literature]
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15
[SID103674322]
IC50 12.5892Antiplasmodial activity against Plasmodium falciparum W2 after 72 hrs by SYBR green assay [AID524796, Type: Literature]
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16
[SID50106461]
Potency 12.5893qHTS for differential inhibitors of proliferation of Plasmodium falciparum line W2 [AID1883, Type: confirmatory]
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17
[SID56422421]
Potency 12.9953qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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18
[SID56422421]
Potency 18.3564A quantitative high throughput screen for small molecules that induce DNA re-replication in MCF 10a normal breast cells. [AID624296, Type: confirmatory]geminin [Homo sapiens] [gi:7705682]
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19
[SID50106461]
Potency 19.9526qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID540256, Type: confirmatory]
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20
[SID50106461]
Potency 19.9526Validation screen for inhibitors of Lassa infection [AID463096, Type: confirmatory]
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