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CHEMBL1934476 (CID 11619439) - Compound BioActivity Data
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BioActivity Outcomes:
Active(12)
 
 
Unspecified(35)
 
 
Top Targets:
NR LBD PPAR(11)
 
 
BioAssay Types:
Literature(47)
 
 
 
BioActivity Types:
EC50(15)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 47    Data Row: 47   Total Pages: 3   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136944681]
EC50 0.008Transactivation of human PPARalpha expressed in CHO-K1 cells [AID638935, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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2
[SID136944681]
EC50 0.19Agonist activity at dog PPARalpha [AID638996, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:24418624]
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3
[SID136944681]
EC50 0.61Agonist activity at hamster PPARalpha [AID638999, Type: Literature]
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4
[SID136944681]
EC50 2.7Agonist activity at dog PPARdelta [AID638998, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:115502562]
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5
[SID136944681]
EC50 3Transactivation of human PPARdelta expressed in CHO-K1 cells [AID638937, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
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6
[SID136944681]
EC50 3.6Agonist activity at rat PPARalpha [AID639002, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:585718]
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7
[SID136944681]
EC50 4.7Agonist activity at mouse PPARalpha [AID639005, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:1709728]
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8
[SID136944681]
EC50 6.6Agonist activity at mouse PPARdelta [AID639007, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:548577]
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9
[SID136944681]
EC50 9.6Transactivation of human PPARgamma expressed in CHO-K1 cells [AID638936, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
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10
[SID136944681]
EC50 11Agonist activity at dog PPARgamma [AID638997, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:75068622]
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11
[SID136944681]
EC50 12Agonist activity at mouse PPARgamma [AID639006, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432235]
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12
[SID136944681]
EC50 13Agonist activity at rat PPARgamma [AID639003, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13431783]
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13
[SID136944681]
EC50 7.1Agonist activity at hamster PPARdelta [AID639001, Type: Literature]
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14
[SID136944681]
EC50 14Agonist activity at rat PPARdelta [AID639004, Type: Literature]
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15
[SID136944681]
EC50 15Agonist activity at hamster PPARgamma [AID639000, Type: Literature]
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16
[SID136944681]
Selectivity ratio of EC50 for dog PPARalpha to EC50 for human PPARalpha [AID639008, Type: Literature]
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17
[SID136944681]
Selectivity ratio of EC50 for hamster PPARalpha to EC50 for human PPARalpha [AID639009, Type: Literature]
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18
[SID136944681]
Selectivity ratio of EC50 for rat PPARalpha to EC50 for human PPARalpha [AID639010, Type: Literature]
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19
[SID136944681]
Selectivity ratio of EC50 for mouse PPARalpha to EC50 for human PPARalpha [AID639011, Type: Literature]
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20
[SID136944681]
Total clearance in rat at 1 mg/kg, po [AID639012, Type: Literature]
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