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olivetol (CID 10377) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(25)
 
 
Inactive(245)
 
 
Inconclusive(61)
 
 
Unspecified(13)
 
 
Top Targets:
NR LBD PPAR(21)
 
 
 
 
NR LBD ER(16)
 
 
 
 
NR LBD AR(16)
 
 
 
 
NR LBD VDR(10)
 
 
 
NR LBD TR(10)
 
 
 
BioAssay Types:
Confirmatory(274)
 
 
 
 
Summary(48)
 
 
 
 
Literature(13)
 
 
 
BioActivity Types:
Potency(273)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 247    Data Row: 344   Total Pages: 7   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144213649]
Potency-Replicate_1 7.6959qHTS assay for small molecule disruptors of the mitochondrial membrane potential [AID720635, Type: confirmatory]
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2
[SID144209547]
Potency-Replicate_1 9.728qHTS assay for small molecule disruptors of the mitochondrial membrane potential [AID720635, Type: confirmatory]
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3
[SID17388829]
Potency 12.5893qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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4
[SID144213649]
Ratio Potency (uM) 14.7772qHTS assay for small molecule disruptors of the mitochondrial membrane potential: Summary [AID720637, Type: summary]
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5
[SID144213649]
AhR Potency (uM) 17.2289qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway: Summary [AID743122, Type: summary]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
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6
[SID144213649]
Potency-Replicate_1 21.8751qHTS assay to identify small molecule antagonists of the peroxisome proliferator-activated receptor gamma (PPARg) signaling pathway [AID743191, Type: confirmatory]peroxisome proliferator activated receptor gamma [Homo sapiens] [gi:216409692]
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7
[SID144209547]
Potency-Replicate_1 24.6584qHTS assay to identify small molecule antagonists of the peroxisome proliferator-activated receptor gamma (PPARg) signaling pathway [AID743191, Type: confirmatory]peroxisome proliferator activated receptor gamma [Homo sapiens] [gi:216409692]
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8
[SID144209547]
Potency-Replicate_1 24.6584qHTS assay to identify small molecule antagonists of the estrogen receptor alpha (ER-alpha) signaling pathway [AID743069, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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9
[SID144209547]
Ratio Potency (uM) 34.8309qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway: Summary [AID743063, Type: summary]AR protein [Homo sapiens] [gi:124375976]
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10
[SID17388829]
Potency 37.578qHTS assay for small molecule disruptors of the mitochondrial membrane potential - 1 hr assay [AID651754, Type: confirmatory]
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11
[SID17388829]
Potency 37.578qHTS assay for small molecule disruptors of the mitochondrial membrane potential - 5 hr assay [AID651755, Type: confirmatory]
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12
[SID17388829]
Potency 42.1632qHTS assay for small molecule agonists of the antioxidant response element (ARE) signaling pathway [AID651741, Type: confirmatory]nuclear factor erythroid 2-related factor 2 isoform 1 [Homo sapiens] [gi:20149576]
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13
[SID144213649]
Ratio Potency (uM) 46.2327qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway: Summary [AID743063, Type: summary]AR protein [Homo sapiens] [gi:124375976]
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14
[SID144213649]
Potency-Replicate_1 48.5577qHTS assay for small molecule agonists of the antioxidant response element (ARE) signaling pathway [AID743202, Type: confirmatory]nuclear factor erythroid 2-related factor 2 isoform 1 [Homo sapiens] [gi:20149576]
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15
[SID144209547]
Potency-Replicate_1 48.7553qHTS assay for small molecule agonists of the antioxidant response element (ARE) signaling pathway [AID743202, Type: confirmatory]nuclear factor erythroid 2-related factor 2 isoform 1 [Homo sapiens] [gi:20149576]
View
16
[SID144209547]
Potency-Replicate_1 49.2qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway [AID720692, Type: confirmatory]glucocorticoid receptor [Homo sapiens] [gi:311348376]
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17
[SID144213649]
Potency-Replicate_1 54.4827qHTS assay for small molecules that induce genotoxicity in human embryonic kidney cells expressing luciferase-tagged ATAD5 - cell viability [AID651634, Type: confirmatory]
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18
[SID144209547]
Ratio Potency (uM) 54.7044qHTS assay for small molecule agonists of the antioxidant response element (ARE) signaling pathway: Summary [AID743219, Type: summary]nuclear factor erythroid 2-related factor 2 isoform 1 [Homo sapiens] [gi:20149576]
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19
[SID144209547]
Ratio Potency (uM) 59.6071qHTS assay to identify small molecule antagonists of the estrogen receptor alpha (ER-alpha) signaling pathway: Summary [AID743078, Type: summary]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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20
[SID144213649]
Potency-Replicate_1 61.1306qHTS assay for small molecule disruptors of the mitochondrial membrane potential - cell viability [AID720634, Type: confirmatory]
View
21
[SID144209547]
Potency-Replicate_1 61.3793qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway [AID743085, Type: confirmatory]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
View
22
[SID144209547]
AhR Potency (uM) 61.3793qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway: Summary [AID743122, Type: summary]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
View
23
[SID144213649]
qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway: Summary [AID720725, Type: summary]glucocorticoid receptor [Homo sapiens] [gi:311348376]
View
24
[SID144209547]
qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway: Summary [AID720725, Type: summary]glucocorticoid receptor [Homo sapiens] [gi:311348376]
View
25
[SID144209547]
qHTS assay to identify small molecule antagonists of the peroxisome proliferator-activated receptor gamma (PPARg) signaling pathway: Summary [AID743199, Type: summary]peroxisome proliferator activated receptor gamma [Homo sapiens] [gi:216409692]
View
26
[SID103404661]
Km 520Activity for Streptomyces coelicolor A3(2) prenyltransferase assessed as formation of 2-(3,7-dimethylocta-2,6-dienyl)-5-pentylbenzene-1,3-diol [AID365324, Type: Literature]Hypothetical protein SCO7190 [gi:81539207]
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27
[SID103404661]
Km 640Activity for Streptomyces coelicolor A3(2) prenyltransferase assessed as formation of 4-(3,7-dimethylocta-2,6-dienyl)-5-pentylbenzene-1,3-diol [AID365151, Type: Literature]Hypothetical protein SCO7190 [gi:81539207]
View
28
[SID103404661]
Ratio of Kcat to Km of Streptomyces coelicolor A3(2) prenyltransferase assessed as formation of 4-(3,7-dimethylocta-2,6-dienyl)-5-pentylbenzene-1,3-diol [AID365336, Type: Literature]Hypothetical protein SCO7190 [gi:81539207]
View
29
[SID103404661]
Ratio of Kcat to Km of Streptomyces coelicolor A3(2) prenyltransferase assessed as formation of 2-(3,7-dimethylocta-2,6-dienyl)-5-pentylbenzene-1,3-diol [AID365337, Type: Literature]Hypothetical protein SCO7190 [gi:81539207]
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30
[SID17388829]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838, Type: other]
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31
[SID103404661]
Capability to induce convulsions in tetrahydrocannabinol-seizure susceptible (THC-SS) rabbit [AID165405, Type: Literature]
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32
[SID103404661]
Number of rabbits convulsed at 20 mg/kg, iv out of 4 rabbits tested [AID167516, Type: Literature]
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33
[SID103404661]
Antibacterial activity against methicillin-resistant Staphylococcus aureus SA1199B after 18 hrs [AID362541, Type: Literature]
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34
[SID103404661]
Antibacterial activity against macrolide-resistant Staphylococcus aureus RN4220 after 18 hrs [AID362542, Type: Literature]
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35
[SID103404661]
Antibacterial activity against tetracycline-resistant Staphylococcus aureus XU212 after 18 hrs [AID362543, Type: Literature]
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36
[SID103404661]
Antibacterial activity against methicillin-resistant Staphylococcus aureus ATCC 25923 after 18 hrs [AID362544, Type: Literature]
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37
[SID103404661]
Antibacterial activity against epidemic methicillin-resistant Staphylococcus aureus 15 after 18 hrs [AID362545, Type: Literature]
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38
[SID103404661]
Antibacterial activity against epidemic methicillin-resistant Staphylococcus aureus 16 after 18 hrs [AID362546, Type: Literature]
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39
[SID144209547]
Potency-Replicate_1 12.2468qHTS assay to identify aromatase inhibitors [AID743083, Type: confirmatory]cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a [Homo sapiens] [gi:119597822]
View
40
[SID17388829]
Potency 12.5893qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
View
41
[SID144213649]
Potency-Replicate_1 21.8751qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway [AID743075, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View
42
[SID17388829]
Potency 26.6032qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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43
[SID144209547]
Potency-Replicate_1 77.272qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line [AID743079, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View
44
[SID144209547]
Potency-Replicate_1 qHTS assay to identify small molecule antagonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line [AID743080, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View
45
[SID144209547]
ER Potency (uM) qHTS assay to identify small molecule antagonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line: Summary [AID743091, Type: summary]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View
46
[SID144209547]
Potency-Replicate_1 qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway [AID743075, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View
47
[SID144209547]
Ratio Potency (uM) qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway: Summary [AID743077, Type: summary]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View
48
[SID144213649]
Ratio Potency (uM) qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway: Summary [AID743077, Type: summary]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View
49
[SID144213649]
Potency-Replicate_1 qHTS assay to identify small molecule agonists of the thyroid receptor (TR) signaling pathway [AID743066, Type: confirmatory]thyroid hormone receptor beta isoform 2 [Rattus norvegicus] [gi:399498506]
View
50
[SID144213649]
Potency-Replicate_1 qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line [AID743079, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
View