GSK_PKIS: PAR-1Balpha mean inhibition at 1 uM [Nanosyn] - BioAssay Summary
GSK_PKIS: PAR-1Balpha mean inhibition at 1 uM [Nanosyn] ..more
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 Tested Compounds
 Tested Compounds
All(368)
 
 
Unspecified(368)
 
 
 Tested Substances
 Tested Substances
All(368)
 
 
Unspecified(368)
 
 
AID: 651129
Data Source: ChEMBL (808577)
Depositor Category: Other
BioAssay Version:
Deposit Date: 2012-09-09
Modify Date: 2013-05-16

Data Table (Complete):           All
Target
Sequence: RecName: Full=Serine/threonine-protein kinase MARK2; AltName: Full=ELKL motif kinase 1; Short=EMK-1; AltName: Full=MAP/microtubule affinity-regulating kinase 2; AltName: Full=PAR1 homolog; AltName: Full=PAR1 homolog b; Short=Par-1b; Short=Par1b
Description ..   
Protein Family: Catalytic domain of AGC family Protein Serine/Threonine Kinases
Comment ..   

Gene:MARK2     Related Protein 3D Structures
Tested Compounds:
Description:
GSK_PKIS: PAR-1Balpha mean inhibition at 1 uM [Nanosyn]
Comment


Publication:
Journal: NULL
Year: NULL
Volume: NULL
Issue: NULL
First Page: NULL
Last Page: NULL
Categorized Comment
ChEMBL Assay Type: Binding

ChEMBL Assay Data Source: GSK Published Kinase Inhibitor Set

ChEMBL Assay Test Type: In vitro

ChEMBL Target ID: 30001

ChEMBL target type: Target is a single protein chain

Result Definitions
TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1Inhibition activity commentInhibition activity commentString
2Inhibition standard flagInhibition standard flagInteger
3Inhibition qualifierInhibition qualifierString
4Inhibition published valueInhibition published valueFloat%
5Inhibition standard valueInhibition standard valueFloat%

Data Table (Concise)
Classification
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