Inhibition of human recombinant p21RAS by GDPX assay - BioAssay Summary
Inhibition of human recombinant p21RAS by GDPX assay ..more
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 Tested Compounds
 Tested Compounds
All(2)
 
 
Inconclusive(1)
 
 
Unspecified(1)
 
 
 Tested Substances
 Tested Substances
All(2)
 
 
Inconclusive(1)
 
 
Unspecified(1)
 
 
AID: 338280
Data Source: ChEMBL (486309)
Depositor Category: Literature, Extracted
BioAssay Version:
Deposit Date: 2010-05-25
Modify Date: 2013-05-07

Data Table (Complete):           All
Target
Sequence: RecName: Full=GTPase HRas; AltName: Full=H-Ras-1; AltName: Full=Ha-Ras; AltName: Full=Transforming protein p21; AltName: Full=c-H-ras; AltName: Full=p21ras; Contains: RecName: Full=GTPase HRas, N-terminally processed; Flags: Precursor
Description ..   
Protein Family: Ras GTPase family containing H-Ras,N-Ras and K-Ras4A/4B
Comment ..   

Gene:HRAS     Related Protein 3D Structures
Tested Compounds:
Description:
Inhibition of human recombinant p21RAS by GDPX assay
Comment


Publication:
Journal: J. Nat. Prod.
Year: 1994
Volume: 57
Issue: 12
First Page: 1751
Last Page: 1754
Categorized Comment
ChEMBL Assay Type: Binding

ChEMBL Assay Data Source: Scientific Literature

ChEMBL Target ID: 10093

ChEMBL target type: Target is a single protein chain

Result Definitions
TIDNameDescriptionHistogramTypeUnit
OutcomeThe BioAssay activity outcomeOutcome
1IC50 activity commentIC50 activity commentString
2IC50 standard flagIC50 standard flagInteger
3IC50 qualifierIC50 qualifierString
4IC50 published valueIC50 published valueFloatug.mL-1
5IC50 standard valueIC50 standard valueFloatug.mL-1

Data Table (Concise)
Classification
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