DRUGMATRIX: GABAA, Flunitrazepam, Central radioligand binding (ligand: [3H] Flunitrazepam) - BioAssay Summary
DRUGMATRIX: GABAA, Flunitrazepam, Central radioligand binding (ligand: [3H] Flunitrazepam) ..more
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 Tested Compounds
 Tested Compounds
All(857)
 
 
Active(16)
 
 
Unspecified(841)
 
 
 Tested Substances
 Tested Substances
All(870)
 
 
Active(16)
 
 
Unspecified(854)
 
 
 Related BioAssays
 Related BioAssays
Table of Contents
AID: 625261
Data Source: ChEMBL (774759)
Depositor Category: Other
BioAssay Version:
Deposit Date: 2012-09-09
Modify Date: 2013-05-15

Data Table (Complete):           Active    All
BioActive Compounds: 16
Description:
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DRUGMATRIX: GABAA, Flunitrazepam, Central radioligand binding (ligand: [3H] Flunitrazepam)
Comment
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Compounds with activity <= 50uM or explicitly reported as active by ChEMBL are flagged as active in this PubChem assay presentation.

Putative Target:

ChEMBL Target ID: 22226
Target Type: UNCHECKED
Pref Name: Unchecked
Confidence: Default value - Target unknown or has yet to be assigned
Relationship Type: Default value - Target has yet to be curated


Publication:
Journal: NULL
Year: NULL
Volume: NULL
Issue: NULL
First Page: NULL
Last Page: NULL
Categorized Comment
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ChEMBL Assay Type: Binding

ChEMBL Assay Data Source: DrugMatrix in vitro pharmacology assays

ChEMBL Assay Test Type: In vitro

ChEMBL Assay Tissue: Brain (except cerebellum)

ChEMBL Assay Subcellular Fraction: membranes

Result Definitions
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TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1IC50*IC50 PubChem standard valueFloatμM
2IC50 activity commentIC50 activity commentString
3IC50 standard flagIC50 standard flagInteger
4IC50 qualifierIC50 qualifierString
5IC50 published valueIC50 published valueFloatnM
6IC50 standard valueIC50 standard valueFloatnM
7Ki activity commentKi activity commentString
8Ki standard flagKi standard flagInteger
9Ki qualifierKi qualifierString
10Ki published valueKi published valueFloatnM
11Ki standard valueKi standard valueFloatnM
* Activity Concentration.

Data Table (Concise)
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