CHEMBL558625
(CID
10047593
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(
2
)
Top Targets:
SK channel(
2
)
BioAssay Types:
Literature(
2
)
BioActivity Types:
IC50(
1
)
Ki(
1
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 2 Data Row: 2 Total Pages: 1
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
103680210
]
Active
Ki
4.4
Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cells [AID
346945
, Type: Literature]
Small conductance calcium-activated potassium channel protein 3 [gi:
17365967
]
View
X
Row No.
1
Structure
Substance
SID
103680210
CID
10047593
Outcome
Active
Ki
4.4 [uM]
BioAssay
Displacement of [I125]apamine from Wistar rat recombinant SK3 channel expressed in HEK293 cells
AID
346945
BioAssay type
Literature
Target
Small conductance calcium-activated potassium channel protein 3 [gi:
17365967
]
PubMed
18998663
Data Table
2
[SID
103680210
]
Active
IC50
7
Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp technique [AID
346946
, Type: Literature]
Small conductance calcium-activated potassium channel protein 3 [gi:
17365967
]
View
X
Row No.
2
Structure
Substance
SID
103680210
CID
10047593
Outcome
Active
IC50
7 [uM]
BioAssay
Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp technique
AID
346946
BioAssay type
Literature
Target
Small conductance calcium-activated potassium channel protein 3 [gi:
17365967
]
PubMed
18998663
Data Table
Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
