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BioActivity Data for Compound 174899-83-3 (CID 11258643)

BioActivity Outcomes:
Active(1)
 
 
Inactive(72)
 
 
Inconclusive(13)
 
 
Unspecified(62)
 
 
Top Targets:
NR LBD PPAR(8)
 
 
 
NR LBD AR(7)
 
 
 
NR LBD ER(7)
 
 
NR LBD Fxr(4)
 
 
 
NR LBD GR(4)
 
 
BioAssay Types:
Confirmatory(64)
 
 
 
 
 
Literature(60)
 
 
Summary(24)
 
 
 
BioAssay Categories:
Biochemical(2)
 
 
Toxicity(6)
 
 
 
 
Cell-based(60)
 
 
BioActivity Types:
Potency(80)
 
 
 
 
IC50(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 148    Data Row: 148   Total Pages: 8   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144209815]
Potency-Replicate_1 61.1306qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rev3 mutant cell line [AID743014, Type: confirmatory]
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2
[SID103718473]
IC50 333Inhibition of HIV1 recombinant integrase 3' processing activity using [32P]-radiolabeled full-length DNA as substrate after 1 hr by densitometric analysis [AID1117864, Type: confirmatory] [gi:82312013]
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3
[SID103718473]
IC50 333Inhibition of HIV1 recombinant integrase strand transfer activity using [32P]-radiolabeled full-length DNA as substrate after 1 hr by densitometric analysis [AID1117866, Type: confirmatory] [gi:82312013]
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4
[SID103718473]
Anticancer activity against human SF539 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455634, Type: Literature]
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5
[SID103718473]
Anticancer activity against human SNB19 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455635, Type: Literature]
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6
[SID103718473]
Anticancer activity against human SNB75 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455636, Type: Literature]
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7
[SID103718473]
Anticancer activity against human U251 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455637, Type: Literature]
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8
[SID103718473]
Anticancer activity against human LOXIMVI cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455638, Type: Literature]
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9
[SID103718473]
Anticancer activity against human MALME-3M cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455639, Type: Literature]
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10
[SID103718473]
Anticancer activity against human M14 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455640, Type: Literature]
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11
[SID103718473]
Anticancer activity against human SK-MEL-2 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455641, Type: Literature]
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12
[SID103718473]
Anticancer activity against human SK-MEL-28 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455642, Type: Literature]
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13
[SID103718473]
Anticancer activity against human SK-MEL-5 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455643, Type: Literature]
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14
[SID103718473]
Anticancer activity against human UACC257 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455644, Type: Literature]
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15
[SID103718473]
Anticancer activity against human UACC62 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455645, Type: Literature]
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16
[SID103718473]
Anticancer activity against human IGROV1 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455646, Type: Literature]
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17
[SID103718473]
Anticancer activity against human OVCAR-3 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455647, Type: Literature]
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18
[SID103718473]
Anticancer activity against human OVCAR4 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455648, Type: Literature]
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19
[SID103718473]
Anticancer activity against human OVCAR5 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455649, Type: Literature]
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20
[SID103718473]
Anticancer activity against human OVCAR8 cells assessed cell growth at 10 uM after 48 hrs by sulforhodamine B assay relative to control [AID455650, Type: Literature]
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