GSK_PKIS: P38alpha mean inhibition at 1 uM [Nanosyn] - BioAssay Summary
GSK_PKIS: P38alpha mean inhibition at 1 uM [Nanosyn] ..more
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 Tested Compounds
 Tested Compounds
All(366)
 
 
Unspecified(366)
 
 
 Tested Substances
 Tested Substances
All(366)
 
 
Unspecified(366)
 
 
AID: 651203
Data Source: ChEMBL (808651)
Depositor Category: Other
BioAssay Version:
Deposit Date: 2012-09-09
Modify Date: 2013-05-16

Data Table (Complete):           All
Target
Sequence: RecName: Full=Mitogen-activated protein kinase 14; Short=MAP kinase 14; Short=MAPK 14; AltName: Full=Cytokine suppressive anti-inflammatory drug-binding protein; Short=CSAID-binding protein; Short=CSBP; AltName: Full=MAP kinase MXI2; AltName: Full=MAX-interacting protein 2; AltName: Full=Mitogen-activated protein kinase p38 alpha; Short=MAP kinase p38 alpha; AltName: Full=Stress-activated protein kinase 2a; Short=SAPK2a
Description ..   
Protein Family: Catalytic domain of the Serine/Threonine Kinase, p38 Mitogen-Activated Protein Kinase
Comment ..   

Gene:MAPK14     Related Protein 3D Structures
Tested Compounds:
Description:
GSK_PKIS: P38alpha mean inhibition at 1 uM [Nanosyn]
Comment


Publication:
Journal: NULL
Year: NULL
Volume: NULL
Issue: NULL
First Page: NULL
Last Page: NULL
Categorized Comment
ChEMBL Assay Type: Binding

ChEMBL Assay Data Source: GSK Published Kinase Inhibitor Set

ChEMBL Assay Test Type: In vitro

ChEMBL Target ID: 10188

ChEMBL target type: Target is a single protein chain

Result Definitions
TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1Inhibition activity commentInhibition activity commentString
2Inhibition standard flagInhibition standard flagInteger
3Inhibition qualifierInhibition qualifierString
4Inhibition published valueInhibition published valueFloat%
5Inhibition standard valueInhibition standard valueFloat%
6Inhibition data validityInhibition data validityString

Data Table (Concise)
Classification
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