omega-Chloroacetophenone (CID 10757) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(151)
 
 
Inactive(108)
 
 
Inconclusive(94)
 
 
Unspecified(11)
 
 
Top Targets:
NR LBD PPAR(10)
 
 
 
NR LBD TR(8)
 
 
 
NR LBD AR(4)
 
 
 
NR LBD ER(4)
 
 
 
NR LBD Fxr(4)
 
 
 
BioAssay Types:
Confirmatory(167)
 
 
 
 
Literature(9)
 
 
 
 
BioActivity Types:
Potency(131)
 
 
 
 
IC50(2)
 
 
EC50(1)
 
 
Ki(1)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 159    Data Row: 364   Total Pages: 8   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103321621]
EC50 0.03Agonist activity at human TRPA1 expressed in T-REx-HEK293 cells assessed as increase of intracellular calcium level by FDSS assay [AID516893, Type: Literature]Transient receptor potential cation channel subfamily A member 1 [gi:313104269]
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2
[SID103321621]
EC50 0.03Agonist activity at human TRPA1 expressed in T-REx-HEK293 cells assessed as increase of intracellular calcium level by FDSS assay [AID516893, Type: Literature]Transient receptor potential cation channel subfamily A member 1 [gi:313104269]
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3
[SID17389975]
Potency 0.0794qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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4
[SID17389975]
Potency 0.0794qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory]aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681]
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5
[SID17389975]
Potency 6.3096Cell Viability - LYMP2-022 [AID987, Type: confirmatory]
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6
[SID17389975]
Potency 7.9433Cell Viability - LYMP2-024 [AID988, Type: confirmatory]
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7
[SID17389975]
Potency 7.9433Cell Viability - LYMP2-010 [AID981, Type: confirmatory]
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8
[SID17389975]
Potency 7.9433Cell Viability - LYMP2-001 [AID921, Type: confirmatory]
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9
[SID17389975]
Potency 7.9433Cell Viability - LYMP2-015 [AID971, Type: confirmatory]
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10
[SID17389975]
Potency 7.9433Cell Viability - LYMP2-020 [AID986, Type: confirmatory]
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11
[SID17389975]
Potency 10Cell Viability - LYMP2-017 [AID972, Type: confirmatory]
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12
[SID17389975]
Potency 10Cell Viability - LYMP2-019 [AID973, Type: confirmatory]
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13
[SID17389975]
Potency 10Cell Viability - LYMP2-021 [AID974, Type: confirmatory]
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14
[SID17389975]
Potency 10Cell Viability - LYMP2-003 [AID965, Type: confirmatory]
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15
[SID17389975]
Potency 10Cell Viability - LYMP2-004 [AID966, Type: confirmatory]
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16
[SID17389975]
Potency 10Cell Viability - LYMP2-005 [AID967, Type: confirmatory]
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17
[SID17389975]
Potency 10Cell Viability - LYMP2-009 [AID968, Type: confirmatory]
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18
[SID17389975]
Potency 10Cell Viability - LYMP2-007 [AID979, Type: confirmatory]
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19
[SID17389975]
Potency 10Cell Viability - LYMP2-012 [AID982, Type: confirmatory]
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20
[SID17389975]
Potency 10Cell Viability - LYMP2-016 [AID984, Type: confirmatory]
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21
[SID17389975]
Potency 10Cell Viability - LYMP2-018 [AID985, Type: confirmatory]
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22
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-014 [AID983, Type: confirmatory]
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23
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-026 [AID989, Type: confirmatory]
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24
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-008 [AID980, Type: confirmatory]
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25
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-011 [AID969, Type: confirmatory]
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26
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-023 [AID975, Type: confirmatory]
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27
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-025 [AID976, Type: confirmatory]
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28
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-002 [AID977, Type: confirmatory]
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29
[SID17389975]
Potency 12.5893Cell Viability - LYMP2-006 [AID978, Type: confirmatory]
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30
[SID17389975]
Potency 12.5893qHTS Assay for Anthrax Lethal Toxin Internalization [AID912, Type: confirmatory]lethal factor [Bacillus anthracis str. A2012] [gi:21392848]
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31
[SID17389975]
Potency 15.8489Cell Viability - LYMP2-013 [AID970, Type: confirmatory]
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32
[SID17389975]
Potency 16.7855qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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33
[SID17389975]
Potency 16.7855qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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34
[SID17389975]
Potency 16.7855qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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35
[SID17389975]
Potency 16.7855qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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36
[SID17389975]
Potency 16.7855qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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37
[SID17389975]
Potency 25.1189MultiTox-Fluor Cytotoxicity Assay - LYMP1-002 - Dead Cells [AID960, Type: confirmatory]
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38
[SID17389975]
Potency 31.6228MultiTox-Fluor Cytotoxicity Assay - LYMP1-003 - Dead Cells [AID961, Type: confirmatory]
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39
[SID17389975]
Potency 31.6228MultiTox-Fluor Cytotoxicity Assay - LYMP1-002 - Live Cells [AID955, Type: confirmatory]
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40
[SID17389975]
Potency 35.4813qHTS assay for small molecule antagonists of vitamin D receptor signaling [AID588541, Type: confirmatory]vitamin D (1,25- dihydroxyvitamin D3) receptor [Homo sapiens] [gi:216409708]
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41
[SID17389975]
Potency 35.4813qHTS assay for small molecule antagonists of vitamin D receptor signaling [AID588541, Type: confirmatory]vitamin D (1,25- dihydroxyvitamin D3) receptor [Homo sapiens] [gi:216409708]
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42
[SID17389975]
Potency 35.4813qHTS assay for small molecule antagonists of vitamin D receptor signaling [AID588541, Type: confirmatory]vitamin D (1,25- dihydroxyvitamin D3) receptor [Homo sapiens] [gi:216409708]
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43
[SID17389975]
Potency 35.4813qHTS assay for small molecule antagonists of vitamin D receptor signaling [AID588541, Type: confirmatory]vitamin D (1,25- dihydroxyvitamin D3) receptor [Homo sapiens] [gi:216409708]
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44
[SID17389975]
Potency 39.8107qHTS assay for small molecule antagonists of glucocorticoid receptor signaling [AID588533, Type: confirmatory]glucocorticoid receptor [Homo sapiens] [gi:311348376]
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45
[SID17389975]
Potency 39.8107qHTS assay for small molecule antagonists of glucocorticoid receptor signaling [AID588533, Type: confirmatory]glucocorticoid receptor [Homo sapiens] [gi:311348376]
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46
[SID17389975]
Potency 39.8107qHTS assay for small molecule antagonists of glucocorticoid receptor signaling [AID588533, Type: confirmatory]glucocorticoid receptor [Homo sapiens] [gi:311348376]
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47
[SID17389975]
Potency 39.8107qHTS assay for small molecule antagonists of glucocorticoid receptor signaling [AID588533, Type: confirmatory]glucocorticoid receptor [Homo sapiens] [gi:311348376]
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48
[SID17389975]
Potency 39.8107MultiTox-Fluor Cytotoxicity Assay - LYMP1-003 - Live Cells [AID962, Type: confirmatory]
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49
[SID17389975]
Potency 50.1187MultiTox-Fluor Cytotoxicity Assay - LYMP1-001 - Dead Cells [AID946, Type: confirmatory]
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50
[SID26752938]
Potency 61.1306qHTS assay for small molecule agonists of the antioxidant response element (ARE) signaling pathway [AID651741, Type: confirmatory]NFE2L2 gene product [Homo sapiens] [gi:20149576]
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