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ethyl 4-{[(5-phenyl-2H-tetrazol-2-yl)acetyl]amino}benzoate (CID 1267856) - Compound BioActivity Data
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BioActivity Outcomes:
Active(14)
 
 
Inactive(824)
 
 
Inconclusive(23)
 
 
Unspecified(3)
 
 
Top Targets:
7TM GPCR Srx(28)
 
 
 
7TM GPCR Srsx(25)
 
 
 
alkPPc(14)
 
 
Bcl-2 like(12)
 
 
Tryp SPc(11)
 
 
BioAssay Types:
Screening(574)
 
 
 
 
 
Confirmatory(257)
 
 
 
 
 
Literature(11)
 
 
 
BioActivity Types:
Potency(167)
 
 
 
 
 
IC50(52)
 
 
 
EC50(16)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 792    Data Row: 864   Total Pages: 44   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID126920242]
EC50_MICROM 0.123Counter screen for HTS for Beta-2AR agonists with FAP-tagged human CCR5 with Powderset2 [AID651728, Type: confirmatory]CCR5, partial [Homo sapiens] [gi:289466095]
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2
[SID126920242]
EC50_MICROM 0.134Counter screen for HTS for Beta-2AR agonists with FAP-tagged GPR32 with Powderset2 [AID651729, Type: confirmatory]G protein-coupled receptor 32 [Homo sapiens] [gi:119592304]
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3
[SID4244167]
EC50_MICROM 1.18Dose response for HTS for Beta-2AR agonists via FAP method from CP1 [AID588763, Type: confirmatory]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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4
[SID126920242]
EC50_MICROM 1.31Dose response for HTS for Beta-2AR agonists via FAP method from Powderset2 [AID623882, Type: confirmatory]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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5
[SID4244167]
Potency 25.1189qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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6
[SID4244167]
Luminescence-based cell-based primary high throughput screening assay to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A) [AID624169, Type: screening]5-hydroxytryptamine receptor 2A [Mus musculus] [gi:27753985]
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7
[SID4244167]
HTS for Beta-2AR agonists via FAP method [AID504454, Type: screening]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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8
[SID4244167]
HTS for Beta-2AR agonists via FAP method, Single Point, Cherry Pick 1 [AID540358, Type: other]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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9
[SID4244167]
Anti-Viral Drugs Against Arbovirus Infections, a Primary Screen [AID1251, Type: screening]
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10
[SID4244167]
KCNQ2 Counter screen for inhibitors that protect hERG from block by proarrhythmic agents [AID1946, Type: screening]potassium voltage-gated channel subfamily KQT member 2 [Rattus norvegicus] [gi:18959272]
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11
[SID4244167]
Multiplex HTS Assay for Inhibitors of MEK Kinase PB1 Domains, specifically MEK5 binding to MEK Kinase 2 Wildtype [AID1531, Type: screening]mitogen-activated protein kinase kinase kinase kinase 2 [Homo sapiens] [gi:22035600]
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12
[SID4244167]
Primary cell-based high-throughput screening assay for identification of compounds that protect hERG from block by proarrhythmic agents [AID1511, Type: screening]putative potassium channel subunit [Homo sapiens] [gi:487738]
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13
[SID4244167]
Primary HTS assay during TNFalpha stimulated VCAM1 expression to assess cytotoxicity. [AID848, Type: other]vascular cell adhesion protein 1 isoform a precursor [Homo sapiens] [gi:4507875]
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14
[SID4244167]
Primary HTS assay for chemical inhibitors of TNF alpha stimulated VCAM1 expression [AID802, Type: screening]
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15
[SID4244167]
Potency 39.8107qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor [AID926, Type: confirmatory]thyroid stimulating hormone receptor [Homo sapiens] [gi:38016895]
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16
[SID4244167]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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17
[SID4244167]
Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
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18
[SID4244167]
Potency 3.5481qHTS of GLP-1 Receptor Inverse Agonists: Cytotox Screen [AID624418, Type: confirmatory]
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19
[SID4244167]
Potency 8.9125qHTS for Inhibitors of TGF-b: Cytotox Counterscreen [AID588856, Type: confirmatory]
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20
[SID4244167]
uHTS determination of small molecule cytotoxicity in a fluorescence assay to identify cystic fibrosis induced NFkb Inhibitors [AID602141, Type: screening]
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