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Epitestosterone (CID 10204) - Compound BioActivity Data
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BioActivity Outcomes:
Active(10)
 
 
Inactive(68)
 
 
Inconclusive(18)
 
 
Unspecified(9)
 
 
Top Targets:
NR LBD AR(7)
 
 
 
 
NR LBD ER(7)
 
 
 
GT1 Gtf like(7)
 
 
NR LBD GR(4)
 
 
 
P53(4)
 
 
BioAssay Types:
Confirmatory(60)
 
 
 
 
Summary(15)
 
 
 
 
Screening(12)
 
 
Literature(9)
 
 
 
BioActivity Types:
Potency(73)
 
 
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 96    Data Row: 105   Total Pages: 6   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144204609]
Potency-Replicate_1 0.0008qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743040, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
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2
[SID144204609]
Ratio Potency (uM) 0.00189959qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway: Summary [AID743053, Type: summary]AR protein [Homo sapiens] [gi:124375976]
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3
[SID144204609]
Potency-Replicate_1 0.0021qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway [AID743036, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
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4
[SID144204609]
Potency-Replicate_1 0.0047qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line [AID743079, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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5
[SID103469411]
IC50 0.01585Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881) [AID255211, Type: Literature]
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6
[SID144204609]
Potency-Replicate_1 4.2527qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway [AID720692, Type: confirmatory]glucocorticoid receptor [Homo sapiens] [gi:311348376]
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7
[SID144204609]
Potency-Replicate_1 6.007qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway [AID743075, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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8
[SID144204609]
Ratio Potency (uM) 9.15311qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway: Summary [AID743077, Type: summary]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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9
[SID144204609]
Potency-Replicate_1 23.7101qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - wild type cell line [AID743012, Type: confirmatory]
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10
[SID144204609]
Potency-Replicate_1 29.8493qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rad54/Ku70 mutant cell line [AID743015, Type: confirmatory]
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11
[SID103469411]
Inhibition of mouse constitutive androstane receptor (mCAR) activity at 10 uM was determined as percent remaining activity [AID50906, Type: Literature]
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12
[SID144204609]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838, Type: other]
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13
[SID103469411]
Specific activity of expressed human recombinant UGT2B7H [AID624620, Type: Literature]UDP-glucuronosyltransferase 2B7 [gi:136727]
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14
[SID103469411]
Specific activity of expressed human recombinant UGT2B7Y [AID624621, Type: Literature]UDP-glucuronosyltransferase 2B7 [gi:136727]
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15
[SID103469411]
Specific activity of expressed human recombinant UGT1A1 [AID624606, Type: Literature]UDP-glucuronosyltransferase 1-1 [gi:136729]
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16
[SID103469411]
Specific activity of expressed human recombinant UGT1A4 [AID624608, Type: Literature]UDP-glucuronosyltransferase 1-4 [gi:136731]
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17
[SID103469411]
Specific activity of expressed human recombinant UGT1A10 [AID624613, Type: Literature]UDP-glucuronosyltransferase 1-10 [gi:29839636]
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18
[SID103469411]
Specific activity of expressed human recombinant UGT1A8 [AID624611, Type: Literature]UDP-glucuronosyltransferase 1-8 [gi:29839637]
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19
[SID103469411]
Specific activity of expressed human recombinant UGT2B15 [AID624616, Type: Literature]UDP-glucuronosyltransferase 2B15 [gi:332278237]
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20
[SID144204609]
Potency-Replicate_1 qHTS assay for small molecule activators of the human pregnane X receptor (PXR) signaling pathway [AID720659, Type: confirmatory]pregnane X nuclear receptor [Homo sapiens] [gi:325495557]
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