aminobenzolamide 18 (CID 11069133) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(29)
 
 
Unspecified(1)
 
 
Top Targets:
alpha CA I II..(11)
 
 
 
alpha CA(2)
 
 
alpha CA IV X..(2)
 
 
alpha CA XII..(2)
 
 
alpha CA V(1)
 
 
BioAssay Types:
Literature(30)
 
 
 
BioActivity Types:
Ki(29)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 30    Data Row: 30   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103265744]
Ki 0.0003Inhibition constant (Ki) against human cloned carbonic anhydrase II (CAH) [AID47931, Type: Literature]
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2
[SID103265744]
Ki 0.0003Inhibition of human carbonic anhydrase II by spectrophotometry at pH 7.5 [AID577527, Type: Literature]Carbonic anhydrase 2 [gi:115456]
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3
[SID103265744]
Ki 0.0003Inhibition of human recombinant carbonic anhydrase 2 after 15 mins by stopped-flow CO2 hydration assay [AID493884, Type: Literature]Carbonic anhydrase 2 [gi:115456]
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4
[SID103265744]
Ki 0.0003Inhibition of human recombinant carbonic anhydrase 2 after 15 mins by stopped flow CO2 hydration assay [AID644381, Type: Literature]Carbonic anhydrase 2 [gi:115456]
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5
[SID103265744]
Ki 0.0007Inhibition of human recombinant carbonic anhydrase 13 after 15 mins by stopped-flow CO2 hydration assay [AID493893, Type: Literature]Carbonic anhydrase 13 [gi:30580350]
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6
[SID103265744]
Ki 0.0009Inhibition of human recombinant carbonic anhydrase 14 after 15 mins by stopped-flow CO2 hydration assay [AID493894, Type: Literature]Carbonic anhydrase 14 [gi:8928036]
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7
[SID103265744]
Ki 0.0014Inhibition of human recombinant carbonic anhydrase 1 after 15 mins by stopped-flow CO2 hydration assay [AID493883, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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8
[SID103265744]
Ki 0.0014Inhibition of human recombinant carbonic anhydrase 1 after 15 mins by stopped flow CO2 hydration assay [AID644380, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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9
[SID103265744]
Ki 0.0014Inhibition of human carbonic anhydrase I by spectrophotometry at pH 7.5 [AID577526, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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10
[SID103265744]
Ki 0.0014Inhibition constant determined against human cloned carbonic anhydrase I [AID50366, Type: Literature]
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11
[SID103265744]
Ki 0.002Inhibition constant against bovine Carbonic anhydrase IV, isolated from lung microsomes [AID48132, Type: Literature]
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12
[SID103265744]
Ki 0.0028Inhibition of GST-tagged astrosclera willeyana Astrosclerin-3 expressed in Escherichia coli after 15 mins preincubation by stopped flow CO2 hydration assay [AID644379, Type: Literature]
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13
[SID103265744]
Ki 0.0029Inhibition of human recombinant carbonic anhydrase 7 after 15 mins by stopped-flow CO2 hydration assay [AID493890, Type: Literature]Carbonic anhydrase 7 [gi:1168744]
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14
[SID103265744]
Ki 0.013Inhibition of human recombinant carbonic anhydrase 12 after 15 mins by stopped-flow CO2 hydration assay [AID493892, Type: Literature]Carbonic anhydrase 12 [gi:5915866]
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15
[SID103265744]
Ki 0.015Inhibition of human recombinant carbonic anhydrase 4 after 15 mins by stopped-flow CO2 hydration assay [AID493886, Type: Literature]Carbonic anhydrase 4 [gi:115465]
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16
[SID103265744]
Ki 0.018Inhibition of human recombinant carbonic anhydrase 5b after 15 mins by stopped-flow CO2 hydration assay [AID493888, Type: Literature]Carbonic anhydrase 5B, mitochondrial [gi:8928041]
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17
[SID103265744]
Ki 0.021Inhibition of human recombinant carbonic anhydrase 5a after 15 mins by stopped-flow CO2 hydration assay [AID493887, Type: Literature]Carbonic anhydrase 5A, mitochondrial [gi:461680]
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18
[SID103265744]
Ki 0.03Inhibition of mouse recombinant carbonic anhydrase 15 after 15 mins by stopped-flow CO2 hydration assay [AID493895, Type: Literature]Carbonic anhydrase 15 [gi:30580362]
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19
[SID103265744]
Ki 0.038Inhibition of human recombinant carbonic anhydrase 9 after 15 mins by stopped-flow CO2 hydration assay [AID493891, Type: Literature]Carbonic anhydrase 9 [gi:83300925]
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20
[SID103265744]
Ki 0.038Inhibition of Salmonella Typhimurium recombinant carbonic anhydrase 2 at pH 8.3 by stopped flow CO2 hydration assay [AID612732, Type: Literature]
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21
[SID103265744]
Ki 0.04Inhibition constant determined against catalytic domain of human cloned carbonic anhydrase IX [AID48299, Type: Literature]
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22
[SID103265744]
Ki 0.041Inhibition of human recombinant carbonic anhydrase 6 after 15 mins by stopped-flow CO2 hydration assay [AID493889, Type: Literature]Carbonic anhydrase 6 [gi:116241278]
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23
[SID103265744]
Ki 0.051Inhibition of Salmonella Typhimurium recombinant carbonic anhydrase 1 at pH 8.3 by stopped flow CO2 hydration assay [AID612731, Type: Literature]
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24
[SID103265744]
Ki 0.186Inhibition of Brucella suis carbonic anhydrase I by spectrophotometry at pH 8.3 [AID577531, Type: Literature]
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25
[SID103265744]
Ki 0.3Inhibition of human recombinant carbonic anhydrase 2 at pH 7.5 by stopped flow CO2 hydration assay [AID612726, Type: Literature]Carbonic anhydrase 2 [gi:115456]
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26
[SID103265744]
Ki 0.663Inhibition of Brucella suis carbonic anhydrase II by spectrophotometry at pH 8.3 [AID577530, Type: Literature]
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27
[SID103265744]
Ki 1.4Inhibition of human recombinant carbonic anhydrase 1 at pH 7.5 by stopped flow CO2 hydration assay [AID612725, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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28
[SID103265744]
Ki 18Inhibition of human recombinant carbonic anhydrase 3 after 15 mins by stopped-flow CO2 hydration assay [AID493885, Type: Literature]Carbonic anhydrase 3 [gi:134047703]
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29
[SID103265744]
 Inhibition of Brucella suis CA1 expressed in Escherichia coli BL21(DE3) by stopped-flow CO2-hydration assay [AID459696, Type: Literature]
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30
[SID103265744]
Ki 80.5Inhibition of human recombinant CA 3 assessed as CO2 hydration by stopped flow kinetic assay [AID301578, Type: Literature]Carbonic anhydrase 3 [gi:134047703]
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