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epicatechin gallate (CID 107905) - Compound BioActivity Data
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BioActivity Outcomes:
Active(52)
 
 
Inactive(30)
 
 
Inconclusive(2)
 
 
Unspecified(72)
 
 
Top Targets:
HIF-1a CTAD(7)
 
 
 
7TM GPCR Srx(6)
 
 
 
PAS(4)
 
 
 
ALBUMIN(3)
 
 
 
ABCC MRP doma..(3)
 
 
BioAssay Types:
Literature(132)
 
 
 
 
 
Screening(3)
 
 
Confirmatory(3)
 
 
 
BioActivity Types:
IC50(31)
 
 
 
Ki(6)
 
 
Kd(1)
 
 
EC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 156    Data Row: 156   Total Pages: 8   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103215553]
Ki 0.016Inhibition of Plasmodium falciparum ENR in presence of triclosan [AID277587, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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2
[SID103215553]
IC50 0.036Binding affinity to opiate receptor [AID311289, Type: Literature]
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3
[SID103215553]
Ki 0.102Inhibition of Plasmodium falciparum ENR using crotonyl-CoA substrate [AID277586, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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4
[SID103215553]
IC50 0.18Inhibition of yeast G6PD [AID319369, Type: Literature]Glucose-6-phosphate 1-dehydrogenase [gi:120734]
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5
[SID103215553]
IC50 0.2Inhibition of FabI [AID265759, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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6
[SID103215553]
IC50 0.21Inhibition of 6PGD [AID319370, Type: Literature]
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7
[SID103215553]
Ki 0.291Inhibition of Plasmodium falciparum ENR using NADH substrate [AID277585, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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8
[SID103215553]
Ki 0.4Displacement of NLWAAQRYGRELRRMSD-K(FITC)-FVD from Bcl-2 (unknown origin) by fluorescence polarization assay [AID1095217, Type: confirmatory]Apoptosis regulator Bcl-2 [gi:231632]
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9
[SID103215553]
IC50 0.4Inhibition of FabZ [AID265758, Type: Literature]Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein) [gi:74844869]
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10
[SID103215553]
IC50 0.5Inhibition of Plasmodium falciparum ENR [AID277583, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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11
[SID103215553]
IC50 0.76Inhibition of polymerization in wild type HIV-1 RT with poly rC/dG12-18 template primer and [3H]dGTP [AID83435, Type: Literature]Reverse transcriptase/RNaseH [gi:82310930]
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12
[SID103215553]
IC50 1Inhibition of FabG [AID265760, Type: Literature]3-oxoacyl-acyl-carrier protein reductase precursor [gi:75020671]
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13
[SID103215553]
IC50 1.47Inhibition of p38alpha after 1 hr by ELISA [AID566611, Type: Literature]
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14
[SID103215553]
IC50 1.5Antioxidant activity assessed as DPPH radical scavenging activity after 30 mins by spectrophotometry [AID650645, Type: Literature]
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15
[SID103215553]
Ki 2.07Ki values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cells [AID977601, Type: Literature]
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16
[SID103215553]
Ki 3.46Ki values for sodium fluorescein (10 uM) uptake in OATP1B3-transfected CHO cells [AID977604, Type: Literature]
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17
[SID103215553]
IC50 3.80189pIC50 values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cells [AID977600, Type: Literature]
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18
[SID103215553]
IC50 4.46684pIC50 values for sodium fluorescein (10 uM) uptake in OATP1B3-transfected CHO cells [AID977603, Type: Literature]
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19
[SID103215553]
IC50 5.4Inhibition of lipid peroxidation in Sprague-Dawley rat heart mitochondria assessed as inhibition of FeSO4-induced malondialdehyde formation [AID398697, Type: Literature]
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20
[SID103215553]
IC50 8.4Inhibition of lipid peroxidation in Sprague-Dawley rat heart mitochondria assessed as inhibition of FeSO4-induced oxygen consumption [AID398696, Type: Literature]
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