Bookmark and Share
BioAssay: AID 540551

GRAC: human TRPM4 blocker

Title: Guide to Receptors and Channels (GRAC), 4th Edition.
..more
_
   
 Tested Compounds
 Tested Compounds
All(6)
 
 
Unspecified(6)
 
 
 Tested Substances
 Tested Substances
All(7)
 
 
Unspecified(7)
 
 
 Related BioAssays
 Related BioAssays
AID: 540551
Data Source: ChEMBL (689061)
Depositor Category: Other
BioAssay Version:
Deposit Date: 2011-09-18
Modify Date: 2013-11-17

Data Table ( Complete ):           All
Target
Sequence: RecName: Full=Transient receptor potential cation channel subfamily M member 4; Short=hTRPM4; AltName: Full=Calcium-activated non-selective cation channel 1; AltName: Full=Long transient receptor potential channel 4; Short=LTrpC-4; Short=LTrpC4; AltName: Full=Melastatin-4
Description ..   
Protein Family: Acetyl co-enzyme A carboxylase carboxyltransferase alpha subunit
Comment ..   

Gene:TRPM4          More BioActivity Data..
Tested Compounds:
Description:
Title: Guide to Receptors and Channels (GRAC), 4th Edition.
Categorized Comment
ChEMBL Assay Type: Binding

ChEMBL Assay Data Source: Guide to Receptors and Channels

ChEMBL Target ID: 103788

ChEMBL Target Type: Target is a single protein chain

Result Definitions
Show more
TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1IC50*IC50 PubChem standard valueFloatμM
2BEIBinding Efficiency Index(nM)Float
3SEISurface Efficiency Index(nM)Float
4LELigand EfficiencyFloat
5LLELipophilic Ligand EfficiencyFloat
6IC50 activity commentIC50 activity commentString
7IC50 standard flagIC50 standard flagInteger
8IC50 qualifierIC50 qualifierString
9IC50 published valueIC50 published valueFloatμM
10IC50 standard valueIC50 standard valueFloatnM
11IC50 data validityIC50 data validityString
12IC50 binding domainsIC50 binding domainsString

* Activity Concentration.

Data Table (Concise)
Classification
PageFrom: