SureCN3936450 (CID 11380248) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(4)
 
 
Unspecified(2)
 
 
Top Targets:
NR LBD ER(3)
 
 
 
NR LBD ERR(2)
 
 
BioAssay Types:
Literature(6)
 
 
 
BioActivity Types:
IC50(4)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 6    Data Row: 6   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103471383]
IC50 0.0046Binding affinity for human Estrogen receptor beta [AID254777, Type: Literature]Estrogen receptor beta [gi:6166154]
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2
[SID103471383]
IC50 0.0046Binding affinity for human Estrogen receptor beta [AID254777, Type: Literature]Estrogen receptor beta [gi:6166154]
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3
[SID103471383]
IC50 0.0046Binding affinity for human Estrogen receptor beta [AID254777, Type: Literature]Estrogen receptor beta [gi:6166154]
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4
[SID103471383]
IC50 0.0046Inhibition of human ERalpha [AID307629, Type: Literature]Steroid hormone receptor ERR1 [gi:215274146]
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5
[SID103471383]
IC50 0.0046Inhibition of human ERalpha [AID307629, Type: Literature]Steroid hormone receptor ERR1 [gi:215274146]
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6
[SID103471383]
IC50 0.213Inhibition of human ERbeta [AID307630, Type: Literature]Steroid hormone receptor ERR2 [gi:374095385]
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7
[SID103471383]
IC50 0.213Inhibition of human ERbeta [AID307630, Type: Literature]Steroid hormone receptor ERR2 [gi:374095385]
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8
[SID103471383]
IC50 0.213Binding affinity for human Estrogen receptor alpha [AID254783, Type: Literature]Estrogen receptor [gi:544257]
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9
[SID103471383]
IC50 0.213Binding affinity for human Estrogen receptor alpha [AID254783, Type: Literature]Estrogen receptor [gi:544257]
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10
[SID103471383]
IC50 0.213Binding affinity for human Estrogen receptor alpha [AID254783, Type: Literature]Estrogen receptor [gi:544257]
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11
[SID103471383]
IC50 0.213Binding affinity for human Estrogen receptor alpha [AID254783, Type: Literature]Estrogen receptor [gi:544257]
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12
[SID103471383]
 Selectivity for human ERalpha over ERbeta [AID307631, Type: Literature]
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13
[SID103471383]
 Selectivity as ratio of IC50 against estrogen receptor alpha and beta [AID255369, Type: Literature]Estrogen receptor [gi:544257]
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14
[SID103471383]
 Selectivity as ratio of IC50 against estrogen receptor alpha and beta [AID255369, Type: Literature]Estrogen receptor [gi:544257]
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15
[SID103471383]
 Selectivity as ratio of IC50 against estrogen receptor alpha and beta [AID255369, Type: Literature]Estrogen receptor [gi:544257]
View
16
[SID103471383]
 Selectivity as ratio of IC50 against estrogen receptor alpha and beta [AID255369, Type: Literature]Estrogen receptor [gi:544257]
View