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BioActivity Data for Compound gamma-Aminobutyric Acid (CID 119)

BioActivity Outcomes:
Active(254)
 
 
Inactive(1310)
 
 
Inconclusive(79)
 
 
Unspecified(225)
 
 
Top Targets:
Neur chan LBD(168)
 
 
 
 
Neur chan mem..(58)
 
 
 
 
7tm 4(55)
 
 
 
PBP1 GABAb re..(17)
 
 
 
SLC5-6-like s..(15)
 
 
 
 
BioAssay Types:
Confirmatory(633)
 
 
 
 
 
Literature(572)
 
 
 
 
 
Screening(547)
 
 
 
 
Summary(16)
 
 
BioAssay Categories:
In vitro(19)
 
 
 
 
In vivo(14)
 
 
 
 
Biochemical(193)
 
 
 
 
 
Toxicity(30)
 
 
 
 
 
ADME(27)
 
 
Cell-based(197)
 
 
 
 
 
Organism-base..(16)
 
 
 
BioActivity Types:
Potency(536)
 
 
 
 
 
IC50(215)
 
 
 
 
 
EC50(72)
 
 
 
 
Ki(21)
 
 
 
AC50(3)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1244    Data Row: 1868   Total Pages: 94   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-2 [gi:120758]
View
2
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:120761]
View
3
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-4 [gi:120763]
View
4
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-5 [gi:120764]
View
5
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-1 [gi:120769]
View
6
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-1 [gi:120782]
View
7
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:120788]
View
8
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-3 [gi:120790]
View
9
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-6 [gi:232127]
View
10
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit delta [gi:544363]
View
11
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit pi [gi:3023821]
View
12
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit epsilon [gi:13959374]
View
13
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-1 [gi:51317298]
View
14
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-2 [gi:52000957]
View
15
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:52000955]
View
16
[SID103173784]
IC50 0.013Inhibition of [3H]GABA binding in GABAA receptor in rat brain synaptic membranes [AID267285, Type: Literature]GABA theta subunit [gi:81902501]
View
17
[SID103173784]
IC50 0.015Displacement of [3H]muscimol from GABAA receptor in Sprague-Dawley rat spinal cord brainstem membranes [AID286350, Type: Literature]
View
18
[SID103173784]
IC50 0.015Displacement of [3H]muscimol from GABA-A receptor in Sprague-Dawley rat spinal cord [AID270052, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-3 [gi:120790]
View
19
[SID103173784]
IC50 0.015Displacement of [3H]muscimol from GABA-A receptor in Sprague-Dawley rat spinal cord [AID270052, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:120788]
View
20
[SID103173784]
IC50 0.015Displacement of [3H]muscimol from GABA-A receptor in Sprague-Dawley rat spinal cord [AID270052, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-1 [gi:120782]
View