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KW 2449 (CID 11427553) - Compound BioActivity Data
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BioActivity Outcomes:
Active(320)
 
 
Unspecified(124)
 
 
Top Targets:
PTKc Abl(16)
 
 
PTKc EGFR(12)
 
 
 
PI3Kc IA alph..(10)
 
 
PKc like(9)
 
 
 
ig(8)
 
 
BioAssay Types:
Literature(444)
 
 
 
BioActivity Types:
Kd(444)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 444    Data Row: 444   Total Pages: 23   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136944791]
Kd 0.0029Binding constant for DRAK1 kinase domain [AID624968, Type: Literature]Serine/threonine-protein kinase 17A [gi:317373279]
View
2
[SID136944791]
Kd 0.0043Binding constant for MLCK kinase domain [AID624738, Type: Literature]Myosin light chain kinase 3 [gi:254763411]
View
3
[SID136944791]
Kd 0.0048Binding constant for DRAK2 kinase domain [AID624942, Type: Literature]Serine/threonine-protein kinase 17B [gi:14423909]
View
4
[SID136944791]
Kd 0.0052Binding constant for YSK4 kinase domain [AID625136, Type: Literature]Mitogen-activated protein kinase kinase kinase 19 [gi:74755104]
View
5
[SID136944791]
Kd 0.0059Binding constant for ABL1(T315I)-phosphorylated kinase domain [AID624989, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
6
[SID136944791]
Kd 0.0066Binding constant for FLT3(K663Q) kinase domain [AID624938, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
7
[SID136944791]
Kd 0.0096Binding constant for BIKE kinase domain [AID625109, Type: Literature]BMP-2-inducible protein kinase [gi:34222653]
View
8
[SID136944791]
Kd 0.011Binding constant for MAP4K2 kinase domain [AID624959, Type: Literature]Mitogen-activated protein kinase kinase kinase kinase 2 [gi:215274019]
View
9
[SID136944791]
Kd 0.012Binding constant for ABL1(T315I)-non phosphorylated kinase domain [AID624988, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
10
[SID136944791]
Kd 0.012Binding constant for KIT(V559D,T670I) kinase domain [AID624792, Type: Literature]Mast/stem cell growth factor receptor Kit [gi:125472]
View
11
[SID136944791]
Kd 0.013Binding constant for LOK kinase domain [AID625030, Type: Literature]Serine/threonine-protein kinase 10 [gi:12643358]
View
12
[SID136944791]
Kd 0.013Binding constant for SLK kinase domain [AID625086, Type: Literature]STE20-like serine/threonine-protein kinase [gi:74762732]
View
13
[SID136944791]
Kd 0.013Binding constant for FLT3(N841I) kinase domain [AID624939, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
14
[SID136944791]
Kd 0.013Binding constant for FLT3(D835H) kinase domain [AID624935, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
15
[SID136944791]
Kd 0.013Binding constant for FLT3(D835Y) kinase domain [AID624936, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
16
[SID136944791]
Kd 0.015Binding affinity to human FLT3 [AID775336, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
17
[SID136944791]
Kd 0.015Binding constant for FLT3 kinase domain [AID624934, Type: Literature]Receptor-type tyrosine-protein kinase FLT3 [gi:156630887]
View
18
[SID136944791]
Kd 0.015Binding constant for SRPK2 kinase domain [AID624768, Type: Literature]SRSF protein kinase 2 [gi:300669676]
View
19
[SID136944791]
Kd 0.017Binding constant for ABL1(H396P)-non phosphorylated kinase domain [AID624983, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
20
[SID136944791]
Kd 0.018Binding constant for YES kinase domain [AID625018, Type: Literature]Tyrosine-protein kinase Yes [gi:125870]
View