CHEMBL57502 (CID 13891346) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(1)
 
 
Inactive(5)
 
 
Unspecified(12)
 
 
Top Targets:
PAD(4)
 
 
 
PAD M(2)
 
 
BioAssay Types:
Literature(12)
 
 
SAR
Target summary
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 14    Data Row: 18   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID118043682]
 Late stage assay provider results from the probe development effort to identify inhibitors of Arginine Deiminase 4 (PAD4): colorimetric biochemical substrate assay to identify inhibitors of PAD4 [AID588559, Type: other]PADI4 gene product [Homo sapiens] [gi:216548487]
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2
[SID118043682]
 Late stage assay provider results from the probe development effort to identify inhibitors of Arginine Deiminase 4 (PAD4): colorimetric biochemical substrate assay to identify inhibitors of PAD4 [AID588559, Type: other]PADI4 gene product [Homo sapiens] [gi:216548487]
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3
[SID103245942]
 Cytotoxic activity against mouse melanoma cell culture(B-16) [AID38038, Type: Literature]
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4
[SID103245942]
 Cytotoxic activity against human lymphoblastic leukemia cell culture (CCRF-CEM) [AID44017, Type: Literature]
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5
[SID103245942]
 Antimicrobial activity was determined against Candida albicans ATCC 10231 [AID44989, Type: Literature]
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6
[SID103245942]
 Antimicrobial activity was determined against Escherichia coli ATCC 9637 [AID69959, Type: Literature]
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7
[SID103245942]
 Cytotoxic activity against human epidermoid carcinoma of the nasopharynx (9KB) [AID70059, Type: Literature]
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8
[SID103245942]
 Antimicrobial activity was determined against Klebsiella pneumoniae ATCC 10031 [AID94298, Type: Literature]
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9
[SID103245942]
 Cytotoxic activity against mouse lymphoblastic leukemia cell culture (L-1210) [AID94732, Type: Literature]
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10
[SID103245942]
 Antimicrobial activity was determined against Mycobacterium smegmatis ATCC 607 [AID144440, Type: Literature]
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11
[SID103245942]
 Cytotoxic activity against P388 mouse leukemia cell culture (9PS(P388)) [AID152574, Type: Literature]
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12
[SID103245942]
 Antimicrobial activity was determined against Pseudomonas aeruginosa ATCC 27853 cells [AID164400, Type: Literature]
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13
[SID103245942]
 Antimicrobial activity was determined against Salmonella gallinarum ATCC 9184 [AID200512, Type: Literature]
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14
[SID103245942]
 Antimicrobial activity was determined against Staphylococcus aureus ATCC 13709 [AID207620, Type: Literature]
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15
[SID118043682]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAD4: colorimetric biochemical substrate assay to identify inhibitors of PADs 1-4 [AID588560, Type: other]PADI1 gene product [Homo sapiens] [gi:122056685]
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16
[SID118043682]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAD4: colorimetric biochemical substrate assay to identify inhibitors of PADs 1-4 [AID588560_1, Type: other]PADI1 gene product [Homo sapiens] [gi:122056685]
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17
[SID118043682]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAD4: colorimetric biochemical substrate assay to identify inhibitors of PADs 1-4 [AID588560_2, Type: other]PADI2 gene product [Homo sapiens] [gi:122939159]
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18
[SID118043682]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAD4: colorimetric biochemical substrate assay to identify inhibitors of PADs 1-4 [AID588560_3, Type: other]PADI3 gene product [Homo sapiens] [gi:122939161]
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19
[SID118043682]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAD4: colorimetric biochemical substrate assay to identify inhibitors of PADs 1-4 [AID588560_4, Type: other]PADI4 gene product [Homo sapiens] [gi:216548487]
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