CHEMBL1627207
(CID
10006229
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(
2
)
Top Targets:
p450(
2
)
BioAssay Types:
Literature(
2
)
BioActivity Types:
IC50(
2
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 1 Data Row: 2 Total Pages: 1
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
160681377
]
Active
IC50
0.028
Inhibition of human CYP24 hydroxylase expressed in V79 cells [AID
282480
, Type: Literature]
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial [gi:
19862747
]
View
X
Row No.
1
Structure
Substance
SID
160681377
CID
10006229
Outcome
Active
IC50
0.028 [uM]
BioAssay
Inhibition of human CYP24 hydroxylase expressed in V79 cells
AID
282480
BioAssay type
Literature
Target
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial [gi:
19862747
]
PubMed
15615534
Data Table
2
[SID
160686734
]
Active
IC50
0.044
Inhibition of human CYP24 hydroxylase expressed in V79 cells [AID
282480
, Type: Literature]
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial [gi:
19862747
]
View
X
Row No.
2
Structure
Substance
SID
160686734
CID
10006229
Outcome
Active
IC50
0.044 [uM]
BioAssay
Inhibition of human CYP24 hydroxylase expressed in V79 cells
AID
282480
BioAssay type
Literature
Target
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial [gi:
19862747
]
PubMed
15615534
Data Table
Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
