Bookmark and Share
dazomet (CID 10788) - Compound BioActivity Data
.
BioActivity Outcomes:
Probe(1)
 
 
Active(269)
 
 
Inactive(973)
 
 
Inconclusive(125)
 
 
Unspecified(10)
 
 
Top Targets:
7tm 4(45)
 
 
 
NR LBD PPAR(30)
 
 
 
NR LBD ER(21)
 
 
 
NR LBD AR(18)
 
 
 
 
alkPPc(16)
 
 
BioAssay Types:
Screening(558)
 
 
 
 
 
Confirmatory(550)
 
 
 
 
 
Summary(49)
 
 
 
 
 
Literature(11)
 
 
BioActivity Types:
Potency(473)
 
 
 
 
 
IC50(53)
 
 
 
 
EC50(12)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 962    Data Row: 1378   Total Pages: 69   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID17389072]
Quantitative High-Throughput Screen for Epigenetic Modulators: Summary [AID1653, Type: summary]
View
2
[SID144208434]
Ratio Potency (uM) 0.37234qHTS assay for small molecule activators of the heat shock response signaling pathway: Summary [AID743228, Type: summary]heat shock protein beta-1 [Homo sapiens] [gi:4504517]
View
3
[SID144211307]
Ratio Potency (uM) 0.435398qHTS assay for small molecule activators of the heat shock response signaling pathway: Summary [AID743228, Type: summary]heat shock protein beta-1 [Homo sapiens] [gi:4504517]
View
4
[SID144211307]
Potency-Replicate_1 1.0937qHTS assay for small molecule activators of the heat shock response signaling pathway - cell viability counter screen [AID743209, Type: confirmatory]
View
5
[SID17389072]
Potency 1.5849qHTS for inhibitors of ROR gamma transcriptional activity [AID2551, Type: confirmatory]nuclear receptor ROR-gamma isoform 1 [Mus musculus] [gi:188536040]
View
6
[SID144208434]
Ratio Potency (uM) 1.72825qHTS assay to identify small molecule agonists of the glucocorticoid receptor (GR) signaling pathway: Summary [AID720719, Type: summary]glucocorticoid receptor [Homo sapiens] [gi:311348376]
View
7
[SID144208434]
Potency-Replicate_1 3.0482qHTS assay to identify small molecule antagonists of the thyroid receptor (TR) signaling pathway [AID743065, Type: confirmatory]thyroid hormone receptor beta isoform 2 [Rattus norvegicus] [gi:399498506]
View
8
[SID17389072]
Potency 3.1623VP16 counterscreen qHTS for inhibitors of ROR gamma transcriptional activity [AID2546, Type: confirmatory]nuclear receptor ROR-gamma isoform 1 [Mus musculus] [gi:188536040]
View
9
[SID144211307]
Potency-Replicate_1 3.4585qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway - cell viability counter screen [AID743033, Type: confirmatory]
View
10
[SID144211307]
Potency-Replicate_1 3.8453qHTS assay to identify aromatase inhibitors [AID743083, Type: confirmatory]cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a [Homo sapiens] [gi:119597822]
View
11
[SID144211307]
Potency-Replicate_1 3.8453qHTS assay to identify small molecule antagonists of the thyroid receptor (TR) signaling pathway [AID743065, Type: confirmatory]thyroid hormone receptor beta isoform 2 [Rattus norvegicus] [gi:399498506]
View
12
[SID144208434]
Potency-Replicate_1 3.8691qHTS assay to identify small molecule agonists of the peroxisome proliferator-activated receptor delta (PPARd) signaling pathway - cell viability counter screen [AID743211, Type: confirmatory]
View
13
[SID144211307]
Potency-Replicate_1 3.8805qHTS assay to identify small molecule agonists of the vitamin D receptor (VDR) signaling pathway - cell viability counter screen [AID743224, Type: confirmatory]
View
14
[SID7976210]
Potency 4.6109qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
View
15
[SID144208434]
AR Potency (uM) 4.83109qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line: Summary [AID743054, Type: summary]AR protein [Homo sapiens] [gi:124375976]
View
16
[SID144208434]
Potency-Replicate_1 4.8311qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743042, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
17
[SID144208434]
Potency-Replicate_1 4.8311qHTS assay to identify aromatase inhibitors [AID743083, Type: confirmatory]cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a [Homo sapiens] [gi:119597822]
View
18
[SID144211307]
Potency-Replicate_1 4.841qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rad54/Ku70 mutant cell line [AID743015, Type: confirmatory]
View
19
[SID144208434]
Potency-Replicate_1 4.8709qHTS assay to identify small molecule agonists of the farnesoid-X-receptor (FXR) signaling pathway - cell viability counter screen [AID743218, Type: confirmatory]
View
20
[SID144208434]
Potency-Replicate_1 5.4206qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rev3 mutant cell line [AID743014, Type: confirmatory]
View