GRAC: human GAL2 selective antagonist - BioAssay Summary
Title: Guide to Receptors and Channels (GRAC), 4th Edition.
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 Tested Substances
 Tested Substances
All(1)
 
 
Unspecified(1)
 
 
AID: 540635
Data Source: ChEMBL (689145)
Depositor Category: Other
BioAssay Version:
Deposit Date: 2011-09-18
Modify Date: 2013-05-13

Data Table (Complete):           All
Target
Sequence: RecName: Full=Galanin receptor type 2; Short=GAL2-R; Short=GALR-2
Description ..   
Protein Family: Serpentine type 7TM GPCR chemoreceptor Srw
Comment ..   

Gene:GALR2     Related Protein 3D Structures
Description:
Title: Guide to Receptors and Channels (GRAC), 4th Edition.
Categorized Comment
ChEMBL Assay Type: Binding

ChEMBL Assay Data Source: Guide to Receptors and Channels

ChEMBL Target ID: 11498

ChEMBL target type: Target is a single protein chain

Result Definitions
TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1Ki*Ki PubChem standard valueFloatμM
2Ki activity commentKi activity commentString
3Ki standard flagKi standard flagInteger
4Ki qualifierKi qualifierString
5Ki published valueKi published valueFloatnM
6Ki standard valueKi standard valueFloatnM

* Activity Concentration.

Data Table (Concise)
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