ZINC01332473 (CID 1434957) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Inactive(10)
 
 
Top Targets:
7TM GPCR Srsx(2)
 
 
 
NR DBD CAR(2)
 
 
BioAssay Types:
Confirmatory(7)
 
 
 
Screening(5)
 
 
BioActivity Types:
IC50(4)
 
 
 
EC50(3)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 12    Data Row: 12   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID99303126]
IC50 3.05SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 [AID485285, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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2
[SID99303126]
IC50 3.05SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 [AID485285, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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3
[SID99303126]
IC50 3.05SAR analysis of antagonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 [AID485285, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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4
[SID99303126]
IC50 9.24SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 4 [AID485287, Type: confirmatory]G-protein coupled receptor 55 [Homo sapiens] [gi:33695107]
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5
[SID99303126]
IC50 16.8SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 [AID485278, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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6
[SID99303126]
IC50 16.8SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 [AID485278, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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7
[SID99303126]
IC50 16.8SAR analysis of antagonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 [AID485278, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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8
[SID99303126]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 [AID485277, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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9
[SID99303126]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 [AID485277, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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10
[SID99303126]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay - Set 3 [AID485277, Type: confirmatory]cannabinoid receptor 2 [Homo sapiens] [gi:4502929]
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11
[SID99303126]
IC50 32SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 6 [AID485283, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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12
[SID99303126]
IC50 32SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 6 [AID485283, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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13
[SID99303126]
IC50 32SAR analysis of Antagonists of the GPR35 Receptor using an Image-Based Assay - Set 6 [AID485283, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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14
[SID99303126]
EC50 32SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay - Set 4 [AID485286, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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15
[SID99303126]
EC50 32SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay - Set 4 [AID485286, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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16
[SID99303126]
EC50 32SAR analysis of Agonists of the GPR35 Receptor using an Image-Based Assay - Set 4 [AID485286, Type: confirmatory]G-protein coupled receptor 35 isoform a [Homo sapiens] [gi:33695097]
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17
[SID99303126]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 [AID485282, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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18
[SID99303126]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 [AID485282, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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19
[SID99303126]
EC50 32SAR analysis of agonists of the Cannabinoid Receptor 1 using an Image-Based Assay - Set 4 [AID485282, Type: confirmatory]Cannabinoid receptor 1 (brain) [Homo sapiens] [gi:71682703]
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20
[SID143472054]
 Luminescence-based cell-based primary high throughput screening assay to identify activators of the DAF-12 from the parasite S. stercoralis (ssDAF-12) [AID652126, Type: screening]Protein DAF-12, isoform a [Caenorhabditis elegans] [gi:71987181]
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21
[SID143472054]
 Luminescence-based cell-based primary high throughput screening assay to identify activators of the DAF-12 from the parasite H. contortus (hcDAF-12) [AID652067, Type: screening]Protein DAF-12, isoform a [Caenorhabditis elegans] [gi:71987181]
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22
[SID143472054]
 Primary biochemical fluorescence polarization-based high throughput screening assay to identify inhibitors of protein arginine methyltransferase 1 (PRMT1) [AID652257, Type: screening]PRMT1 protein [Homo sapiens] [gi:32425330]
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23
[SID143472054]
 Primary biochemical fluorescence polarization-based high throughput screening assay to identify inhibitors of protein arginine methyltransferase 1 (PRMT1) [AID652257, Type: screening]PRMT1 protein [Homo sapiens] [gi:32425330]
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24
[SID143472054]
 Luminescence-based cell-based primary high throughput screening assay to identify inhibitors of COUP-TFII (NR2F2) [AID686940, Type: screening]NR2F2 gene product [Homo sapiens] [gi:14149746]
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25
[SID143472054]
 Luminescence-based cell-based primary high throughput screening assay to identify inhibitors of COUP-TFII (NR2F2) [AID686940, Type: screening]NR2F2 gene product [Homo sapiens] [gi:14149746]
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26
[SID143472054]
 TRFRET-based biochemical primary high throughput screening assay to identify inhibitors of 5-meCpG-binding domain protein 2 (MBD2)-DBD binding to methylated oligonucleotide [AID686964, Type: screening]Methyl-CpG binding domain protein 2 [Homo sapiens] [gi:21595776]
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